Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC10595threo Ifenprodil hemitartrateCAS: 1312991-83-5
σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist
- GC107817-Chlorokynurenic acidCAS: 18000-24-3纯度: >99.50%
A glycine-site selective NMDA receptor antagonist
- GC10792Co 101244 hydrochlorideCAS: 193356-17-1
Co 101244 (PD 174494) hydrochloride 是一种含有 NR2B 的 NMDA 受体拮抗剂。
- GC10835Nitrobenzylthioinosine (NBMPR)CAS: 38048-32-7纯度: >99.00%
Nitrobenzylthioinosine (NBMPR)是一种平衡型核苷转运子亚型1(ENT1)转运蛋白抑制剂,以高亲和力与ENT1转运蛋白结合。
- GC10856THIP hydrochlorideCAS: 85118-33-8纯度: >99.00%
A GABA A receptor agonist and GABA C receptor antagonist
- GC10861Domiphen BromideCAS: 538-71-6纯度: >99.00%
A quaternary ammonium compound and cationic surfactant with antimicrobial activity
- GC108985-(N,N-dimethyl)-Amiloride (hydrochloride)CAS: 2235-97-4纯度: >98.00%
An inhibitor of Na + /H + exchangers
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10595 | threo Ifenprodil hemitartrate | 1312991-83-5 | - | |
σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist | ||||
| GC10641 | AA 29504 | 945828-50-2 | - | |
GABAA receptor modulator | ||||
| GC10669 | pep2-EVKI | 1315378-67-6 | - | |
选择性破坏 GluR2 亚基(在 C 末端 PDZ 位点)与 PICK1 结合的抑制肽 | ||||
| GC10678 | Nicardipine HCl | 54527-84-3 | >99.50% | |
An L-type calcium channel blocker | ||||
| GC10688 | MNI-caged-D-aspartate | 845555-94-4 | - | |
Agonist at NMDA receptors and EAAT substrate | ||||
| GC10696 | L-689,560 | 139051-78-8 | >99.00% | |
L-689,560 是一种有效的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂,作用于 GluN1 甘氨酸结合位点。 | ||||
| GC10741 | TCS 1205 | 355022-97-8 | - | |
TCS 1205 (compound 2b) 是一种有效的选择性 GABAA 激动剂。 | ||||
| GC10781 | 7-Chlorokynurenic acid | 18000-24-3 | >99.50% | |
A glycine-site selective NMDA receptor antagonist | ||||
| GC10786 | DHBP dibromide | 6159-05-3 | >99.50% | |
DHBP 二溴化物是一种钙释放抑制剂和一种肌肉松弛剂。 | ||||
| GC10792 | Co 101244 hydrochloride | 193356-17-1 | - | |
Co 101244 (PD 174494) hydrochloride 是一种含有 NR2B 的 NMDA 受体拮抗剂。 | ||||
| GC10823 | YM 244769 | 837424-39-2 | - | |
YM 244769 是一种有效的、选择性的和具有口服活性的 Na+/Ca2+ 交换剂 (NCX) 抑制剂。 | ||||
| GC10830 | GS967 | 1262618-39-2 | >99.50% | |
GS967是一种强效、选择性的晚期钠电流抑制剂,在心室肌细胞和离体心脏中的IC 50 值分别为0.13μM和0.21μM。 | ||||
| GC10835 | Nitrobenzylthioinosine (NBMPR) | 38048-32-7 | >99.00% | |
Nitrobenzylthioinosine (NBMPR)是一种平衡型核苷转运子亚型1(ENT1)转运蛋白抑制剂,以高亲和力与ENT1转运蛋白结合。 | ||||
| GC10836 | Jingzhaotoxin III | 925463-91-8 | - | |
NaV1.5 channels blocker | ||||
| GC10844 | SCS | 3232-36-8 | - | |
GABAA receptor antagonist | ||||
| GC10856 | THIP hydrochloride | 85118-33-8 | >99.00% | |
A GABA A receptor agonist and GABA C receptor antagonist | ||||
| GC10861 | Domiphen Bromide | 538-71-6 | >99.00% | |
A quaternary ammonium compound and cationic surfactant with antimicrobial activity | ||||
| GC10866 | Spermidine trihydrochloride | 334-50-9 | >99.00% | |
An endogenous polyamine | ||||
| GC10873 | α-Spinasterol | 481-18-5 | >99.00% | |
A TRPV1 antagonist | ||||
| GC10874 | Fumitremorgin C | 118974-02-0 | >98.00% | |
Inhibitor of BCRP multidrug transporter | ||||
| GC10875 | LDN 212320 | 894002-50-7 | >98.00% | |
An activator of EAAT2 | ||||
| GC10877 | CHC | 28166-41-8 | >98.00% | |
An MCT1 inhibitor | ||||
| GC10888 | SCH 50911 | 733717-87-8 | - | |
SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-乙酸,一种选择性、口服活性和竞争性 γ-氨基丁酸 B GABA(B) 受体拮抗剂,与 GABA(B ) 受体,IC50 为 1.1 μM。 | ||||
| GC10898 | 5-(N,N-dimethyl)-Amiloride (hydrochloride) | 2235-97-4 | >98.00% | |
An inhibitor of Na + /H + exchangers | ||||
