Membrane Transporter/Ion Channel
Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(58)
- ATPase(80)
- Calcium Channel(331)
- Cannabinoid Transporters(6)
- CFTR(45)
- Chloride Channels(13)
- GABA Receptor(239)
- Gardos Channel(1)
- Glucose Transporters(13)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(19)
- GTPase(32)
- Kv1.3(1)
- ICB(2)
- Lipophilic platinum complex(1)
- M2 ion Channel(1)
- MCT2(2)
- Monoamine transporter(18)
- Monocarboxylate Transporters(12)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(16)
- NKCC(7)
- NMDA Receptor(81)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(68)
- P-gp(11)
- Proton Pump(56)
- Potassium Channel(308)
- Sodium Channel(211)
- TRP Channel(165)
- TRPV1(10)
- URAT1(12)
- Other Channel Modulators(10)
- MCT(3)
- Kainate Receptors(12)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(27)
- CRAC Channel(13)
- EAAT2(6)
- HCN Channel(6)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(49)
- iGluR(164)
- nAChR(103)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Ferroportin(1)
- Urea Transporter(1)
- Na+/H+ Exchanger (NHE)(1)
- NTPDase(1)
- EAAT(1)
- Piezo Channel(1)
- ASCT(2)
Membrane Transporter/Ion Channel 相关产品(2265)
- GC13283Ralfinamide mesylateCAS: 202825-45-4
Ralfinamide mesylate (FCE-26742A mesylate) 是一种来自 α-氨基酰胺的口服 Na+ 通道阻滞剂,具有抑制疼痛的作用。
- GC13375Dofequidar fumarateCAS: 153653-30-6纯度: >98.00%
A quinoline derivative and inhibitor of multidrug resistance
- GC13455VU 591 hydrochlorideCAS: 1315380-70-1纯度: >98.00%
VU 591 hydrochloride 是一种有效的、选择性的肾外髓质钾通道 (ROMK 或 Kir1.1) 抑制剂,IC50 为 0.24 μM。
- GC13482NBQX disodium saltCAS: 479347-86-9纯度: >98.00%
NBQX 二钠盐是 α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate (AMPA) 受体 (AMPAR) 的强效、高选择性和竞争性拮抗剂。
- GC13494Phrixotoxin 3CAS: 880886-00-0纯度: >95.00%
Phrixotoxin 3 是一种有效的电压门控钠通道阻滞剂,对 NaV1.2、NaV1.3、NaV1.4、NaV1.1 和 NaV1.5 的 IC50 分别为 0.6、42、72、288、610 nM。
- GC13515AlphaxaloneCAS: 23930-19-0
activates and potentiates GABAA receptor-activated membrane current (IGABA)
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13283 | Ralfinamide mesylate | 202825-45-4 | - | |
Ralfinamide mesylate (FCE-26742A mesylate) 是一种来自 α-氨基酰胺的口服 Na+ 通道阻滞剂,具有抑制疼痛的作用。 | ||||
| GC13289 | Barnidipine (hydrochloride) | 104757-53-1 | >98.50% | |
A calcium channel blocker | ||||
| GC13290 | CMPDA | 380607-77-2 | - | |
A positive allosteric modulator of GluA2 | ||||
| GC13323 | BDS I | - | - | |
Kv3.4 potassium channel blocker, potent and reversible | ||||
| GC13349 | Naspm trihydrochloride | 1049731-36-3 | >98.00% | |
A synthetic analog of Joro spider toxin | ||||
| GC13352 | Neomycin sulfate | 1405-10-3 | >98.00% | |
An antibiotic used in tissue culture studies | ||||
| GC13353 | Spadin | 1270083-24-3 | >99.00% | |
An inhibitor of K 2P 2.1/TREK1 | ||||
| GC13374 | CGP 13501 | 56189-68-5 | >98.00% | |
Positive modulator of GABAB receptors,allosteric | ||||
| GC13375 | Dofequidar fumarate | 153653-30-6 | >98.00% | |
A quinoline derivative and inhibitor of multidrug resistance | ||||
| GC13381 | WZB117 | 1223397-11-2 | >99.50% | |
WZB117是一种靶向葡萄糖转运蛋白1(GLUT1)的小分子抑制剂。 | ||||
| GC13387 | Vigabatrin Hydrochloride | 1391054-02-6 | >99.00% | |
Inhibitor of GABA transaminase | ||||
| GC13405 | DMCM hydrochloride | 1215833-62-7 | >98.00% | |
DMCM hydrochloride 是苯二氮卓类的非选择性全反向激动剂。 | ||||
| GC13455 | VU 591 hydrochloride | 1315380-70-1 | >98.00% | |
VU 591 hydrochloride 是一种有效的、选择性的肾外髓质钾通道 (ROMK 或 Kir1.1) 抑制剂,IC50 为 0.24 μM。 | ||||
| GC13457 | ML 204 | 5465-86-1 | >98.00% | |
A selective TRPC4 channel blocker | ||||
| GC13466 | Flufenamic acid | 530-78-9 | >99.50% | |
An NSAID and COX inhibitor | ||||
| GC13469 | Piracetam | 7491-74-9 | >99.00% | |
An Analytical Reference Standard | ||||
| GC13482 | NBQX disodium salt | 479347-86-9 | >98.00% | |
NBQX 二钠盐是 α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate (AMPA) 受体 (AMPAR) 的强效、高选择性和竞争性拮抗剂。 | ||||
| GC13490 | E-4031 | 113558-89-7 | >99.00% | |
An antiarrhythmic, ERG potassium channel blocker | ||||
| GC13494 | Phrixotoxin 3 | 880886-00-0 | >95.00% | |
Phrixotoxin 3 是一种有效的电压门控钠通道阻滞剂,对 NaV1.2、NaV1.3、NaV1.4、NaV1.1 和 NaV1.5 的 IC50 分别为 0.6、42、72、288、610 nM。 | ||||
| GC13505 | Licarbazepine | 29331-92-8 | >98.00% / >97.00% | |
A metabolite of oxcarbazepine | ||||
| GC13509 | U 90042 | 134516-99-7 | - | |
GABAA receptor ligand | ||||
| GC13515 | Alphaxalone | 23930-19-0 | - | |
activates and potentiates GABAA receptor-activated membrane current (IGABA) | ||||
| GC13542 | Adiphenine HCl | 50-42-0 | >99.50% | |
An anticholinergic agent | ||||
| GC13557 | PHP 501 trifluoroacetate | 1236105-75-1 | - | |
GABAA antagonist | ||||
