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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel(跨膜转运)

Cat.No. 产品名称 Information
GC18564 MK6-83 A TRPML1 activator
GC18505 Carisbamate
RWJ-333369
An antiepileptic agent
GC18503 DK-AH 269
西洛雷定盐酸盐,DK-AH 269
An HCN channel blocker
GC18474 Acetyldigitoxin
乙酰洋地黄毒甙; Digitoxin 3'''-Acetate
An Na⁺/K⁺ ATPase inhibitor
GC18470 NSC 23925 An inhibitor of P-gp
GC18460 Roquefortine C
异烟棒曲霉素 C
A mycotoxin
GC18445 N-Deacetylcolchicine
NSC 201400
An inhibitor of microtubule polymerization
GC18426 8-Nitroguanine A mutagenic nitrative guanine derivative
GC18410 Ro 25-6981 (maleate) A potent, NR2B-selective NMDA receptor antagonist
GC18358 MONNA
2-(4-甲氧基萘-2-基氨基)-5-硝基苯甲酸
MONNA是ANO1（anoctamin-1/TMEM16A）钙激活氯通道的特异性阻断剂，对非洲爪蟾卵母细胞中xANO1的IC₅₀为0.08μM。
GC18341 meta-Fluoxetine (hydrochloride)
氟西汀相关物质A
An isomer of fluoxetine
GC18299 Lorediplon A ligand for α₁ subunit-containing GABA_A receptors
GC18296 M8-B (hydrochloride) A selective TRPM8 antagonist
GC18274 Amiprofos-methyl
甲基胺草磷,BAY-NTN 6867
An herbicide
GC18260 FTase Inhibitor I
N-[(2S)-((2R)-2-氨基-3-巯基丙基氨基)-3-甲基丁基]-L-苯丙氨酰-L-蛋氨酸,B581
A potent and selective FTase inhibitor
GC18223 Farampator
CX-691; Org24448
A positive allosteric modulator of AMPA receptors
GC18210 GAL-021 A BK_Ca channel blocker
GC18203 Annonacin A mitochondrial complex I inhibitor
GC18189 Marinobufagenin
南美蟾毒精
An α₁ Na⁺/K⁺ ATPase sodium pump inhibitor
GC18176 5α,6β-Dihydroxycholestanol
胆甾烷-3,5,6-三醇
An oxysterol metabolite of cholesterol
GC14041 Ethacrynic Acid
依他尼酸; 利尿酸; Etacrynic acid
Ethacrynic Acid是一种强效的、口服有效的袢利尿剂。
GC15411 Clopamide
氯帕胺；氯哌酰胺
A thiazide-like diuretic
GC16533 Oligomycin Complex
寡霉素
寡霉素复合物(Oligomycin complex)由寡霉素A、B和C的混合物组成。
GC12421 Brilliant blue G-250
酸性蓝90,Acid Blue 90,CBBG,Coomassie Brilliant Blue G-250,NSC 328382

A dye for staining or quantifying proteins
GC15461 Guanidinoethyl sulfonate
脒基牛磺酸,NSC 667063,Taurocyamine
Guanidinoethyl sulfonate（GES）是一种牛磺酸类似物，可竞争性抑制牛磺酸的摄取，通过作为TauT、PAT1和GAT2的竞争性抑制剂导致牛磺酸耗竭，并干扰牛磺酸的生物合成。
GC11284 6-(4-Methoxyphenyl)-3-pyridazinamine
6-(4-甲氧基苯基)哒嗪-3-胺
A GABA_A receptor antagonist
GC17940 GSK1016790A GSK1016790A是一种有效的选择性瞬时受体电位香草酸4（TRPV4）通道激动剂。
GC12439 Quinacrine (hydrochloride hydrate)
Atebrine,Mepacrine
An acridine compound with diverse biological activities and cell labeling properties
GC11492 Fluspirilene
帕罗西汀杂质C,McN-JR 6218,R 6218,Redeptin
An L-type calcium channel antagonist
GC11010 AZD 3965 MCT1 的 Ki = 1.6 nMAZD 3965 是单羧酸转运蛋白 1 (MCT1) 的有效抑制剂。
GC15117 ML-297
CID-56642816,VU0456810
A selective GIRK1/2 activator
GC17442 Methsuximide
甲琥胺,(±)-Mesuximide,PM 396
An anticonvulsant
GC15308 IAA-94
R-(+)-甲基吲唑酮,R(+)-IAA 94
IAA-94 (Indanyloxyacetic acid-94) 是一种细胞内氯离子通道阻滞剂。
GC11351 VU590 (hydrochloride)
CID-4536383,ML-111
inhibitor of KCNJ1
GC10934 Bafilomycin C1
巴菲霉素C1
A fungal metabolite with diverse biological activities
GC13381 WZB117
Glucose Transporter Inhibitor IV
WZB117是一种靶向葡萄糖转运蛋白1（GLUT1）的小分子抑制剂。
GC12636 Capsiconiate
Coniferyl (E)-8-methyl-6-nonenoate
A partial agonist of TRPV1
GC17001 Verruculogen
疣孢青霉原
A tremorgenic mycotoxin
GC12302 Bafilomycin D
巴佛洛霉素D
A fungal metabolite with diverse biological activities
GC12742 CP-465022 (maleate) An AMPA receptor antagonist
GC16627 Docosahexaenoyl Serotonin Potential TRPV1 antagonist
GC15580 Stearoyl Serotonin Potential TRPV1 antagonist
GC12097 Palmitoyl Serotonin Potential TRPV1 antagonist
GC11147 Oleoyl Serotonin TRPV1 antagonist
GC12772 Eicosapentaenoyl Serotonin A potential TRPV1 antagonist
GC12927 (±)-Baclofen
巴氯芬
(±)-Baclofen是γ-氨基丁酸（GABA）的亲脂性衍生物，是一种口服有效，选择性的代谢型GABAB受体激动剂，IC₅₀为200nM。
GC10964 Estradiol 17-(β-D-Glucuronide) (sodium salt)
Β雌二醇17-(Β-D-葡萄糖醛酸)钠盐,E217G,β-Estradiol 17-(β-D-Glucuronide),17β-Estradiol 17-(β-D-Glucuronide),17β-Oestradiol 17-(β-D-Glucuronide)
Estradiol 17-(β-D-Glucuronide)是雌二醇(一种主要的女性性激素)经过代谢形成的产物。
GC16924 Eniporide
N-(二氨基亚甲基)-2-甲基-5-(甲基磺酰基)-4-(1H-吡咯-1-基)苯甲酰胺
A NHE-1 inhibitor
GC13289 Barnidipine (hydrochloride)
盐酸巴尼地平,YM 09730-5
A calcium channel blocker
GC12700 Ivermectin B1a
伊维菌素 B1a
An anthelmintic