Signaling Pathways
Signaling Pathways(信号通路)
- Proteases(63)
- Apoptosis(1190)
- Chromatin/Epigenetics(17)
- Metabolism(420)
- MAPK Signaling(32)
- Tyrosine Kinase(97)
- DNA Damage/DNA Repair(62)
- PI3K/Akt/mTOR Signaling(56)
- Microbiology & Virology(68)
- Cell Cycle/Checkpoint(205)
- Ubiquitination/ Proteasome(43)
- JAK/STAT Signaling(13)
- TGF-β / Smad Signaling(30)
- Angiogenesis(85)
- GPCR/G protein(3)
- Stem Cell(27)
- Membrane Transporter/Ion Channel(273)
- Cancer Biology(514)
- Endocrinology and Hormones(168)
- Neuroscience(462)
- Obesity, Appetite Control & Diabetes(9)
- Peptide Inhibitors and Substrate(1)
- Other Signal Transduction(141)
- Immunology/Inflammation(1111)
- Cardiovascular(63)
- Vitamin D Related
- Antibody-drug Conjugate/ADC Related
- PROTAC(254)
- Ox Stress Reagents(25)
- Others(1718)
- Antiparasitics(21)
- Toxins(90)
Signaling Pathways 相关产品(35130)
- GC12301MizoribineCAS: 50924-49-7纯度: >98.50%
An imidazole nucleoside with immunosuppressive properties
- GC12308Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) DisodiumCAS: 168555-66-6纯度: >99.00%
Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium是一种微管解聚药物,作为Combretastatin A4(CA4)的水溶性前体药物。
- GC12350T-705 (Favipiravir)CAS: 259793-96-9纯度: >99.50%
T-705 (Favipiravir)是一种广谱抗病毒药物。T-705通过选择性抑制RNA病毒的RNA依赖性RNA聚合酶(RdRp),发挥抗病毒作用。
- GC12356GlibenclamideCAS: 10238-21-8纯度: >99.50%
格列本脲 (Glyburide) 是一种具有口服活性的 ATP 敏感性 K+ 通道 (KATP) 抑制剂,可用于糖尿病和肥胖症的研究。
- GC12391XanthohumolCAS: 6754-58-1纯度: >99.50% / >98.00%
Xanthohumol是啤酒花中主要的异戊烯基黄酮类化合物,能够抑制二酰甘油酰基转移酶(DGAT),IC 50 值为50.3μM。
- GC12405ABT-263 (Navitoclax)CAS: 923564-51-6纯度: >98.00%
ABT-263 (Navitoclax) 是 Bcl-xL、Bcl-2 和 Bcl-w 的抑制剂,Ki 分别≤0.5 nM、≤1 nM 和≤1 nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC12299 | Telaprevir (VX-950) | 402957-28-2 | >98.00% | |
An HCV NS3/4A protease inhibitor | ||||
| GC12301 | Mizoribine | 50924-49-7 | >98.50% | |
An imidazole nucleoside with immunosuppressive properties | ||||
| GC12303 | Desmopressin | 16679-58-6 | - | |
A vasopressin receptor agonist | ||||
| GC12308 | Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium | 168555-66-6 | >99.00% | |
Fosbretabulin (Combretastatin A4 Phosphate (CA4P)) Disodium是一种微管解聚药物,作为Combretastatin A4(CA4)的水溶性前体药物。 | ||||
| GC12312 | Cilnidipine | 132203-70-4 | >99.50% | |
An L- and N-type calcium channel blocker | ||||
| GC12332 | NU 7026 | 154447-35-5 | >99.50% | |
Inhibitor of DNA-dependent protein kinase | ||||
| GC12335 | GSK461364 | 929095-18-1 | >99.50% | |
A reversible inhibitor of Plk1 | ||||
| GC12339 | Ivermectin | 70288-86-7 | >98.00% | |
Ivermectin是一种大环内酯类内外抗寄生虫药,对体内和体外寄生虫均有活性。 | ||||
| GC12350 | T-705 (Favipiravir) | 259793-96-9 | >99.50% | |
T-705 (Favipiravir)是一种广谱抗病毒药物。T-705通过选择性抑制RNA病毒的RNA依赖性RNA聚合酶(RdRp),发挥抗病毒作用。 | ||||
| GC12356 | Glibenclamide | 10238-21-8 | >99.50% | |
格列本脲 (Glyburide) 是一种具有口服活性的 ATP 敏感性 K+ 通道 (KATP) 抑制剂,可用于糖尿病和肥胖症的研究。 | ||||
| GC12361 | Darapladib | 356057-34-6 | >99.50% | |
A reversible inhibitor of Lp-PLA 2 | ||||
| GC12363 | LY2109761 | 700874-71-1 | >99.50% | |
LY2109761是一种口服小分子双TGF-β受体(TβR)I/II激酶抑制剂(TβRI: K i = 38nM;TβRII: K i = 300nM)。 | ||||
| GC12365 | Ranitidine hydrochloride | 66357-59-3 | >98.00% | |
A histamine H 2 receptor antagonist | ||||
| GC12374 | Alarelin Acetate | 79561-22-1 | >98.00% | |
Alarelin Acetate是一种合成的促性腺激素释放激素激动剂。 | ||||
| GC12376 | Maprotiline HCl | 10347-81-6 | >99.00% | |
A tricyclic antidepressant | ||||
| GC12379 | Drospirenone | 67392-87-4 | >98.00% | |
A synthetic progestogen | ||||
| GC12381 | Natamycin | 7681-93-8 | >99.00% | |
A macrolide polyene antifungal agent | ||||
| GC12384 | D-64131 | 74588-78-6 | >99.00% | |
An inhibitor of tubulin polymerization | ||||
| GC12389 | Efavirenz | 154598-52-4 | >99.00% | |
Efavirenz是一种非核苷逆转录酶抑制剂(NNRTI)。 | ||||
| GC12390 | A-966492 | 934162-61-5 | >99.00% | |
A PARP1 and PARP2 inhibitor | ||||
| GC12391 | Xanthohumol | 6754-58-1 | >99.50% / >98.00% | |
Xanthohumol是啤酒花中主要的异戊烯基黄酮类化合物,能够抑制二酰甘油酰基转移酶(DGAT),IC 50 值为50.3μM。 | ||||
| GC12398 | Granisetron | 109889-09-0 | - | |
Granisetron (BRL 43694) 是一种血清素 5-HT3 受体拮抗剂,用作止吐剂,用于治疗化疗后的恶心和呕吐。 | ||||
| GC12405 | ABT-263 (Navitoclax) | 923564-51-6 | >98.00% | |
ABT-263 (Navitoclax) 是 Bcl-xL、Bcl-2 和 Bcl-w 的抑制剂,Ki 分别≤0.5 nM、≤1 nM 和≤1 nM。 | ||||
| GC12408 | Progesterone | 57-83-0 | >98.00% | |
An endogenous hormone and hormone precursor | ||||
