GlpBio

GABA Receptor

GABA Receptor(γ-氨基丁酸受体)

GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.

GABA Receptor 相关产品(154)

  • GC10772 structure
    GC10772Flumazenil
    CAS: 78755-81-4
    纯度: >99.50% / >98.00%

    A GABA A receptor antagonist and partial agonist

  • GC10974 structure
    GC10974AWD 131-138
    CAS: 188116-07-6
    纯度: >99.00%

    A partial agonist of the GABA A receptor

  • GC11901 structure
    GC11901Nefiracetam
    CAS: 77191-36-7
    纯度: >99.00%

    An Analytical Reference Standard

  • GC12599 structure
    GC12599Retigabine dihydrochloride
    CAS: 150812-13-8
    纯度: >99.00%

    An Analytical Reference Standard

  • GC12714 structure
    GC12714Gabapentin
    CAS: 60142-96-3
    纯度: >98.00%

    An approved antiepileptic drug

  • GC13792 structure
    GC13792Rufinamide
    CAS: 106308-44-5
    纯度: >99.50%

    An anticonvulsant

  • GC14111 structure
    GC14111(R)-baclofen
    CAS: 69308-37-8
    纯度: >99.00% / >98.00%

    (R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。

  • GC14916 structure
    GC14916Acamprosate calcium
    CAS: 77337-73-6
    纯度: >98.00%

    An NMDA modulator

  • GC15264 structure
    GC15264Etifoxine hydrochloride
    CAS: 56776-32-0
    纯度: >99.50%

    A positive allosteric modulator of GABA A receptors

  • GC16564 structure
    GC16564Niflumic acid
    CAS: 4394-00-7
    纯度: >99.50%

    A selective COX-2 inhibitor

  • GA10004 structure
    GA10004H-D-Met-OH
    CAS: 348-67-4
    纯度: >98.00%

    H-D-Met-OH (MRX-1024; D-H-D-Met-OH) 是一种有效的化学保护剂，还可以通过 GABAA 受体激活抑制神经元活性。

  • GA10664 structure
    GA10664H-Dab•HBr
    CAS: 1758-80-1
    纯度: >98.00%

    H-Dab•HBr (L-2,4-Diaminobutyric acid) 是一周 GABA 转氨酶抑制剂，IC50 大于 500 μM;在体内和体外均表现出抗肿瘤活性。

  • GC10101 structure
    GC10101SR 95531 hydrobromide
    CAS: 104104-50-9
    纯度: >98.00% / >97.00%

    SR 95531 氢溴酸盐 (Gabazine) 是 GABAA 受体上 GABA 结合位点的选择性拮抗剂 。

  • GC10186 structure
    GC10186Tiagabine
    CAS: 115103-54-3
    纯度: 99.98%

    A GAT-1 inhibitor

  • GC10530 structure
    GC10530Dihydroergotoxine mesylate
    CAS: 8067-24-1
    纯度: >98.00%

    A mixture of alkaloids with diverse biological activities

  • GC10888 structure
    GC10888SCH 50911
    CAS: 733717-87-8

    SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-乙酸，一种选择性、口服活性和竞争性 γ-氨基丁酸 B GABA(B) 受体拮抗剂，与 GABA(B ) 受体，IC50 为 1.1 μM。

  • GC11013 structure
    GC11013U 93631
    CAS: 152273-12-6
    纯度: >99.50%

    A GABA A receptor ligand

  • GC11054 structure
    GC11054Epiallopregnanolone
    CAS: 567-01-1
    纯度: >95.00%

    A neurosteroid

  • GC11143 structure
    GC11143NS 11394
    CAS: 951650-22-9
    纯度: >99.50%

    A subunit-selective positive allosteric modulator of the GABA A receptor

  • GC11963 structure
    GC11963Oxiracetam
    CAS: 62613-82-5
    纯度: >98.00%

    An Analytical Reference Standard

  • GC12414 structure
    GC12414Bemegride
    CAS: 64-65-3
    纯度: >99.50%

    Bemegride (3-Ethyl-3-methylglutarimide) 是一种中枢神经系统兴奋剂和巴比妥类中毒的解毒剂。

  • GC12568 structure
    GC12568FG 7142
    CAS: 78538-74-6
    纯度: >99.00%

    A benzodiazepine receptor ligand

  • GC12927 structure
    GC12927(±)-Baclofen
    CAS: 1134-47-0
    纯度: >99.00% / >98.00%

    (±)-Baclofen是γ-氨基丁酸（GABA）的亲脂性衍生物，是一种口服有效，选择性的代谢型GABAB受体激动剂，IC 50 为200nM。

  • GC13387 structure
    GC13387Vigabatrin Hydrochloride
    CAS: 1391054-02-6
    纯度: >99.00%

    Inhibitor of GABA transaminase