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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel(跨膜转运)

  1. Cat.No. 产品名称 Information
  2. GC30418 SKF96067 SKF96067是一种可逆的H+/K+-ATPase抑制剂。
  3. GC30415 Propafenone D7 hydrochloride (SA-79 (D7 hydrochloride))

    盐酸普罗帕酮 D7; SA-79 D7 hydrochloride

     Propafenone D7 (SA-79 D7) hydrochloride 是氘标记的 Propafenone，是一种经典的抗心律失常药物。
  4. GC30371 Alisol F

    泽泻醇 F

     A triterpene with anti-inflammatory and hepatoprotective activities
  5. GC30361 CRAC intermediate 2

    4-(3,5-双(三氟甲基)-1H-吡唑-1-基)-苯胺

     CRACintermediate2是摘自专利WO2013059666A1中用于CRAC系列抑制剂合成的中间体。
  6. GC30322 PF-05241328 PF-05241328是有效的、人电压依赖性钠通道(Nav1.7)的选择性抑制剂，其IC50值为31nM。
  7. GC30280 Chlorpromazine D6 hydrochloride

    盐酸氯丙嗪 D6

     Chlorpromazine D6 hydrochloride是 Chlorpromazine 的氘代物，可被用于 NMR、GC-MS 或 LC-MS 分析中的内标品，用于定量分析。
  8. GC30267 Pinacidil monohydrate

    吡那地尔一水合物; P-1134 monohydrate

     Pinacidil monohydrate一种抗高血压药物，属于钾通道开放剂，通过激活ATP敏感性钾通道使血管平滑肌松弛。
  9. GC30212 (S)-Willardiine ((-)-Willardiine)

    尿嘧啶基丙氨酸; (-)-Willardiine

     (S)-Willardiine ((-)-Willardiine)是一种强效的AMPA/kainate受体激动剂，EC50值为45μM。
  10. GC30130 Soraprazan (BYK61359)

    BYK61359

    Soraprazan (BYK61359) (BYK61359) 是一种选择性的、可逆的 K 竞争性 H,K-ATPase 抑制剂 (Ki=6.4 nM)，在胃腺中的 IC50 为 0.19 μM。
  11. GC30110 Oleic acid (9-cis-Octadecenoic acid)

    油酸; 9-cis-Octadecenoic acid; 9Z-Octadecenoic acid

     油酸（9-顺式-十八碳烯酸）是一种单不饱和的Omega-9脂肪酸，存在于植物和动物中。
  12. GC30096 Pyr10

    Pyr10是一种新型TRPC3选择性抑制剂,作用于转染YFP-TRPC3的HEK293细胞,抑制ROCE,IC50为0.72uM。
  13. GC30088 Fluxametamide

    4-[5-(3,5-二氯苯基)-4,5-二氢-5-(三氟甲基)-3-异恶唑基]-N-[(甲氧基氨基)亚甲基]-2-甲基苯甲酰胺

     Fluxametamide是一种GABA和谷氨酸门控氯离子通道的拮抗剂，对GABACls和GluCls的IC50值分别为1.95nM和225nM。
  14. GC30063 Eleclazine hydrochloride (GS 6615 hydrochloride)

    GS 6615 hydrochloride

     Eleclazine hydrochloride (GS 6615 hydrochloride)是一种新型、具有高度选择性的心脏晚期钠电流抑制剂，IC50值<1μM。
  15. GC30055 Pinaverium bromide

    匹维溴铵

     Pinaverium bromide (Icosapentaenoic acid) acts as a calcium channel blocker and is useful for functional gastrointestinal disorders.
  16. GC30054 Dantrolene sodium hemiheptahydrate (Dantrolene sodium hydrate)

    丹曲林钠,Dantrolene sodium hydrate

     Dantrolene sodium hemiheptahydrate (Dantrium) ia a skeletal muscle relaxant that acts by interfering with excitation-contraction coupling in the muscle fiber.
  17. GC30033 Sinapine thiocyanate

    芥子碱硫氰酸盐

     Sinapine thiocyanate is the thiocyanate salt form of Sinapine, which shows favorable biological activities such as antioxidant and radio-protective activities.
  18. GC19480 AUT1 A positive modulator of Kv3.1b, Kv3.2a, and Kv3.3
  19. GC19438 TMB 8 (hydrochloride)

    3,4,5-三甲氧基苯甲酸(8-二乙氨基正辛基)酯盐酸盐

     A non-competitive antagonist of nAChRs and an inhibitor of intracellular calcium availability
  20. GC19422 Gefapixant

    吉法匹生,AF219; MK-7264)

     Gefapixant 是一种具有口服活性的强效嘌呤能 P2X3 受体 (P2X3R) 拮抗剂，与重组 hP2X3 同源三聚体相比，IC50 值约为 30 nM，对 hP2X2/3 异源三聚体受体的 IC50 值为 100-250 nM。
  21. GC19373 Verinurad

    维立诺雷; RDEA3170

     A URAT1 inhibitor
  22. GC19370 Valbenazine

    缬苯那嗪,NBI-98854

     An inhibitor of VMAT2
  23. GC19352 Tenapanor

    AZD1722; RDX5791

     A NHE-3 inhibitor
  24. GC19351 Tebanicline hydrochloride

    ABT594盐酸盐

     A potent agonist of neuronal α4β2 subunit-containing nAChRs
  25. GC19346 Talampanel

    (8R)-7-乙酰基-5-(4-氨基苯基)-8,9-二氢-8-甲基-7H-1,3-二氧杂环戊烯并[4,5-H][2,3]苯并二氮杂卓,GYKI-53773; LY-300164

     An allosteric AMPA receptor antagonist
  26. GC19310 Ro 25-6981 A potent, NR2B-selective NMDA receptor antagonist
  27. GC19291 PF-4840154 A TRPA1 channel agonist
  28. GC19289 PF-06869206 An NaPi2a inhibitor
  29. GC19281 PF-01247324

    2-吡啶甲酰胺,6-氨基-N-甲基-5-(2,3,5-三氯苯基)-

     An inhibitor of Nav1.8 channels
  30. GC19271 ONO-8590580 A negative allosteric modulator of α5 subunit-containing GABAA receptors
  31. GC19252 MK-8998

    MK-8998

     MK-8998 (MK-8998; Compound 33) 是一种有效的选择性 T 型钙通道抑制剂。
  32. GC19183 GSK369796 Dihydrochloride

    N-tert-butyl Isoquine

     An antimalarial agent
  33. GC19169 GLPG1837

    ABBV-974

     A CFTR potentiator
  34. GC19152 Fantofarone

    泛托法隆,SR 33557

     A calcium channel inhibitor
  35. GC19107 CM-4620

    CM-4620

     CM-4620是一种选择性Orai通道抑制剂，对Orai1和Orai2的IC50值分别为0.119μM和0.895μM。
  36. GC19057 Basmisanil

    巴米沙尼,RG1662; RO5186582

     A negative allosteric modulator of α5 subunit-containing GABAA receptors
  37. GC19025 AM-0902 AM-0902 是一种有效的选择性瞬时受体电位 A1 (TRPA1) 拮抗剂，对 rTRPA1 和 hTRPA1 的 IC50 分别为 71 和 131 nM。
  38. GC19022 AF-353

    Ro-4

     A dual P2X3 and P2X2/3 receptor antagonist
  39. GC19021 Adjudin

    男用口服避孕药,AF-2364

     A derivative of lonidamine
  40. GC19016 ABT-639 A T-type calcium channel blocker
  41. GC19004 SKA-121 A positive-gating modulator of IKCa1/KCa3.1 channels
  42. GC19000 BAY-588

    A glucose transporter inhibitor
  43. GC18947 PF-05089771 (tosylate) An Nav1.7 channel blocker
  44. GC18890 Emamectin B1a

    依马菌素B1A

     An insecticide
  45. GC18827 Supercinnamaldehyde A TRPA1 channel activator
  46. GC18762 Remogliflozin A

    Remogliflozin A

     A potent inhibitor of SGLT2
  47. GC18641 Ferutinin An ERα agonist
  48. GC18631 4BP-TQS An agonist of α7 subunit-containing nAChRs
  49. GC18629 VU0071063 A Kir6.2/SUR1 activator
  50. GC18603 (±)-Methoxyverapamil (hydrochloride)

    Methoxyverapamil hydrochloride

     An L-type channel blocker
  51. GC18583 D-α-Hydroxyglutaric Acid

    R-2-羟基戊二酸,(R)-2-Hydroxyglutarate; (R)-2-Hydroxyglutaric acid; (R)-2-Hydroxypentanedioic acid

     D-α-Hydroxyglutaric Acid是α-酮戊二酸（α-KG）的弱竞争性拮抗剂（Ki = 10.87mM）。

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