Cell Cycle/Checkpoint
Cell Cycle/Checkpoint(细胞周期/检查点)
Cell Cycle
Cells undergo a complex cycle of growth and division that is referred to as the cell cycle. The cell cycle consists of four phases, G1 (GAP 1), S (synthesis), G2 (GAP 2) and M (mitosis). DNA replication occurs during S phase. When cells stop dividing temporarily or indefinitely, they enter a quiescent state called G0. read more
- ATM/ATR(29)
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- Cyclin-Dependent Kinases(77)
- E1 enzyme(1)
- G-quadruplex(12)
- Haspin(6)
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- Mps1(15)
- Mitotic(7)
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- ROCK(74)
- Rho(13)
- PERK(11)
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- Wee1(9)
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- Arp2/3 Complex(8)
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- Cytoskeleton & Motor Proteins(65)
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- G2/M(40)
- G2/S(17)
- Inositol Phosphates(67)
- Proteolysis(183)
- Cellular Chaperones(14)
- Cyclin G-associated Kinase (GAK)(1)
- MARK(3)
- NEKs(1)
Cell Cycle/Checkpoint 相关产品(1379)
- GC426167-oxo StaurosporineCAS: 125035-83-8纯度: >98.00%
An antibiotic with diverse biological activities
- GC42683Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnpCAS: 824405-61-0纯度: >95.00%
A sensitive substrate for neutrophil elastase
- GC42684Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp (trifluoroacetate salt)纯度: >98.80% / >98.50%
Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp (trifluoroacetate salt)是一种含有荧光共振能量转移(FRET)基团的修饰多肽。
- GC42715Ac-VDVAD-CHO (trifluoroacetate salt)纯度: >95.00%
A caspase-2, caspase-3, and caspase-7 inhibitor
- GC42719Ac-WEAD-pNA (trifluoroacetate salt)纯度: >95.00%
A colorimetric caspase-1 and caspase-4 substrate
- GC42721Ac-YVAD-CMKCAS: 178603-78-6纯度: >98.00%
Ac-YVAD-CMK 是一种选择性不可逆的 caspase-1 抑制剂 (Ki=0.8nM),可阻止促炎细胞因子 IL-1β 的激活。
- GC42788Aminopeptidase N InhibitorCAS: 596108-59-7纯度: >95.00%
Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM).
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC42548 | 5-hydroxy Saxagliptin (hydrochloride) | - | >95.00% | |
A major active metabolite of saxagliptin | ||||
| GC42586 | 6α-hydroxy Paclitaxel | 153212-75-0 | >95.00% | |
A metabolite of paclitaxel | ||||
| GC42610 | 7-hydroxy Pestalotin | 41164-59-4 | >99.00% | |
A fungal metabolite | ||||
| GC42616 | 7-oxo Staurosporine | 125035-83-8 | >98.00% | |
An antibiotic with diverse biological activities | ||||
| GC42665 | AAF-CMK (trifluoroacetate salt) | 184901-82-4 | >95.00% | |
An inhibitor of TPPII | ||||
| GC42683 | Abz-Ala-Pro-Glu-Glu-Ile-Met-Arg-Arg-Gln-EDDnp | 824405-61-0 | >95.00% | |
A sensitive substrate for neutrophil elastase | ||||
| GC42684 | Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp (trifluoroacetate salt) | - | >98.80% / >98.50% | |
Abz-Val-Ala-Asp-Nva-Arg-Asp-Arg-Gln-EDDnp (trifluoroacetate salt)是一种含有荧光共振能量转移(FRET)基团的修饰多肽。 | ||||
| GC42687 | Ac-DMQD-AMC (trifluoroacetate salt) | - | >95.00% | |
A fluorogenic substrate for caspase-3 | ||||
| GC42688 | Ac-DMQD-CHO (trifluoroacetate salt) | - | >95.00% | |
An inhibitor of caspase-3 | ||||
| GC42689 | Ac-DNLD-AMC | 958001-92-8 | >95.00% | |
A fluorogenic caspase-3 substrate | ||||
| GC42701 | Acetyl Tetrapeptide-3 | 827306-88-7 | >95.00% | |
A biomimetic peptide | ||||
| GC42706 | Ac-IEPD-AMC (trifluoroacetate salt) | - | >98.00% | |
A fluorogenic substrate for granzyme B | ||||
| GC42708 | Ac-LEHD-AFC (trifluoroacetate salt) | - | >95.00% | |
A caspase-4, -5, and -9 fluorogenic substrate | ||||
| GC42709 | Ac-LEVD-CHO (trifluoroacetate salt) | - | >95.00% | |
A caspase-4 inhibitor | ||||
| GC42715 | Ac-VDVAD-CHO (trifluoroacetate salt) | - | >95.00% | |
A caspase-2, caspase-3, and caspase-7 inhibitor | ||||
| GC42716 | Ac-VDVAD-pNA (trifluoroacetate salt) | - | >95.00% | |
A colorimetric caspase-2 substrate | ||||
| GC42718 | Ac-VEID-CHO (trifluoroacetate salt) | - | >95.00% | |
A caspase-6 inhibitor | ||||
| GC42719 | Ac-WEAD-pNA (trifluoroacetate salt) | - | >95.00% | |
A colorimetric caspase-1 and caspase-4 substrate | ||||
| GC42721 | Ac-YVAD-CMK | 178603-78-6 | >98.00% | |
Ac-YVAD-CMK 是一种选择性不可逆的 caspase-1 抑制剂 (Ki=0.8nM),可阻止促炎细胞因子 IL-1β 的激活。 | ||||
| GC42747 | Afuresertib (hydrochloride) | 1047645-82-8 | >98.00% | |
A pan-Akt inhibitor | ||||
| GC42788 | Aminopeptidase N Inhibitor | 596108-59-7 | >95.00% | |
Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM). | ||||
| GC42897 | BAY 61-3606 (hydrochloride) | 1615197-10-8 | >98.00% | |
A Syk inhibitor | ||||
| GC42933 | Binucleine 2 | 220088-42-6 | >98.00% | |
An inhibitor of Drosophila Aurora B kinase | ||||
| GC42936 | Biotin Tripeptide-1 | 299157-54-3 | >95.00% | |
An ECM peptide conjugated to biotin | ||||
