Chk
Chk(细胞周期检查点激酶)
Chk (Csk homologous kinase)
Chk 相关产品(13)
- GC16374MK-8776(SCH-900776)CAS: 891494-63-6纯度: >99.50%
MK-8776(SCH-900776) 是一种新型、选择性更高的Chk1抑制剂,旨在通过废除细胞周期阻滞来增强DNA损伤剂和抗代谢物的细胞毒性。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11648 | BML-277 | 516480-79-8 | >98.00% | |
A selective DNA damage control kinase inhibitor | ||||
| GC14234 | PF-477736 | 952021-60-2 | >99.00% | |
A selective inhibitor of checkpoint kinase 1 | ||||
| GC15663 | LY2606368 | 1234015-52-1 | >98.00% | |
LY2606368 是一种 ATP 竞争性 CHK1 抑制剂,目前处于临床阶段,Ki 为 0.9 nM,IC50 <1 nM。 | ||||
| GC15741 | LY2603618 | 911222-45-2 | >98.00% | |
A Chk1 inhibitor | ||||
| GC10546 | AZD7762 | 860352-01-8 | >99.50% | |
A selective checkpoint kinase inhibitor | ||||
| GC10793 | TCS 2312 | 838823-31-7 | - | |
checkpoint kinase 1 (chk1) inhibitor | ||||
| GC11022 | SB 218078 | 135897-06-2 | >98.00% | |
A potent Chk1 inhibitor | ||||
| GC13448 | NSC 109555 ditosylate | 66748-43-4 | - | |
An inhibitor of Chk2 | ||||
| GC14772 | CCT244747 | 1404095-34-6 | >99.00% | |
A potent Chk1 inhibitor | ||||
| GC15739 | CHIR-124 | 405168-58-3 | >98.00% | |
A selective Chk1 inhibitor | ||||
| GC16374 | MK-8776(SCH-900776) | 891494-63-6 | >99.50% | |
MK-8776(SCH-900776) 是一种新型、选择性更高的Chk1抑制剂,旨在通过废除细胞周期阻滞来增强DNA损伤剂和抗代谢物的细胞毒性。 | ||||
| GC17105 | CCT241533 hydrochloride | 1431697-96-9 | >99.00% | |
A selective Chk2 inhibitor | ||||
| GC18053 | CCT241533 | 1262849-73-9 | - | |
A selective Chk2 inhibitor | ||||
