Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC18027Huwentoxin XVICAS: 1600543-88-1
Huwentoxin XVI 是一种镇痛剂,是一种来自中国狼蛛 Ornithoctonus huwena 的高度可逆和选择性的哺乳动物 N 型钙通道 (IC50 为 ~60 nM) 拮抗剂。
- GC18069CardamoninCAS: 19309-14-9纯度: >98.00%
A chalconoid with anti-inflammatory and anti-tumor activity
- GC18105EnterostatinCAS: 117830-79-2纯度: >99.50% / >98.00%
A pentapeptide involved in the regulation of food intake
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC18005 | Tenatoprazole | 113712-98-4 | >98.00% | |
A proton pump inhibitor | ||||
| GC18020 | AP 18 | 55224-94-7 | >98.00% / >99.50% | |
A reversible channel blocker of TRPA1 | ||||
| GC18027 | Huwentoxin XVI | 1600543-88-1 | - | |
Huwentoxin XVI 是一种镇痛剂,是一种来自中国狼蛛 Ornithoctonus huwena 的高度可逆和选择性的哺乳动物 N 型钙通道 (IC50 为 ~60 nM) 拮抗剂。 | ||||
| GC18033 | γDGG | 6729-55-1 | - | |
γDGG 是一种竞争性 AMPA 受体阻滞剂。 | ||||
| GC18052 | AZ 11645373 | 227088-94-0 | - | |
Human P2X7 antagonist,potent and selective | ||||
| GC18069 | Cardamonin | 19309-14-9 | >98.00% | |
A chalconoid with anti-inflammatory and anti-tumor activity | ||||
| GC18070 | ω-Conotoxin MVIIC | 147794-23-8 | - | |
An N-, P-, and Q-type calcium channel blocker | ||||
| GC18079 | CFM-2 | 178616-26-7 | >98.50% | |
CFM-2 是一种有效且选择性的非竞争性 AMPAR 拮抗剂。 | ||||
| GC18105 | Enterostatin | 117830-79-2 | >99.50% / >98.00% | |
A pentapeptide involved in the regulation of food intake | ||||
| GC18113 | UCM 707 | 390824-20-1 | - | |
An endocannabinoid analog that potentiates AEA activity | ||||
| GC18142 | Eact | 461000-66-8 | >98.00% | |
Eact是一种高特异性、强效的TMEM16A激活剂,能在钙离子浓度升高时激活TMEM16A。 | ||||
| GC18150 | L-CCG-lll | 117857-95-1 | - | |
L-CCG-lll (L-CCG III) 是一种有效的、竞争性的谷氨酸摄取抑制剂。 | ||||
| GC18176 | 5α,6β-Dihydroxycholestanol | 1253-84-5 | - | |
An oxysterol metabolite of cholesterol | ||||
| GC18189 | Marinobufagenin | 470-42-8 | >99.00% | |
An α 1 Na + /K + ATPase sodium pump inhibitor | ||||
| GC18203 | Annonacin | 111035-65-5 | >98.00% | |
A mitochondrial complex I inhibitor | ||||
| GC18210 | GAL-021 | 1380341-99-0 | >98.00% | |
A BK Ca channel blocker | ||||
| GC18223 | Farampator | 211735-76-1 | >99.50% | |
A positive allosteric modulator of AMPA receptors | ||||
| GC18260 | FTase Inhibitor I | 149759-96-6 | >95.00% | |
A potent and selective FTase inhibitor | ||||
| GC18262 | Acetamiprid | 135410-20-7 | >99.50% | |
A neonicotinoid insecticide | ||||
| GC18274 | Amiprofos-methyl | 36001-88-4 | - | |
An herbicide | ||||
| GC18296 | M8-B (hydrochloride) | 883976-12-3 | >98.00% | |
A selective TRPM8 antagonist | ||||
| GC18299 | Lorediplon | 917393-39-6 | >99.50% | |
A ligand for α 1 subunit-containing GABA A receptors | ||||
| GC18341 | meta-Fluoxetine (hydrochloride) | 79088-29-2 | - | |
An isomer of fluoxetine | ||||
| GC18358 | MONNA | 1572936-83-4 | - | |
MONNA是ANO1(anoctamin-1/TMEM16A)钙激活氯通道的特异性阻断剂,对非洲爪蟾卵母细胞中xANO1的IC 50 为0.08μM。 | ||||
