Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC10519Ethacrynic acid - d5CAS: 1330052-59-9
An internal standard for the quantification of ethacrynic acid
- GC10530Dihydroergotoxine mesylateCAS: 8067-24-1纯度: >98.00%
A mixture of alkaloids with diverse biological activities
- GC10574Norketamine hydrochlorideCAS: 79499-59-5纯度: >98.00%
Major metabolite of ketamine, NMDA receptor antagonist
- GC10579Ouabain OctahydrateCAS: 11018-89-6纯度: >99.50%
Ouabain Octahydrate是一种Na + /K + -ATPase抑制剂,能够用于研究充血性心力衰竭。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10371 | PSB 06126 | 1052089-16-3 | >98.00% | |
PSB 06126 是一种选择性三磷酸核苷二磷酸水解酶 (NTPDase) 抑制剂,对大鼠 NTPDase 1 的 Ki 值分别为 0.33 μM,对 NTPDase 2 和 NTPDase 3 的 Ki 值分别为 19.1 μM 和 2.22 μM。 | ||||
| GC10391 | Hypophyllanthin | 33676-00-5 | >98.00% | |
A P-glycoprotein inhibitor | ||||
| GC10392 | 9-AC | 723-62-6 | - | |
A chloride channel inhibitor | ||||
| GC10395 | Dynasore | 304448-55-3 | >98.50% / >98.00% | |
Dynasore 作为 GTPase 抑制剂,可以快速、可逆地抑制发动蛋白活性,从而阻止内吞作用。 | ||||
| GC10411 | MRS 2219 | 14141-47-0 | - | |
P2X1 receptor potentiator | ||||
| GC10443 | Meclofenoxate hydrochloride | 3685-84-5 | >98.00% | |
A nootropic agent | ||||
| GC10444 | PF-03716556 | 928774-43-0 | - | |
A potent and selective H + /K + -ATPase inhibitor | ||||
| GC10458 | Penfluridol | 26864-56-2 | >99.50% | |
A typical antipsychotic | ||||
| GC10471 | Ifenprodil hemitartrate | 23210-58-4 | >99.50% | |
An NMDA receptor antagonist | ||||
| GC10476 | (RS)-CPP | 100828-16-8 | - | |
NMDA antagonist | ||||
| GC10489 | CGP 54626 hydrochloride | 149184-21-4 | ≥95.00% | |
A selective GABA B receptor antagonist | ||||
| GC10492 | ML 277 | 1401242-74-7 | >99.00% | |
An activator of KCNQ1 | ||||
| GC10497 | Hexachlorophene | 70-30-4 | - | |
KCNQ1/KCNE1 potassium channel activator | ||||
| GC10498 | LOE 908 hydrochloride | 143482-60-4 | - | |
广谱阳离子通道阻断剂 | ||||
| GC10506 | FPL 64176 | 120934-96-5 | >98.50% | |
An L-type Ca 2+ channel agonist | ||||
| GC10515 | Tertiapin-Q | 252198-49-5 | >99.50% | |
A peptide derivative of tertiapin | ||||
| GC10519 | Ethacrynic acid - d5 | 1330052-59-9 | - | |
An internal standard for the quantification of ethacrynic acid | ||||
| GC10530 | Dihydroergotoxine mesylate | 8067-24-1 | >98.00% | |
A mixture of alkaloids with diverse biological activities | ||||
| GC10540 | NS 11021 | 956014-19-0 | >99.00% | |
NS 11021是一种具有高效选择性的大电导钙激活钾通道(BKCa/KCa1.1)激活剂。 | ||||
| GC10551 | pep4c | 243843-43-8 | - | |
Inactive control peptide analog of pep2m | ||||
| GC10560 | ICA 110381 | 325457-99-6 | - | |
ICA 110381 (Compound 16) 是一种 KCNQ2/Q3 钾通道开放剂,用于治疗癫痫。 | ||||
| GC10574 | Norketamine hydrochloride | 79499-59-5 | >98.00% | |
Major metabolite of ketamine, NMDA receptor antagonist | ||||
| GC10578 | ZD 7288 | 133059-99-1 | >99.50% / >98.00% | |
ZD 7288是一种超极化激活环核苷酸门控(HCN)通道阻滞剂。 | ||||
| GC10579 | Ouabain Octahydrate | 11018-89-6 | >99.50% | |
Ouabain Octahydrate是一种Na + /K + -ATPase抑制剂,能够用于研究充血性心力衰竭。 | ||||
