Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC17597Bafilomycin A1CAS: 88899-55-2纯度: >95.00% / >97.00% / >96.00% / >96.50%
巴菲霉素A1是一种大环内酯类抗生素,从链霉菌属中分离出来,它是真空泡H ATPase(V-ATPase)的抑制剂。
- GC17646L-(-)-threo-3-Hydroxyaspartic acidCAS: 7298-99-9纯度: >98.00%
L-(-)-threo-3-Hydroxyaspartic acid 是一种天然存在的、具有特定立体化学构型的氨基酸衍生物。L-(-)-threo-3-Hydroxyaspartic acid是谷氨酸受体(特别是NMDA受体)的一种选择性激动剂。
- GC17661E-4031 dihydrochlorideCAS: 113559-13-0纯度: >98.50%
An antiarrhythmic, ERG potassium channel blocker
- GC17739PNU 37883 hydrochlorideCAS: 57568-80-6
PNU 37883 hydrochloride (PNU 37883A) 是一种选择性血管 ATP 敏感性钾 (Kir6, KATP) 通道阻滞剂。
- GC17786Istaroxime hydrochlorideCAS: 374559-48-5纯度: >99.00%
Istaroxime hydrochloride 是 Na+/K+-ATPase 抑制剂 (IC50=0.11 μM) 和肌质/内质网钙 ATPase 2 (SERCA 2) 激活剂。
- GC17787UK 78282 hydrochlorideCAS: 136647-02-4
KV1.3 and KV1.4 voltage-gated potassium channel blocker
- GC17823L-Cysteinesulfinic acidCAS: 1115-65-7纯度: >98.00%
L-半胱氨酸亚磺酸是几种大鼠代谢型谷氨酸受体 (mGluR) 的有效激动剂,对 mGluR1、mGluR5、mGluR2、mGluR4、mGluR6 和 mGluR8 的 pEC50 分别为 3.92、4.6、3.9、2.7、4.0 和 3.94 .
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC17592 | CP 100356 hydrochloride | 142715-48-8 | >99.00% | |
A P-glycoprotein inhibitor | ||||
| GC17595 | CP 339818 hydrochloride | 478341-55-8 | - | |
KV1.3 channel antagonist | ||||
| GC17597 | Bafilomycin A1 | 88899-55-2 | >95.00% / >97.00% / >96.00% / >96.50% | |
巴菲霉素A1是一种大环内酯类抗生素,从链霉菌属中分离出来,它是真空泡H ATPase(V-ATPase)的抑制剂。 | ||||
| GC17608 | Lidocaine | 137-58-6 | >99.50% | |
An Analytical Reference Standard | ||||
| GC17646 | L-(-)-threo-3-Hydroxyaspartic acid | 7298-99-9 | >98.00% | |
L-(-)-threo-3-Hydroxyaspartic acid 是一种天然存在的、具有特定立体化学构型的氨基酸衍生物。L-(-)-threo-3-Hydroxyaspartic acid是谷氨酸受体(特别是NMDA受体)的一种选择性激动剂。 | ||||
| GC17652 | N-(4-Hydroxyphenylacetyl)spermine | 130210-32-1 | - | |
NMDA receptor antagonist | ||||
| GC17661 | E-4031 dihydrochloride | 113559-13-0 | >98.50% | |
An antiarrhythmic, ERG potassium channel blocker | ||||
| GC17675 | 4,4-Pentamethylenepiperidine hydrochloride | 1125-01-5 | - | |
M2 proton channel blocker | ||||
| GC17687 | CALP3 | 261969-05-5 | >99.00% | |
A calcium-like peptide | ||||
| GC17690 | Cromolyn sodium | 15826-37-6 | >99.00% | |
A mast cell stabilizer | ||||
| GC17693 | Enniatin B | 917-13-5 | - | |
A natural inhibitor of Pdr5p in yeast | ||||
| GC17739 | PNU 37883 hydrochloride | 57568-80-6 | - | |
PNU 37883 hydrochloride (PNU 37883A) 是一种选择性血管 ATP 敏感性钾 (Kir6, KATP) 通道阻滞剂。 | ||||
| GC17786 | Istaroxime hydrochloride | 374559-48-5 | >99.00% | |
Istaroxime hydrochloride 是 Na+/K+-ATPase 抑制剂 (IC50=0.11 μM) 和肌质/内质网钙 ATPase 2 (SERCA 2) 激活剂。 | ||||
| GC17787 | UK 78282 hydrochloride | 136647-02-4 | - | |
KV1.3 and KV1.4 voltage-gated potassium channel blocker | ||||
| GC17823 | L-Cysteinesulfinic acid | 1115-65-7 | >98.00% | |
L-半胱氨酸亚磺酸是几种大鼠代谢型谷氨酸受体 (mGluR) 的有效激动剂,对 mGluR1、mGluR5、mGluR2、mGluR4、mGluR6 和 mGluR8 的 pEC50 分别为 3.92、4.6、3.9、2.7、4.0 和 3.94 . | ||||
| GC17842 | CARIPORIDE | 159138-80-4 | >98.50% | |
An NHE-1 inhibitor | ||||
| GC17853 | Amiloride HCl | 2016-88-8 | >98.00% | |
An Analytical Reference Standard | ||||
| GC17870 | A 804598 | 1125758-85-1 | >98.50% | |
A potent and selective competitive antagonist of the P2X 7 receptor | ||||
| GC17879 | OLDA | 105955-11-1 | >98.00% | |
A synthetic endocannabinoid analog and potent 5-lipoxygenase inhibitor | ||||
| GC17909 | NS 6180 | 353262-04-1 | >99.50% | |
An inhibitor of IKCa1/K Ca 3.1 channels | ||||
| GC17928 | IDRA 21 | 22503-72-6 | - | |
IDRA 21 是 AMPA 受体的阳性和口服活性调节剂。 | ||||
| GC17930 | T16Ainh - A01 | 552309-42-9 | >99.00% / >98.50% | |
An inhibitor of TMEM16A channels | ||||
| GC17934 | TB 21007 | 207306-50-1 | - | |
An inverse agonist of α 5 β 3 γ 2 subunit-containing GABA A receptors | ||||
| GC17940 | GSK1016790A | 942206-85-1 | >99.50% / >98.00% | |
GSK1016790A是一种有效的选择性瞬时受体电位香草酸4(TRPV4)通道激动剂。 | ||||
