AChE(乙酰胆碱脂酶)
AChE, also know as acetylcholinesterase, is a hydrolase that hydrolyzes the neurotransmitter acetylcholine.
Products for AChE
- Cat.No. 产品名称 Information
-
GN10155
(+)- Corydaline
紫堇碱; (+)-Corydaline; Corydalin
An alkaloid with diverse biological activities -
GN10654
(+)-Corynoline
紫蓳灵
An isoquinoline alkaloid with diverse biological activities -
GC34947
(-)-Corynoxidine
延胡索乙素N氧化物
(-)-Corynoxidine 分离自延胡索 Corydalis speciosa,是一种乙酰胆碱酯酶 acetylcholinesterase 抑制剂,IC50 值为 89.0 μM。(-)-Corynoxidine 对金黄色葡萄球菌和耐甲氧西林金黄色葡萄球菌菌株有不同程度的抗菌活性。
-
GC14400
(-)-Huperzine A
石杉碱甲; Huperzine A
A neuroprotective AChE inhibitor -
GC48551
(-)-Physostigmine (salicylate)
水杨酸毒扁豆碱; Eserine salicylate
An alkaloid and cholinergic agent -
GC34993
(R)-Rivastigmine D6 tartrate
酒石酸卡巴拉汀 D6
An internal standard for the quantification of rivastigmine -
GC11965
(±)-Huperzine A
(±)-石杉碱甲
A neuroprotective AChE inhibitor -
GC41774
1,2,3-Trimyristoyl-rac-glycerol
三肉豆蔻酸甘油酯
A triacylglycerol -
GC38698
1-Naphthyl acetate
乙酸-1-萘酯
1-Naphthyl acetate is usually used in a rapid staining method for identification of macrophages. 1-Naphthyl acetate is a potent chromogenic substrate for the detection of erythrocyte acetylcholinesterase (AChE) activity. -
GC11606
4-Methylbenzylidene camphor
4-甲基苄亚基樟脑; 4-MBC; Enzacamene
A UV blocker with estrogenic effects -
GC15203
Acephate
乙酰甲胺磷
An organophosphate insecticide -
GC35236
Acetylshikonin
乙酰紫草素
Acetylshikonin,来源于紫草根,具有抗癌、抗炎作用。Acetylshikonin 是一种非选择性的细胞色素 P450 抑制剂,对所有 P450 亚型抑制的 IC50 值范围为 1.4-4.0 μM。Acetylshikonin 是一种 AChE 抑制剂,具有很强的抗凋亡活性。 -
GC62827
Acotiamide D6
Z-338-d6 free base; YM443-d6 free base
Acotiamide D6 是 Acotiamide 的氘代物。Acotiamide 是有潜力用于功能性消化不良的首创的且具有口服活性的胃肠动力药。 -
GC38732
Acotiamide monohydrochloride trihydrate
盐酸阿考替胺三水合物
Acotiamide Hydrochloride (YM-443, Z-338) is the hydrochloride salt form of acotiamide, a prokinetic agent with gastrointestinal (GI) motility-enhancing activity. It is a new orally active selective acetylcholinesterase inhibitor. -
GC35272
Ajmalicine
萝巴新,Raubasine
A terpenoid indole alkaloid -
GC35279
Aldicarb sulfone
涕灭威砜
A metabolite of aldicarb -
GC16974
Ambenonium dichloride
安贝氯铵,WIN 8077 chloride
Ambenonium (WIN 8077) chloride 是一种具有高亲和力的具有口服活性且可逆的乙酰胆碱酯酶 (AChE) 抑制剂。 -
GC15438
Asoxime (chloride)
HI-6
An AChE reactivator -
GC31193
Benactyzine hydrochloride
胃复康
Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety. -
GC15628
bis(7)-Tacrine
1,7-N-heptylene-bis-9,9'-amino-1,2,3,4-tetrahydro-acridine
A potent acetylcholinesterase inhibitor -
GC35564
BuChE-IN-TM-10
TM-10
BuChE-IN-TM-10 (TM-10)是一种有效的丁基胆碱酯酶 (BuChE) 抑制剂,其IC50 值为8.9 nM。BuChE inhibitor 1能够抑制和分解自诱导的Aβ聚合, 表现出强大的抗氧化活性和良好的血脑屏障 (BBB) 渗透性。有治疗阿尔兹海默症的潜能。 -
GC60108
Chlorpyrifos
毒死蜱
毒死蜱作为一种广谱有机硫代磷酸酯类杀虫剂,其主要致毒机制是通过使神经接头处的乙酰胆碱酯酶失活。 -
GC39836
Coumaran
2,3-二氢苯并呋喃; 2,3-Dihydrobenzofuran
Coumaran (2,3-Dihydrobenzofuran) 是一种从 L. camara 中提取的 (AChE) 抑制剂。Coumaran 可以用作生物农药。 -
GC43336
Cyanidin 3-O-β-D-Galactopyranoside (chloride)
矢车菊素半乳糖苷; Ideain chloride
An anthocyanin flavonoid with antioxidant properties -
GC38625
Dehydronuciferine
去氢荷叶碱
Dehydronuciferine 从 Nelumbo nucifera Gaertn 的叶子中分离,是一种乙酰胆碱酯酶 (AChE) 抑制剂,其 IC50 为 25 μg/mL。 -
GC31190
Demecarium Bromide (BC-48)
地美溴铵; BC-48
Demecarium Bromide (BC-48) (BC-48) 是一种有效的胆碱酯酶抑制剂,表观亲和力 (Kiapp) 为 0.15 μM. -
GC60774
Dihydro Donepezil
盐酸多奈哌齐二氢杂质,Dihydro E2020
DihydroDonepezil(DihydroE2020)是Donepezil的代谢产物。Donepezil是一种有效的特异性AChE抑制剂,对bAChE和hAChE的IC50分别为8.12nM和11.6nM。 -
GC63620
Dihydrowithaferin A
二氢醉茄素A; 2,3-Dihydrowithaferin A
Dihydrowithaferin A (2, 3-dihydrowithaferin A) 是一种从 Withania somnifera 分离的睡茄内酯类化合物。Dihydrowithaferin A 对乙酰胆碱酯酶有抑制活性。 -
GC30810
Donepezil (E2020)
多奈哌齐; E2020 free base
Donepezil (E2020)是一种乙酰胆碱酯酶(AChE)抑制剂,IC50为6.7nM。 -
GC14490
Donepezil HCl
盐酸多奈哌齐; E2020
An AChE inhibitor
-
GC63334
Donepezil-d7 hydrochloride
E2020-d7
Donepezil-d7 (hydrochloride) (E2020-d7) 是 Donepezil 的氘代物。Donepezil (E2020 free base) 是 AChE 抑制剂,对牛 AChE 和人 AChE 的 IC50 分别为 8.12 nM 和 11.6 nM。 -
GC30908
Drofenine hydrochloride (Hexahydroadiphenine hydrochloride)
盐酸六氢芬宁,Hexahydroadiphenine hydrochloride
Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers. -
GC17705
Edrophonium (chloride)
依酚氯铵
An AChE inhibitor -
GN10716
Epiberberine
表小檗碱
An alkaloid with diverse biological activities -
GC35996
Epiberberine chloride
表小檗碱氯化物
An alkaloid with diverse biological activities -
GC60164
Fenitrothion
杀螟松
Fenitrothion 是应用最广泛的有机磷农药之一,是一种抑制胆碱酯酶的杀虫剂/杀螨剂。Fenitrothion 作为一种广谱杀虫剂,广泛应用于棉田作物、蔬菜作物、水果作物和大田作物,尤其是水稻。Fenitrothion 导致硝基酚的积累。 -
GC16573
Galanthamine
加兰他敏; Galantamine
An alkaloid with AChE inhibitory and nAChR potentiating activities -
GC36103
Galanthamine hydrobromide
Galanthamine氢溴酸盐是长效的中心活性的乙酰胆碱酯酶(AChE)抑制剂,IC50为410 nM,同时是神经元烟碱乙酰胆碱受体的变构增强剂。
-
GC36104
Galanthaminone
氢溴酸加兰他敏,(-)-Narwedine; Narwedin
Galanthaminone是竞争性可逆的胆碱酯酶(AChE)抑制剂,可作用于多种记忆障碍疾病。 -
GC13474
Garcinol
山竹子素
Garcinol是组蛋白乙酰转移酶p300和PCAF的非特异性抑制剂,IC50分别为7μM和5μM。
-
GC15832
GSK 264220A
An endothelial lipase inhibitor
-
GC64193
Hemicholinium 3
半胆碱基-3,Hemicholinium dibromide
Hemicholinium 3 是一种竞争性的高亲和力胆碱转运蛋白 (HACU) 抑制剂,Ki 值为 25 nM。Hemicholinium 3抑制乙酰胆碱 (ACh)的合成和释放,用作一种神经肌肉阻滞剂。Hemicholinium 3 抑制Epibatidine诱发的收缩和 [3H] 乙酰胆碱释放,IC50 分别为 897 nM 和 693 nM。 -
GC38793
Huperzine B
石杉碱乙
An alkaloid with neuroprotective activity -
GC60913
Huperzine C
石杉碱丙
HuperzineC是从Huperziaserrate中分离的一种生物碱。HuperzineC是一种乙酰胆碱酯酶(AChE)抑制剂,其IC50值为0.6μM。HuperzineC可用于阿尔茨海默症的研究。 -
GC15604
Hydroxytacrine (maleate)
马来酸维吖啶,HP 029,1-Hydroxytacrine,P 83-6029A,Velnacrine
A major active metabolite of tacrine -
GN10437
Imperatorin
欧前胡素; Ammidin
A furanocoumarin with diverse biological activities -
GC36334
Isoeugenol acetate
乙酸异丁香酚酯; Acetyl isoeugenol
Isoeugenol acetate 是一种肉豆蔻,丁香和肉桂的精油成分,对某些代谢酶如乙酰胆碱酯酶 (AChE) 酶 (IC50=77 nM; Ki=16 nM),α-糖苷酶 (IC50=19.25 nM; Ki=21 nM) 和 α-淀粉酶 (IC50=411.5 nM) 具有良好的抑制作用。 Isoeugenol acetate 用于医疗和化妆品工业,具有抗氧化,抗癌,抗菌和抗炎特性。 -
GN10352
Isoimperatorin
异欧前胡素
A furanocoumarin that inhibits CYP1A -
GC36336
Isomerazin
异橙皮内酯
A coumarin with antioxidant and anti-inflammatory activities -
GC36340
Isorosmanol
异迷迭香酚
Isorosmanol 是从鼠尾草叶中分离出的一种松香烷型二萜,具有抗氧化、神经保护和神经营养作用。Isorosmanol 能抑制 AChE 活性和黑色素的合成。