Signaling Pathways
Signaling Pathways(信号通路)
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Signaling Pathways 相关产品(35130)
- GC15879Resminostat (RAS2410)CAS: 864814-88-0
Resminostat (RAS2410) (RAS2410; 4SC-201) 是一种有效的 HDAC1、HDAC3 和 HDAC6 抑制剂,平均 IC50 值分别为 42.5、50.1、71.8 nM,对 HDAC8 的活性较低,IC50 为 877 nM .
- GC15944(-)-U-50488 hydrochlorideCAS: 114528-79-9纯度: >99.00% / >98.00%
(-)-U-50488 hydrochloride((-)-U-50488盐酸盐)是一种选择性kappa阿片受体(KOR)激动剂,IC 50 值为 0.25μM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15847 | Ciproxifan maleate | 184025-19-2 | >99.00% | |
A histamine H 3 receptor antagonist | ||||
| GC15848 | Torcetrapib | 262352-17-0 | >99.00% | |
A CETP inhibitor | ||||
| GC15853 | Genz-644282 | 529488-28-6 | >98.50% | |
An inhibitor of topoisomerase I | ||||
| GC15860 | Ibutilide Fumarate | 122647-32-9 | >98.00% | |
A class III antiarrhythmic drug | ||||
| GC15864 | CCT128930 | 885499-61-6 | >99.50% | |
An inhibitor of Akt2 | ||||
| GC15873 | Adrafinil | 63547-13-7 | - | |
Wakefulness-promoting agent;modafinil analog | ||||
| GC15875 | ABT-751 (E7010) | 141430-65-1 | >99.50% | |
An inhibitor of microtubule polymerization | ||||
| GC15879 | Resminostat (RAS2410) | 864814-88-0 | - | |
Resminostat (RAS2410) (RAS2410; 4SC-201) 是一种有效的 HDAC1、HDAC3 和 HDAC6 抑制剂,平均 IC50 值分别为 42.5、50.1、71.8 nM,对 HDAC8 的活性较低,IC50 为 877 nM . | ||||
| GC15885 | (±)-U-50488 hydrochloride | 67197-96-0 | >98.00% | |
An Analytical Reference Material | ||||
| GC15889 | SANT-1 | 304909-07-7 | >99.50% | |
An antagonist of Smoothened | ||||
| GC15890 | Cilostazol | 73963-72-1 | >99.50% | |
A PDE3A inhibitor | ||||
| GC15891 | Nesbuvir | 691852-58-1 | >98.50% | |
Nesbuvir 是丙型肝炎病毒 (HCV) 非结构蛋白 5B (NS5B) 聚合酶的非核苷抑制剂。 | ||||
| GC15901 | Niclosamide monohydrate | 73360-56-2 | - | |
An anthelmintic mitochondrial uncoupler | ||||
| GC15903 | CYM 50308 | 1345858-76-5 | >98.00% | |
A selective S1P 4 receptor agonist | ||||
| GC15908 | AM-095 free base | 1228690-36-5 | >99.00% | |
A selective LPA 1 receptor antagonist | ||||
| GC15918 | Formoterol Hemifumarate | 43229-80-7 | >98.50% | |
强效、选择性和长效 β2-肾上腺素能受体激动剂 | ||||
| GC15920 | Besifloxacin HCl | 405165-61-9 | >98.50% | |
An ophthalmologic fluoroquinolone antibiotic | ||||
| GC15926 | BAN ORL 24 | 475150-69-7 | >98.00% | |
A nociceptin receptor antagonist | ||||
| GC15928 | Phenacetin | 62-44-2 | >99.50% | |
An Analytical Reference Standard | ||||
| GC15932 | BMN 673 | 1207456-01-6 | >98.50% | |
BMN 673是一种新型且高效的聚ADP核糖聚合酶1和2(PARP1/2)抑制剂,对PARP1的K i 为1.2nM,对PARP2的K i 为0.87nM。 | ||||
| GC15934 | Guanethidine Sulfate | 645-43-2 | >98.00% | |
An antihypertensive agent | ||||
| GC15936 | MSDC-0160 | 146062-49-9 | >99.00% | |
A thiazolidinedione | ||||
| GC15941 | EVP-6124 | 550999-75-2 | - | |
A partial agonist of α7 subunit-containing nAChRs | ||||
| GC15944 | (-)-U-50488 hydrochloride | 114528-79-9 | >99.00% / >98.00% | |
(-)-U-50488 hydrochloride((-)-U-50488盐酸盐)是一种选择性kappa阿片受体(KOR)激动剂,IC 50 值为 0.25μM。 | ||||
