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AChE(乙酰胆碱脂酶)

AChE, also know as acetylcholinesterase, is a hydrolase that hydrolyzes the neurotransmitter acetylcholine.

Products for  AChE

  1. Cat.No. 产品名称 Information
  2. GN10155 (+)- Corydaline

    紫堇碱; (+)-Corydaline; Corydalin

    An alkaloid with diverse biological activities
  3. GN10654 (+)-Corynoline

    紫蓳灵

    An isoquinoline alkaloid with diverse biological activities
  4. GC34947 (-)-Corynoxidine

    延胡索乙素N氧化物

    (-)-Corynoxidine 分离自延胡索 Corydalis speciosa,是一种乙酰胆碱酯酶 acetylcholinesterase 抑制剂,IC50 值为 89.0 μM。(-)-Corynoxidine 对金黄色葡萄球菌和耐甲氧西林金黄色葡萄球菌菌株有不同程度的抗菌活性。

  5. GC14400 (-)-Huperzine A

    石杉碱甲; Huperzine A

    A neuroprotective AChE inhibitor
  6. GC48551 (-)-Physostigmine (salicylate)

    水杨酸毒扁豆碱; Eserine salicylate

    An alkaloid and cholinergic agent
  7. GC34993 (R)-Rivastigmine D6 tartrate

    酒石酸卡巴拉汀 D6

    An internal standard for the quantification of rivastigmine
  8. GC11965 (±)-Huperzine A

    (±)-石杉碱甲

    A neuroprotective AChE inhibitor
  9. GC41774 1,2,3-Trimyristoyl-rac-glycerol

    三肉豆蔻酸甘油酯

    A triacylglycerol
  10. GC38698 1-Naphthyl acetate

    乙酸-1-萘酯

    1-Naphthyl acetate is usually used in a rapid staining method for identification of macrophages. 1-Naphthyl acetate is a potent chromogenic substrate for the detection of erythrocyte acetylcholinesterase (AChE) activity.
  11. GC11606 4-Methylbenzylidene camphor

    4-甲基苄亚基樟脑; 4-MBC; Enzacamene

    A UV blocker with estrogenic effects
  12. GC15203 Acephate

    乙酰甲胺磷

    An organophosphate insecticide
  13. GC35236 Acetylshikonin

    乙酰紫草素

    Acetylshikonin,来源于紫草根,具有抗癌、抗炎作用。Acetylshikonin 是一种非选择性的细胞色素 P450 抑制剂,对所有 P450 亚型抑制的 IC50 值范围为 1.4-4.0 μM。Acetylshikonin 是一种 AChE 抑制剂,具有很强的抗凋亡活性。
  14. GC62827 Acotiamide D6

    Z-338-d6 free base; YM443-d6 free base

    Acotiamide D6 是 Acotiamide 的氘代物。Acotiamide 是有潜力用于功能性消化不良的首创的且具有口服活性的胃肠动力药。
  15. GC38732 Acotiamide monohydrochloride trihydrate

    盐酸阿考替胺三水合物

    Acotiamide Hydrochloride (YM-443, Z-338) is the hydrochloride salt form of acotiamide, a prokinetic agent with gastrointestinal (GI) motility-enhancing activity. It is a new orally active selective acetylcholinesterase inhibitor.
  16. GC35272 Ajmalicine

    萝巴新,Raubasine

    A terpenoid indole alkaloid
  17. GC35279 Aldicarb sulfone

    涕灭威砜

    A metabolite of aldicarb
  18. GC16974 Ambenonium dichloride

    安贝氯铵,WIN 8077 chloride

    Ambenonium (WIN 8077) chloride 是一种具有高亲和力的具有口服活性且可逆的乙酰胆碱酯酶 (AChE) 抑制剂。
  19. GC15438 Asoxime (chloride)

    HI-6

    An AChE reactivator
  20. GC31193 Benactyzine hydrochloride

    胃复康

    Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.
  21. GC15628 bis(7)-Tacrine

    1,7-N-heptylene-bis-9,9'-amino-1,2,3,4-tetrahydro-acridine

    A potent acetylcholinesterase inhibitor
  22. GC35564 BuChE-IN-TM-10

    TM-10

    BuChE-IN-TM-10 (TM-10)是一种有效的丁基胆碱酯酶 (BuChE) 抑制剂,其IC50 值为8.9 nM。BuChE inhibitor 1能够抑制和分解自诱导的Aβ聚合, 表现出强大的抗氧化活性和良好的血脑屏障 (BBB) 渗透性。有治疗阿尔兹海默症的潜能。
  23. GC60108 Chlorpyrifos

    毒死蜱

    毒死蜱作为一种广谱有机硫代磷酸酯类杀虫剂,其主要致毒机制是通过使神经接头处的乙酰胆碱酯酶失活。
  24. GC39836 Coumaran

    2,3-二氢苯并呋喃; 2,3-Dihydrobenzofuran

    Coumaran (2,3-Dihydrobenzofuran) 是一种从 L. camara 中提取的 (AChE) 抑制剂。Coumaran 可以用作生物农药。
  25. GC43336 Cyanidin 3-O-β-D-Galactopyranoside (chloride)

    矢车菊素半乳糖苷; Ideain chloride

    An anthocyanin flavonoid with antioxidant properties
  26. GC38625 Dehydronuciferine

    去氢荷叶碱

    Dehydronuciferine 从 Nelumbo nucifera Gaertn 的叶子中分离,是一种乙酰胆碱酯酶 (AChE) 抑制剂,其 IC50 为 25 μg/mL。
  27. GC31190 Demecarium Bromide (BC-48)

    地美溴铵; BC-48

    Demecarium Bromide (BC-48) (BC-48) 是一种有效的胆碱酯酶抑制剂,表观亲和力 (Kiapp) 为 0.15 μM.
  28. GC60774 Dihydro Donepezil

    盐酸多奈哌齐二氢杂质,Dihydro E2020

    DihydroDonepezil(DihydroE2020)是Donepezil的代谢产物。Donepezil是一种有效的特异性AChE抑制剂,对bAChE和hAChE的IC50分别为8.12nM和11.6nM。
  29. GC63620 Dihydrowithaferin A

    二氢醉茄素A; 2,3-Dihydrowithaferin A

    Dihydrowithaferin A (2, 3-dihydrowithaferin A) 是一种从 Withania somnifera 分离的睡茄内酯类化合物。Dihydrowithaferin A 对乙酰胆碱酯酶有抑制活性。
  30. GC30810 Donepezil (E2020)

    多奈哌齐; E2020 free base

    Donepezil (E2020)是一种乙酰胆碱酯酶(AChE)抑制剂,IC50为6.7nM。
  31. GC14490 Donepezil HCl

    盐酸多奈哌齐; E2020

    An AChE inhibitor

  32. GC63334 Donepezil-d7 hydrochloride

    E2020-d7

    Donepezil-d7 (hydrochloride) (E2020-d7) 是 Donepezil 的氘代物。Donepezil (E2020 free base) 是 AChE 抑制剂,对牛 AChE 和人 AChE 的 IC50 分别为 8.12 nM 和 11.6 nM。
  33. GC30908 Drofenine hydrochloride (Hexahydroadiphenine hydrochloride)

    盐酸六氢芬宁,Hexahydroadiphenine hydrochloride

    Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
  34. GC17705 Edrophonium (chloride)

    依酚氯铵

    An AChE inhibitor
  35. GN10716 Epiberberine

    表小檗碱

    An alkaloid with diverse biological activities
  36. GC35996 Epiberberine chloride

    表小檗碱氯化物

    An alkaloid with diverse biological activities
  37. GC60164 Fenitrothion

    杀螟松

    Fenitrothion 是应用最广泛的有机磷农药之一,是一种抑制胆碱酯酶的杀虫剂/杀螨剂。Fenitrothion 作为一种广谱杀虫剂,广泛应用于棉田作物、蔬菜作物、水果作物和大田作物,尤其是水稻。Fenitrothion 导致硝基酚的积累。
  38. GC16573 Galanthamine

    加兰他敏; Galantamine

    An alkaloid with AChE inhibitory and nAChR potentiating activities
  39. GC36103 Galanthamine hydrobromide Galanthamine氢溴酸盐是长效的中心活性的乙酰胆碱酯酶(AChE)抑制剂,IC50为410 nM,同时是神经元烟碱乙酰胆碱受体的变构增强剂。
  40. GC36104 Galanthaminone

    氢溴酸加兰他敏,(-)-Narwedine; Narwedin

    Galanthaminone是竞争性可逆的胆碱酯酶(AChE)抑制剂,可作用于多种记忆障碍疾病。
  41. GC13474 Garcinol

    山竹子素

    Garcinol是组蛋白乙酰转移酶p300和PCAF的非特异性抑制剂,IC50分别为7μM和5μM。

  42. GC15832 GSK 264220A An endothelial lipase inhibitor
  43. GC64193 Hemicholinium 3

    半胆碱基-3,Hemicholinium dibromide

    Hemicholinium 3 是一种竞争性的高亲和力胆碱转运蛋白 (HACU) 抑制剂,Ki 值为 25 nM。Hemicholinium 3抑制乙酰胆碱 (ACh)的合成和释放,用作一种神经肌肉阻滞剂。Hemicholinium 3 抑制Epibatidine诱发的收缩和 [3H] 乙酰胆碱释放,IC50 分别为 897 nM 和 693 nM。
  44. GC38793 Huperzine B

    石杉碱乙

    An alkaloid with neuroprotective activity
  45. GC60913 Huperzine C

    石杉碱丙

    HuperzineC是从Huperziaserrate中分离的一种生物碱。HuperzineC是一种乙酰胆碱酯酶(AChE)抑制剂,其IC50值为0.6μM。HuperzineC可用于阿尔茨海默症的研究。
  46. GC15604 Hydroxytacrine (maleate)

    马来酸维吖啶,HP 029,1-Hydroxytacrine,P 83-6029A,Velnacrine

    A major active metabolite of tacrine
  47. GN10437 Imperatorin

    欧前胡素; Ammidin

    A furanocoumarin with diverse biological activities
  48. GC36334 Isoeugenol acetate

    乙酸异丁香酚酯; Acetyl isoeugenol

    Isoeugenol acetate 是一种肉豆蔻,丁香和肉桂的精油成分,对某些代谢酶如乙酰胆碱酯酶 (AChE) 酶 (IC50=77 nM; Ki=16 nM),α-糖苷酶 (IC50=19.25 nM; Ki=21 nM) 和 α-淀粉酶 (IC50=411.5 nM) 具有良好的抑制作用。 Isoeugenol acetate 用于医疗和化妆品工业,具有抗氧化,抗癌,抗菌和抗炎特性。
  49. GN10352 Isoimperatorin

    异欧前胡素

    A furanocoumarin that inhibits CYP1A
  50. GC36336 Isomerazin

    异橙皮内酯

    A coumarin with antioxidant and anti-inflammatory activities
  51. GC36340 Isorosmanol

    异迷迭香酚

    Isorosmanol 是从鼠尾草叶中分离出的一种松香烷型二萜,具有抗氧化、神经保护和神经营养作用。Isorosmanol 能抑制 AChE 活性和黑色素的合成。

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