Neuroscience
Neuroscience(神经科学)
Neuroscience
Neurons communicate with each other, effector organs and sensory organs through the neurotransmitter – receptor pathway at synapses. Neurotransmitters can be divided into 4 major groups: 1. Amino acids (glumate, aspartate, serine, glycine and GABA); 2. Monoamines (norepinephrine, epinephrine, dopamine, histamine, and serotonin); 3. Peptides (opioid peptides, substance P, somatostatin); and 4. Others (acetylcholine, NO, nucleosides). read more
- 5-HT Receptor(442)
- AChR(58)
- AChE(103)
- Alzheimer(115)
- Amyloid β(131)
- BACE(5)
- CGRP (34)
- COX(302)
- DAPK(7)
- Dopamine Receptor(312)
- GABA Receptor(168)
- Gap Junction(18)
- GluR(121)
- Histamine(3)
- Histamine Receptor(243)
- mPEGS-1(4)
- Muscarinic Receptor(43)
- Neuroscience Peptides(48)
- Nicotinic Receptor(66)
- P2 Receptor(2)
- P2X7 receptor(4)
- SSRIs(8)
- Substance P/NK1 Receptor(22)
- NMDA(2)
- Beta-secretase(25)
- CaMK(33)
- Dopamine Transporter(20)
- Monoamine Oxidase(91)
- Serotonin Transporter(57)
- nAChR(103)
- iGluR(163)
- Neurokinin Receptor(75)
- MCHR1 (GPR24)(16)
- mAChR(185)
- GPR139(4)
- Cholecystokinin Receptor(25)
- Behavioral Neuroscience(372)
- DREADD(1)
- Huntington(17)
- Neuroendocrinology(65)
- Neuroprotection(128)
- Ophthalmology(168)
- Pain Research(241)
- Parkinson(78)
- Prion(7)
- Seizure Disorders(99)
- Cholinesterases(13)
- AAK1
- Huntingtin
- α-synuclein
- Transthyretin (TTR)
- Tau Protein(4)
- Neurodegenerative Disorders(7)
- Cholinesterase (ChE)(4)
- Amyloid-β(9)
- γ-secretase(1)
- Ischemia(3)
Neuroscience 相关产品(3932)
- GC35428Atropine sulfateCAS: 55-48-1纯度: >98.00%
A non- selective muscarinic acetylcholine receptor antagonist
- GC35444Azaphen dihydrochloride monohydrateCAS: 63302-99-8纯度: >99.50%
Pipofezine(Azafen,Azaphen)是5-羟色胺重吸收抑制剂。
- GC35455BACE1-IN-4CAS: 2361157-92-6
BACE1-IN-4 是一种有效、高度选择性的 BACE1 抑制剂,IC50 值为 3.8 nM,Ki 值为 1.9 nM。抗阿尔滋海默症。
- GC35473Bavisant dihydrochloride hydrateCAS: 1103522-80-0纯度: >99.50%
Bavisant dihydrochloride hydrate (JNJ31001074AAC) 是口服活性人H3 受体拮抗剂。
- GC35492Benzamide Derivative 1CAS: 108226-05-7
Benzamide Derivative 1是来自专利EP0213775A1,化合物18,的苯甲酰胺衍生物。Benzamide Derivative 1可能用于治疗胃肠疾病的研究。
- GC35493Benzoylgomisin OCAS: 130783-32-3
Benzoylgomisin O 是从 Schisandra rubriflora 中分离的化合物,对 15-LOX、COX-1、COX-2 酶有抑制作用,且具有抗炎活性。
- GC35564BuChE-IN-TM-10CAS: 2313524-95-5
BuChE-IN-TM-10 (TM-10)是一种有效的丁基胆碱酯酶 (BuChE) 抑制剂,其IC50 值为8.9 nM。BuChE inhibitor 1能够抑制和分解自诱导的Aβ聚合, 表现出强大的抗氧化活性和良好的血脑屏障 (BBB) 渗透性。有治疗阿尔兹海默症的潜能。
- GC35601CaMKII-IN-1CAS: 1208123-85-6纯度: >99.50% / >98.00%
CaMKII-IN-1是一种强效且高度选择性的CaMKII抑制剂,IC 50 值为63nM。
- GC35656Cetirizine D8 dihydrochlorideCAS: 2070015-04-0
An internal standard for the quantification of cetirizine,(R)-cetirizine, and (S)-cetirizine
- GC35751CS-003 Free baseCAS: 191672-52-3
CS-003 Free base (CS-003)是一种三速激肽受体拮抗剂,对人神经激肽 (Neurokinin) NK1,NK2 和 NK3 受体具有高亲和力,Ki 值分别为 2.3 nM,0.54 nM 和 0.74 nM。CS-003 Free base (CS-003) 对与神经激肽有关的呼吸系统疾病具有治疗功效。
- GC35807Danegaptide HydrochlorideCAS: 943133-81-1纯度: >99.00%
Danegaptide Hydrochloride是一种有效的、选择性的、具有口服活性的间隙连接(gap-junction)修饰剂。
- GC35810DarifenacinCAS: 133099-04-4纯度: >98.00%
Darifenacin HBr (UK-88525) is a selective M3 muscarinic receptor antagonist with pKi of 8.9.
- GC35820DDD107498 succinateCAS: 2444781-71-7纯度: >98.50%
DDD107498 (M-5717, DDD-498) is a P. falciparum translation elongation factor 2 inhibitor. DDD107498 exhibits a potent and novel spectrum of antimalarial activity against multiple life-cycle stages of the Plasmodium parasite.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC35428 | Atropine sulfate | 55-48-1 | >98.00% | |
A non- selective muscarinic acetylcholine receptor antagonist | ||||
| GC35432 | Autocamtide-2-related inhibitory peptide (TFA) | - | >95.00% | |
A CaMKII inhibitor | ||||
| GC35443 | Azaphen | 24853-80-3 | - | |
Pipofezine(Azafen,Azaphen)是5-羟色胺重吸收抑制剂。 | ||||
| GC35444 | Azaphen dihydrochloride monohydrate | 63302-99-8 | >99.50% | |
Pipofezine(Azafen,Azaphen)是5-羟色胺重吸收抑制剂。 | ||||
| GC35455 | BACE1-IN-4 | 2361157-92-6 | - | |
BACE1-IN-4 是一种有效、高度选择性的 BACE1 抑制剂,IC50 值为 3.8 nM,Ki 值为 1.9 nM。抗阿尔滋海默症。 | ||||
| GC35471 | Bavisant | 929622-08-2 | - | |
Bavisant (JNJ-31001074)是口服活性人H3受体拮抗剂。 | ||||
| GC35472 | Bavisant dihydrochloride | 929622-09-3 | - | |
Bavisant盐酸盐(JNJ-31001074)是口服活性人H3受体拮抗剂。 | ||||
| GC35473 | Bavisant dihydrochloride hydrate | 1103522-80-0 | >99.50% | |
Bavisant dihydrochloride hydrate (JNJ31001074AAC) 是口服活性人H3 受体拮抗剂。 | ||||
| GC35492 | Benzamide Derivative 1 | 108226-05-7 | - | |
Benzamide Derivative 1是来自专利EP0213775A1,化合物18,的苯甲酰胺衍生物。Benzamide Derivative 1可能用于治疗胃肠疾病的研究。 | ||||
| GC35493 | Benzoylgomisin O | 130783-32-3 | - | |
Benzoylgomisin O 是从 Schisandra rubriflora 中分离的化合物,对 15-LOX、COX-1、COX-2 酶有抑制作用,且具有抗炎活性。 | ||||
| GC35524 | Biperiden | 514-65-8 | - | |
Biperiden(KL 373)有抗帕金森症活性,是中枢M1胆碱受体阻断剂。 | ||||
| GC35538 | BNC375 | 1557240-80-8 | >99.50% | |
BNC375 是一种口服有效的选择性 α7nAChRs I 型正向变构调节剂,EC50 为 1.9 μM。 | ||||
| GC35564 | BuChE-IN-TM-10 | 2313524-95-5 | - | |
BuChE-IN-TM-10 (TM-10)是一种有效的丁基胆碱酯酶 (BuChE) 抑制剂,其IC50 值为8.9 nM。BuChE inhibitor 1能够抑制和分解自诱导的Aβ聚合, 表现出强大的抗氧化活性和良好的血脑屏障 (BBB) 渗透性。有治疗阿尔兹海默症的潜能。 | ||||
| GC35601 | CaMKII-IN-1 | 1208123-85-6 | >99.50% / >98.00% | |
CaMKII-IN-1是一种强效且高度选择性的CaMKII抑制剂,IC 50 值为63nM。 | ||||
| GC35610 | Cariprazine hydrochloride | 1083076-69-0 | >98.50% | |
An atypical antipsychotic | ||||
| GC35655 | Cetirizine D4 dihydrochloride | - | - | |
Cetirizine D4二盐酸盐是Cetirizine氘代化合物标准品。 | ||||
| GC35656 | Cetirizine D8 dihydrochloride | 2070015-04-0 | - | |
An internal standard for the quantification of cetirizine,(R)-cetirizine, and (S)-cetirizine | ||||
| GC35669 | CGP 36742 | 123690-78-8 | >98.00% | |
A GABA B receptor antagonist | ||||
| GC35720 | Colivelin TFA | 2803948-60-7 | >95.00% | |
A potent STAT3 activator and neuroprotective agent | ||||
| GC35751 | CS-003 Free base | 191672-52-3 | - | |
CS-003 Free base (CS-003)是一种三速激肽受体拮抗剂,对人神经激肽 (Neurokinin) NK1,NK2 和 NK3 受体具有高亲和力,Ki 值分别为 2.3 nM,0.54 nM 和 0.74 nM。CS-003 Free base (CS-003) 对与神经激肽有关的呼吸系统疾病具有治疗功效。 | ||||
| GC35806 | Danegaptide | 943134-39-2 | >98.00% | |
Danegaptide是一种有效的、选择性的、具有口服活性的间隙连接(gap-junction)修饰剂。 | ||||
| GC35807 | Danegaptide Hydrochloride | 943133-81-1 | >99.00% | |
Danegaptide Hydrochloride是一种有效的、选择性的、具有口服活性的间隙连接(gap-junction)修饰剂。 | ||||
| GC35810 | Darifenacin | 133099-04-4 | >98.00% | |
Darifenacin HBr (UK-88525) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. | ||||
| GC35820 | DDD107498 succinate | 2444781-71-7 | >98.50% | |
DDD107498 (M-5717, DDD-498) is a P. falciparum translation elongation factor 2 inhibitor. DDD107498 exhibits a potent and novel spectrum of antimalarial activity against multiple life-cycle stages of the Plasmodium parasite. | ||||
