DNA Damage/DNA Repair
DNA Damage/DNA Repair(DNA损伤/DNA修复)
- MTH1(4)
- PARP(124)
- ATM/ATR(29)
- DNA Alkylating(25)
- DNA Ligases(3)
- DNA Methyltransferase(32)
- DNA-PK(31)
- HDAC(182)
- Nucleoside Antimetabolite/Analogue(160)
- Telomerase(16)
- Topoisomerase(185)
- tankyrase(5)
- Antifolate(33)
- CDK(271)
- Checkpoint Kinase (Chk)(33)
- CRISPR/Cas9(9)
- Deubiquitinase(76)
- DNA Alkylator/Crosslinker(73)
- DNA/RNA Synthesis(473)
- Eukaryotic Initiation Factor (eIF)(27)
- IRE1(23)
- LIM Kinase (LIMK)(12)
- TOPK(6)
- Casein Kinase(48)
- DNA Intercalating Agents(8)
- DNA/RNA Oxidative Damage(13)
- Poly(ADP-ribose) Glycohydrolase (PARG)(1)
- Early 2 Factor (E2F)(1)
DNA Damage/DNA Repair 相关产品(1788)
- GC13249Rucaparib (free base)CAS: 283173-50-2纯度: >99.00%
Rucaparib (free base)是一种口服生物可利用的三环吲哚类聚(ADP-核糖)聚合酶(PARP)抑制剂。
- GC13704Mercaptopurine (6-MP)CAS: 50-44-2纯度: >99.00%
巯基嘌呤(6-MP)是一种嘌呤类似物,可作为内源性嘌呤的拮抗剂,被广泛用作抗白血病药和免疫抑制剂。
- GC14016SulforaphaneCAS: 4478-93-7纯度: >98.00% / >99.00% / >97.00%
萝卜硫素 (SFN) 称为 [1-isothiocyanato-4-(methylsulfinyl)butane]。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13070 | Cytarabine | 147-94-4 | >99.50% | |
Cytarabine(Ara-C)是一种胞嘧啶类似物,主要抑制DNA聚合酶的功能来阻断DNA合成。 | ||||
| GC13104 | 4E1RCat | 328998-25-0 | >98.00% | |
An eIF4F inhibitor | ||||
| GC13202 | D4476 | 301836-43-1 | >98.00% | |
Inhibitor of CK1 and ALK5 | ||||
| GC13208 | PR-619 | 2645-32-1 | >98.50% / >98.00% | |
PR-619是一种广谱的去泛素酶抑制剂。 | ||||
| GC13249 | Rucaparib (free base) | 283173-50-2 | >99.00% | |
Rucaparib (free base)是一种口服生物可利用的三环吲哚类聚(ADP-核糖)聚合酶(PARP)抑制剂。 | ||||
| GC13328 | XL413 hydrochloride | 2062200-97-7 | >99.50% | |
A potent inhibitor of Cdc7 | ||||
| GC13398 | RG 108 | 48208-26-0 | >99.50% | |
RG 108是一种强效的DNA甲基转移酶抑制剂,IC 50 值为115nM。 | ||||
| GC13399 | Trimidox | 95933-74-7 | - | |
A ribonucleotide reductase inhibitor | ||||
| GC13401 | SJB3-019A | 2070015-29-9 | >97.00% | |
SJB3-019A是一种新颖的、有效的USP1抑制剂,对K562细胞USP1的IC₅₀为0.0781μM。 | ||||
| GC13511 | THZ2 | 1604810-84-5 | >99.50% | |
A Cdk7 inhibitor | ||||
| GC13541 | G007-LK | 1380672-07-0 | >99.00% | |
G007-LK是一种有效的、选择性的TNKS1(IC 50 =46nM)和TNKS2(IC 50 =25nM)抑制剂。 | ||||
| GC13690 | BS-181 HCl | 1397219-81-6 | >99.00% | |
A selective Cdk7 inhibitor | ||||
| GC13704 | Mercaptopurine (6-MP) | 50-44-2 | >99.00% | |
巯基嘌呤(6-MP)是一种嘌呤类似物,可作为内源性嘌呤的拮抗剂,被广泛用作抗白血病药和免疫抑制剂。 | ||||
| GC13742 | Uridine | 58-96-8 | >99.50% | |
Uridine是一种核苷,包含尿嘧啶,通过β-N1-糖苷键与核糖环连接。 | ||||
| GC13764 | Nexturastat A | 1403783-31-2 | >98.00% | |
A potent, cell-permeable HDAC6 inhibitor | ||||
| GC13803 | Triflurdine (Viroptic) | 70-00-8 | >99.50% | |
A thymidine analog that inhibits DNA synthesis | ||||
| GC13825 | TA 01 | 1784751-18-3 | >99.50% | |
An inducer of cardiomyocyte differentiation | ||||
| GC13858 | Torin 2 | 1223001-51-1 | >99.50% | |
Selective inhibitor of mTOR | ||||
| GC13892 | C527 | 192718-06-2 | >99.50% | |
An inhibitor of the USP1/UAF complex | ||||
| GC13925 | Nullscript | 300816-11-9 | >98.00% | |
A negative control for scriptaid | ||||
| GC13978 | JW 74 | 863405-60-1 | >99.00% | |
An inhibitor of TNKS1/2 | ||||
| GC13998 | AT7519 Hydrochloride | 902135-91-5 | >99.00% | |
A Cdk inhibitor | ||||
| GC14016 | Sulforaphane | 4478-93-7 | >98.00% / >99.00% / >97.00% | |
萝卜硫素 (SFN) 称为 [1-isothiocyanato-4-(methylsulfinyl)butane]。 | ||||
| GC14058 | CBHA | 174664-65-4 | >98.00% | |
Inhibitor of histone deacetylases | ||||
