Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
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- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC16240MNI-caged-NMDACAS: 1227675-52-6
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group
- GC16353N-ArachidonylGABACAS: 128201-89-8纯度: >98.00%
A natural arachidonoyl amino acid with analgesic activity
- GC16354Dequalinium ChlorideCAS: 522-51-0纯度: >99.00%
An ammonium cation with diverse biological activities
- GC16409Oligomycin BCAS: 11050-94-5纯度: >85.00%
A nonselective inhibitor of the mitochondrial F 1 F O ATP synthase
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16167 | K 858 | 72926-24-0 | >99.50% | |
An inhibitor of Eg5 | ||||
| GC16182 | Co 102862 | 181144-66-1 | - | |
Co 102862 (V 102862) 是一种强效、广谱、依赖于状态的 Na+ 通道阻滞剂。 | ||||
| GC16188 | CL 218872 | 66548-69-4 | - | |
An anxiolytic agent | ||||
| GC16199 | 8-pCPT-2-O-Me-cAMP-AM | 1152197-23-3 | >97.00% | |
Epac activator | ||||
| GC16221 | Oligomycin C | 11052-72-5 | - | |
A mitochondrial F 1 F O ATP synthase inhibitor | ||||
| GC16238 | FGIN-1-43 | 145040-29-5 | - | |
ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor) | ||||
| GC16240 | MNI-caged-NMDA | 1227675-52-6 | - | |
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group | ||||
| GC16254 | Iberiotoxin | 129203-60-7 | - | |
Selective blocker of K Ca 1.1/BK channels | ||||
| GC16255 | Decamethonium Bromide | 541-22-0 | >98.00% | |
A depolarizing neuromuscular blocking agent | ||||
| GC16272 | CGS 19755 | 110347-85-8 | >98.00% | |
NMDA receptor antagonist | ||||
| GC16300 | ZK 200775 | 161605-73-8 | >99.00% | |
ZK 200775 (ZK200775) 是一种高度选择性的 AMPA/红藻氨酸拮抗剂,对 NMDA 几乎没有活性; Ki 值分别为 3.2 nM、100 nM 和 8.5 μ;M 分别针对 quisqualate、红藻氨酸和 NMDA。 | ||||
| GC16311 | Chlormethiazole hydrochloride | 6001-74-7 | >98.00% | |
A potentiator of GABA A receptors | ||||
| GC16315 | D-AP5 | 79055-68-8 | >98.00% | |
D-AP5是一种选择性N-甲基-D-天门冬胺酸(NMDA)受体拮抗剂,K d 值为1.4μM。 | ||||
| GC16322 | trans-Ned 19 | 1354235-96-3 | >99.50% | |
An antagonist of NAADP receptors | ||||
| GC16330 | Ro 51 | 1050670-85-3 | - | |
Ro 51 是一种有效的选择性双重 P2X3/P2X2/3 拮抗剂,对 P2X3 和 P2X2/3 的 IC50 分别为 2 nM 和 5 nM。 | ||||
| GC16342 | PPNDS | 1021868-77-8 | - | |
PPNDS 是一种选择性和竞争性的 meprin ⋲;抑制剂 (IC50: 80 nM, Ki: 8 nM),并且还抑制 ADAM10 (IC50: 1.2 μM)。 | ||||
| GC16353 | N-ArachidonylGABA | 128201-89-8 | >98.00% | |
A natural arachidonoyl amino acid with analgesic activity | ||||
| GC16354 | Dequalinium Chloride | 522-51-0 | >99.00% | |
An ammonium cation with diverse biological activities | ||||
| GC16356 | SB 205384 | 160296-13-9 | - | |
positive GABAA receptor modulator | ||||
| GC16359 | Rosuvastatin | 287714-41-4 | - | |
Rosuvastatin是一种竞争性HMG-CoA还原酶抑制剂,IC 50 值为11nM。 | ||||
| GC16360 | TP 003 | 628690-75-5 | - | |
GABAA receptor (α3 subtype) partial agonist | ||||
| GC16390 | Ropivacaine hydrochloride monohydrate | 132112-35-7 | >99.50% | |
A sodium channel blocker | ||||
| GC16409 | Oligomycin B | 11050-94-5 | >85.00% | |
A nonselective inhibitor of the mitochondrial F 1 F O ATP synthase | ||||
| GC16419 | OMDM-2 | 616884-63-0 | - | |
An inhibitor of AEA uptake | ||||
