Muscarinic Receptor
Muscarinic Receptor(毒蕈碱受体)
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
Muscarinic Receptor 相关产品(41)
- GC11831Umeclidinium bromideCAS: 869113-09-7纯度: >98.00%
A muscarinic acetylcholine receptor antagonist
- GC17157Cevimeline hydrochloride hemihydrateCAS: 153504-70-2纯度: >98.00%
Cevimeline hydrochloride hemihydrate (SNI-2011) 是乙酰胆碱的奎宁环衍生物，是一种选择性和口服活性的毒蕈碱 M1 和 M3 受体激动剂。
- GC17182Solifenacin succinateCAS: 242478-38-2纯度: >99.00%
A muscarinic M 1 , M 2 , and M 3 receptor antagonist
- GC17954Tolterodine tartrateCAS: 124937-52-6纯度: >99.50%
A muscarinic acetylcholine receptor antagonist
- GC11415Arecaidine but-2-ynyl ester tosylateCAS: 119630-77-2纯度: >98.00%
Arecaidine but-2-ynyl ester tosylate是一种选择性的毒蕈碱型乙酰胆碱受体（mAChR）M2激动剂。
- GC13129W-84 dibromideCAS: 21093-51-6纯度: >98.00%
W-84 (dibromide) 是一种有效的 M2-胆碱受体变构调节剂，可延缓 [3H]N-甲基东莨菪碱的解离。
- GC13174Telenzepine dihydrochlorideCAS: 147416-96-4
Telenzepine dihydrochloride 是一种选择性和口服活性的毒蕈碱 M1 受体拮抗剂，Ki 为 0.94 nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10621 | Biperiden HCl | 1235-82-1 | - | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC11831 | Umeclidinium bromide | 869113-09-7 | >98.00% | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC14096 | Aclidinium Bromide | 320345-99-1 | >98.00% | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC14215 | Cevimeline | 107233-08-9 | >98.00% | |
Cevimeline是一种强效的直接作用muscarinic受体激动剂，具有口服生物利用度。 | ||||
| GC15772 | Darifenacin HBr | 133099-07-7 | >98.00% | |
A muscarinic M 3 receptor antagonist | ||||
| GC16087 | Fesoterodine Fumarate | 286930-03-8 | - | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC17157 | Cevimeline hydrochloride hemihydrate | 153504-70-2 | >98.00% | |
Cevimeline hydrochloride hemihydrate (SNI-2011) 是乙酰胆碱的奎宁环衍生物，是一种选择性和口服活性的毒蕈碱 M1 和 M3 受体激动剂。 | ||||
| GC17182 | Solifenacin succinate | 242478-38-2 | >99.00% | |
A muscarinic M 1 , M 2 , and M 3 receptor antagonist | ||||
| GC17954 | Tolterodine tartrate | 124937-52-6 | >99.50% | |
A muscarinic acetylcholine receptor antagonist | ||||
| GC10219 | AF-DX 116 | 102394-31-0 | >99.50% | |
A muscarinic M 2 receptor antagonist | ||||
| GC10378 | N-Isopropylnoratropine | 22235-81-0 | - | |
An intermediate in the synthesis of ipratropium | ||||
| GC10464 | VU 0255035 | 1135243-19-4 | - | |
A selective muscarinic M 1 receptor antagonist | ||||
| GC10525 | Nitrocaramiphen hydrochloride | 98636-73-8 | - | |
M1 muscarinic antagonist | ||||
| GC10633 | DAU 5884 hydrochloride | 131780-48-8 | - | |
muscarinic M3 receptor antagonist | ||||
| GC10725 | VU 10010 | 633283-39-3 | >98.50% | |
VU 10010 是一种有效的、高选择性的变构 M4 mAChR 增强剂，EC50 为 400 nM。 | ||||
| GC10736 | (+)-Muscarine iodide | 24570-49-8 | - | |
毒蕈碱 ((+)-Muscarine) 碘化物是一种可以刺激副交感神经系统的毒素。 | ||||
| GC11415 | Arecaidine but-2-ynyl ester tosylate | 119630-77-2 | >98.00% | |
Arecaidine but-2-ynyl ester tosylate是一种选择性的毒蕈碱型乙酰胆碱受体（mAChR）M2激动剂。 | ||||
| GC12056 | J 104129 fumarate | 244277-89-2 | - | |
M3 muscarinic receptor antagonist | ||||
| GC12311 | Trihexyphenidyl hydrochloride | 52-49-3 | >99.50% | |
A muscarinic M 1 receptor antagonist | ||||
| GC12787 | Aceclidine (hydrochloride) | 6109-70-2 | >95.00% | |
A muscarinic receptor agonist | ||||
| GC13129 | W-84 dibromide | 21093-51-6 | >98.00% | |
W-84 (dibromide) 是一种有效的 M2-胆碱受体变构调节剂，可延缓 [3H]N-甲基东莨菪碱的解离。 | ||||
| GC13174 | Telenzepine dihydrochloride | 147416-96-4 | - | |
Telenzepine dihydrochloride 是一种选择性和口服活性的毒蕈碱 M1 受体拮抗剂，Ki 为 0.94 nM。 | ||||
| GC13340 | AQ-RA 741 | 123548-16-3 | - | |
M2 antagonist,selective and high affinity | ||||
| GC13348 | 4-DAMP | 1952-15-4 | >95.00% | |
An antagonist of the muscarinic M 3 receptor | ||||