Drug Metabolite
Drug Metabolite(药物代谢物)
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Drug Metabolite 相关产品(498)
- GC20007Ginsenoside CKCAS: 39262-14-1纯度: >98.00%
Ginsenoside CK，一种由主要人参皂苷化合物转化而来的次级人参皂苷，比其母体人参皂苷具有更高的生物利用度和溶解性，具有极其重要的意义。
- GC30505N-Desmethyl Clomipramine D3 hydrochloride (Desmethylclomipramine D3 hydrochloride)CAS: 1189971-04-7
N-Desmethyl Clomipramine D3 hydrochloride (Desmethylclomipramine D3 hydrochloride) 是氘标记的 N-Desmethyl Clomipramine。
- GC30994Vanilpyruvic acid (Vanylpyruvic acid)CAS: 1081-71-6纯度: >98.00%
香草丙酮酸 (Vanylpyruvic acid) 是儿茶酚胺代谢物和香草乳酸的前体。
- GC31328Thyroxine sulfate (T4 Sulfate)CAS: 77074-49-8纯度: >99.50%
硫酸甲状腺素 (T4 Sulfate) 是一种甲状腺激素代谢物。
- GC32482Hydroxyhexamide ((±)-Hydroxyhexamid)CAS: 3168-01-2
Hydroxyhexamide is a pharmacologically active metabolite of acetohexamide, which is a sulfonylurea hypoglycemic agent.
- GC32518Norverapamil hydrochloride ((±)-Norverapamil hydrochloride)CAS: 67812-42-4纯度: >98.00%
An L-type calcium channel blocker
- GC32519Vinburnine ((-)-Eburnamonine)CAS: 4880-88-0纯度: >99.50%
Vinburnine ((-)-Eburnamonine, Vincamone, L-Eburnamonine) is a vasodilator. It is a vinca alkaloid and a metabolite of vincamine.
- GC32535Modecainide (BMY 40327)CAS: 81329-71-7
Modecainide (BMY 40327) 是 Encainide 的主要代谢物，Encainide 是一种抗心律失常药物。
- GC33333Regorafénib N-oxyde M2CAS: 835621-11-9纯度: >99.50%
Regorafénib N-oxyde M2是Regorafenib的一种活性代谢产物。
- GC33452Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1)CAS: 1476777-06-6纯度: >99.50%
Niraparib 代谢物 M1 (Niraparib carboxy acid metabolite M1) 是 niraparib 的代谢物，后者作为一种新型聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂。
- GC33484Ampyrone (4-Aminoantipyrine)CAS: 83-07-8
4-Aminoantipyrine(Ampyrone) is a metabolite of aminopyrine with analgesic, anti-inflammatory, and antipyretic properties. It is used as a reagent for biochemical reactions producing peroxides or phenols.
- GC33532Norgestimate metabolite Norelgestromin (17-Deacetyl norgestimate)CAS: 53016-31-2纯度: >99.50%
An active metabolite of norgestimate
- GC33548Netupitant metabolite Netupitant N-oxide (Netupitant N-oxide)CAS: 910808-11-6
A metabolite of netupitant
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC18622 | (2'S)-Nicotine-1-oxide | 2820-55-5 | - | |
A nicotine metabolite | ||||
| GC18632 | 6-hydroxy Bexarotene | 368451-07-4 | - | |
An oxidative metabolite of bexarotene | ||||
| GC18654 | 8-hydroxy Loxapine | 61443-77-4 | - | |
A loxapine metabolite | ||||
| GC18702 | Propiverine N-oxide (hydrochloride) | 1329509-71-8 | - | |
An active propiverine metabolite | ||||
| GC18831 | Tolmetin β-D-Glucuronide | 71595-19-2 | - | |
A major phase II metabolite of tolmetin | ||||
| GC19442 | 15-Acetyldeoxy Nivalenol | 88337-96-6 | - | |
A natural mycotoxin | ||||
| GC20007 | Ginsenoside CK | 39262-14-1 | >98.00% | |
Ginsenoside CK，一种由主要人参皂苷化合物转化而来的次级人参皂苷，比其母体人参皂苷具有更高的生物利用度和溶解性，具有极其重要的意义。 | ||||
| GC20062 | trans-3'-Hydroxycotinine | 34834-67-8 | >98.00% | |
A metabolite of nicotine | ||||
| GC30505 | N-Desmethyl Clomipramine D3 hydrochloride (Desmethylclomipramine D3 hydrochloride) | 1189971-04-7 | - | |
N-Desmethyl Clomipramine D3 hydrochloride (Desmethylclomipramine D3 hydrochloride) 是氘标记的 N-Desmethyl Clomipramine。 | ||||
| GC30994 | Vanilpyruvic acid (Vanylpyruvic acid) | 1081-71-6 | >98.00% | |
香草丙酮酸 (Vanylpyruvic acid) 是儿茶酚胺代谢物和香草乳酸的前体。 | ||||
| GC31328 | Thyroxine sulfate (T4 Sulfate) | 77074-49-8 | >99.50% | |
硫酸甲状腺素 (T4 Sulfate) 是一种甲状腺激素代谢物。 | ||||
| GC31734 | S-methyl-KE-298 (M-2) | 143584-75-2 | - | |
S-methyl-KE-298 (M-2) 是 KE-298 的活性代谢物。 | ||||
| GC32482 | Hydroxyhexamide ((±)-Hydroxyhexamid) | 3168-01-2 | - | |
Hydroxyhexamide is a pharmacologically active metabolite of acetohexamide, which is a sulfonylurea hypoglycemic agent. | ||||
| GC32518 | Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) | 67812-42-4 | >98.00% | |
An L-type calcium channel blocker | ||||
| GC32519 | Vinburnine ((-)-Eburnamonine) | 4880-88-0 | >99.50% | |
Vinburnine ((-)-Eburnamonine, Vincamone, L-Eburnamonine) is a vasodilator. It is a vinca alkaloid and a metabolite of vincamine. | ||||
| GC32535 | Modecainide (BMY 40327) | 81329-71-7 | - | |
Modecainide (BMY 40327) 是 Encainide 的主要代谢物，Encainide 是一种抗心律失常药物。 | ||||
| GC33072 | AZ7550 | 1421373-99-0 | - | |
An active metabolite of AZ 9291 | ||||
| GC33333 | Regorafénib N-oxyde M2 | 835621-11-9 | >99.50% | |
Regorafénib N-oxyde M2是Regorafenib的一种活性代谢产物。 | ||||
| GC33438 | Hydroxy Itraconazole | 112559-91-8 | >99.50% | |
A metabolite of itraconazole | ||||
| GC33452 | Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) | 1476777-06-6 | >99.50% | |
Niraparib 代谢物 M1 (Niraparib carboxy acid metabolite M1) 是 niraparib 的代谢物，后者作为一种新型聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂。 | ||||
| GC33484 | Ampyrone (4-Aminoantipyrine) | 83-07-8 | - | |
4-Aminoantipyrine(Ampyrone) is a metabolite of aminopyrine with analgesic, anti-inflammatory, and antipyretic properties. It is used as a reagent for biochemical reactions producing peroxides or phenols. | ||||
| GC33495 | N-Desmethyl imatinib | 404844-02-6 | >98.00% | |
A major active metabolite of imatinib | ||||
| GC33532 | Norgestimate metabolite Norelgestromin (17-Deacetyl norgestimate) | 53016-31-2 | >99.50% | |
An active metabolite of norgestimate | ||||
| GC33548 | Netupitant metabolite Netupitant N-oxide (Netupitant N-oxide) | 910808-11-6 | - | |
A metabolite of netupitant | ||||