Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
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- GlyT(19)
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- Na+/H+ Exchanger (NHE)(1)
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Membrane Transporter/Ion Channel 相关产品(2265)
- GC17225ARL 67156 trisodium saltCAS: 1021868-83-6纯度: >98.00%
ARL 67156 trisodium salt是一种选择性的细胞外ATP酶抑制剂。
- GC17355TNP-ATP triethylammonium saltCAS: 61368-63-6
An antagonist of P2X 1 , P2X 3 , and P2X 2/3 receptors and a fluorescent probe
- GC17496W-7 hydrochlorideCAS: 61714-27-0纯度: >98.00%
W-7 hydrochloride是一种强效的钙调蛋白拮抗剂,可抑制钙离子-钙调蛋白诱导的肌球蛋白轻链激酶激活,IC 50 值为25μM。
- GC17519Concanamycin ACAS: 80890-47-7纯度: >95.00% / >98.00%
Concanamycin A 是液泡型 ATP 酶 (V-ATPase) 的特异性抑制剂,IC50 值为 10 nM 。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC17225 | ARL 67156 trisodium salt | 1021868-83-6 | >98.00% | |
ARL 67156 trisodium salt是一种选择性的细胞外ATP酶抑制剂。 | ||||
| GC17257 | Saclofen | 125464-42-8 | >98.00% / >99.00% | |
Saclofen是一种口服竞争性GABAB受体拮抗剂,IC 50 值为7.8μM。 | ||||
| GC17264 | ZM 226600 | 147695-92-9 | - | |
Kir6 (KATP) channel opener | ||||
| GC17267 | RN 1734 | 946387-07-1 | >98.00% | |
A TRPV4 antagonist | ||||
| GC17272 | Charybdotoxin | 95751-30-7 | - | |
A blocker of K+ channels | ||||
| GC17280 | NS 5806 | 426834-69-7 | >98.00% | |
An I to current activator | ||||
| GC17313 | (S)-CPW 399 | 389888-02-2 | - | |
AMPA agonist,subtype-selective,weakly desensitizing | ||||
| GC17320 | NF 157 | 104869-26-3 | >90.00% | |
NF 157 是一种高度选择性的纳摩尔 P2Y11 拮抗剂,pKi 为 7.35。 | ||||
| GC17321 | RuBi-GABA | 1028141-88-9 | - | |
RuBi-GABA 是一种新型的钌基笼状 GABA 化合物。 | ||||
| GC17350 | L-655,708 | 130477-52-0 | >99.00% / >98.00% / >98.50% | |
A ligand for α 5 subunit-containing GABA A receptors with nootropic activity | ||||
| GC17355 | TNP-ATP triethylammonium salt | 61368-63-6 | - | |
An antagonist of P2X 1 , P2X 3 , and P2X 2/3 receptors and a fluorescent probe | ||||
| GC17375 | AZ 10606120 dihydrochloride | 607378-18-7 | >99.00% | |
A P2X 7 receptor antagonist | ||||
| GC17381 | trans-4-Hydroxycrotonic acid | 24587-49-3 | - | |
ligand of γ-hydroxybutyric acid (GHB) receptor | ||||
| GC17395 | ICA 121431 | 313254-51-2 | >98.00% | |
A selective Na v 1.1 and Na v 1.3 channel blocker | ||||
| GC17399 | Pregnanolone | 128-20-1 | - | |
GABAA receptor positive allosteric modulator | ||||
| GC17402 | Tiagabine hydrochloride | 145821-59-6 | >99.50% | |
A GAT-1 inhibitor | ||||
| GC17442 | Methsuximide | 77-41-8 | - | |
An anticonvulsant | ||||
| GC17456 | NMDA (N-Methyl-D-aspartic acid) | 6384-92-5 | >98.00% | |
An excitatory neurotransmitter | ||||
| GC17481 | Gavestinel | 153436-38-5 | - | |
An NMDA receptor antagonist | ||||
| GC17495 | QX 314 chloride | 5369-03-9 | >99.50% | |
A selective sodium channel blocker | ||||
| GC17496 | W-7 hydrochloride | 61714-27-0 | >98.00% | |
W-7 hydrochloride是一种强效的钙调蛋白拮抗剂,可抑制钙离子-钙调蛋白诱导的肌球蛋白轻链激酶激活,IC 50 值为25μM。 | ||||
| GC17518 | YS-035 hydrochloride | 89805-39-0 | - | |
A calcium channel blocker | ||||
| GC17519 | Concanamycin A | 80890-47-7 | >95.00% / >98.00% | |
Concanamycin A 是液泡型 ATP 酶 (V-ATPase) 的特异性抑制剂,IC50 值为 10 nM 。 | ||||
| GC17562 | 2-APB | 524-95-8 | >98.00% | |
2-APB是一种钙离子通道的非特异性拮抗剂,通常被用于研究钙信号传导,如细胞凋亡、肌肉收缩和神经传导等方面。 | ||||
