Drug Metabolite
Drug Metabolite(药物代谢物)
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Drug Metabolite 相关产品(498)
- GC33558Acetaminophen metabolite 3-hydroxy-acetaminophen (3-Hydroxyacetaminophen)CAS: 37519-14-5纯度: >99.50% / >98.00%
Acetaminophen metabolite 3-hydroxy-acetaminophen (3-Hydroxyacetaminophen)是一种稳定的、羟基化的对乙酰氨基酚中间体。
- GC33559Netupitant metabolite Monohydroxy Netupitant (Monohydroxy Netupitant)CAS: 910808-12-7
Monohydroxy Netupitant 是 Netupitant 的代谢物，Netupitant 是一种高选择性的 NK1 受体拮抗剂。
- GC33563Netupitant metabolite N-desmethyl Netupitant (N-desmethyl Netupitant)CAS: 290296-72-9
N-desmethyl Netupitant 是 Netupitant 的代谢物，Netupitant 是一种止吐药。
- GC33571Duloxetine metabolite Para-Naphthol Duloxetine (Para-Naphthol duloxetine)CAS: 949095-98-1
对萘酚度洛西汀是度洛西汀的代谢产物，度洛西汀是一种血清素去甲肾上腺素再摄取抑制剂 (SNRI)。
- GC33578Ivabradine metabolite N-Demethyl Ivabradine hydrochlorideCAS: 1246638-08-3纯度: >99.00%
An active metabolite of ivabradine
- GC33579Carvedilol metabolite 4-Hydroxyphenyl CarvedilolCAS: 142227-49-4
An active metabolite of carvedilol
- GC33672Lurasidone Metabolite 14283 hydrochlorideCAS: 186204-32-0纯度: >99.00%
LurasidoneMetabolite14283hydrochloride是Lurasidone的主要的活性代谢物。
- GC337383-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride)CAS: 1477-68-5纯度: >98.00%
A natural metabolite of dopamine
- GC34027N-Acetylprocainamide (Acecainide)CAS: 32795-44-1纯度: >98.00%
N-Acetylprocainamide (Accecainide) 是一种 III 类抗心律失常药，可阻断 K+ 通道。
- GC34411Lurasidone Metabolite 14326 D8
LurasidoneMetabolite14326D8是LurasidoneMetabolite14326的氘代化合物标准品。
- GC34412Lurasidone metabolite 14326 hydrochloride
Lurasidonemetabolite14326(hydrochloride)是一种非典型抗精神病药物Lurasidone的活性代谢物。
- GC34413Lurasidone Metabolite 14283 D8
LurasidoneMetabolite14283D8是LurasidoneMetabolite14283的氘代化合物标准品。
- GC3507924, 25-Dihydroxy VD2CAS: 58050-55-8纯度: >99.50%
24, 25-Dihydroxy VD2 是一种维生素D2的羟基化代谢产物，是合成的维生素D类似物。
- GC350902-Hydroxy atorvastatin calcium saltCAS: 265989-46-6纯度: >98.00%
An active metabolite of atorvastatin
- GC35219Abiraterone metabolite 1CAS: 1940176-03-3纯度: >99.50%
Abiraterone metabolite 1 是 abiraterone 的 5β-还原代谢物。Abiraterone 是一种甾体药物，可抑制 CYP17A1，阻断雄激素的合成，延长前列腺癌的生存期。
- GC35780CycloguanilCAS: 516-21-2
Cycloguanil hydrochloride, an active metabolite of proguanil, acts on malaria schizonts in erythrocytes and hepatocytes.
- GC35990Endoxifen hydrochlorideCAS: 1197194-41-4纯度: >98.00%
Endoxifen hydrochloride 是 Tamoxifen 的活性代谢物，是有效的雌激素受体 (estrogen receptor) 拮抗剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC33558 | Acetaminophen metabolite 3-hydroxy-acetaminophen (3-Hydroxyacetaminophen) | 37519-14-5 | >99.50% / >98.00% | |
Acetaminophen metabolite 3-hydroxy-acetaminophen (3-Hydroxyacetaminophen)是一种稳定的、羟基化的对乙酰氨基酚中间体。 | ||||
| GC33559 | Netupitant metabolite Monohydroxy Netupitant (Monohydroxy Netupitant) | 910808-12-7 | - | |
Monohydroxy Netupitant 是 Netupitant 的代谢物，Netupitant 是一种高选择性的 NK1 受体拮抗剂。 | ||||
| GC33563 | Netupitant metabolite N-desmethyl Netupitant (N-desmethyl Netupitant) | 290296-72-9 | - | |
N-desmethyl Netupitant 是 Netupitant 的代谢物，Netupitant 是一种止吐药。 | ||||
| GC33564 | Lurasidone metabolite 14326 | 186204-33-1 | - | |
An active metabolite of lurasidone | ||||
| GC33571 | Duloxetine metabolite Para-Naphthol Duloxetine (Para-Naphthol duloxetine) | 949095-98-1 | - | |
对萘酚度洛西汀是度洛西汀的代谢产物，度洛西汀是一种血清素去甲肾上腺素再摄取抑制剂 (SNRI)。 | ||||
| GC33578 | Ivabradine metabolite N-Demethyl Ivabradine hydrochloride | 1246638-08-3 | >99.00% | |
An active metabolite of ivabradine | ||||
| GC33579 | Carvedilol metabolite 4-Hydroxyphenyl Carvedilol | 142227-49-4 | - | |
An active metabolite of carvedilol | ||||
| GC33672 | Lurasidone Metabolite 14283 hydrochloride | 186204-32-0 | >99.00% | |
LurasidoneMetabolite14283hydrochloride是Lurasidone的主要的活性代谢物。 | ||||
| GC33738 | 3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) | 1477-68-5 | >98.00% | |
A natural metabolite of dopamine | ||||
| GC34027 | N-Acetylprocainamide (Acecainide) | 32795-44-1 | >98.00% | |
N-Acetylprocainamide (Accecainide) 是一种 III 类抗心律失常药，可阻断 K+ 通道。 | ||||
| GC34287 | AZ7550 hydrochloride | 2309762-40-9 | - | |
An active metabolite of AZ 9291 | ||||
| GC34408 | Monohydroxy Netupitant D6 | - | - | |
MonohydroxyNetupitantD6是MonohydroxyNetupitant的氘代化合物标准品。 | ||||
| GC34409 | Netupitant N-oxide D6 | - | - | |
NetupitantN-oxideD6是NetupitantN-oxide的氘代化合物标准品。 | ||||
| GC34410 | N-desmethyl Netupitant D6 | - | - | |
N-desmethylNetupitantD6是N-desmethylNetupitant的氘代化合物标准品。 | ||||
| GC34411 | Lurasidone Metabolite 14326 D8 | - | - | |
LurasidoneMetabolite14326D8是LurasidoneMetabolite14326的氘代化合物标准品。 | ||||
| GC34412 | Lurasidone metabolite 14326 hydrochloride | - | - | |
Lurasidonemetabolite14326(hydrochloride)是一种非典型抗精神病药物Lurasidone的活性代谢物。 | ||||
| GC34413 | Lurasidone Metabolite 14283 D8 | - | - | |
LurasidoneMetabolite14283D8是LurasidoneMetabolite14283的氘代化合物标准品。 | ||||
| GC34414 | AZ7550 Mesylate (AZ7550 trimesylate salt) | - | - | |
An active metabolite of AZ 9291 | ||||
| GC35079 | 24, 25-Dihydroxy VD2 | 58050-55-8 | >99.50% | |
24, 25-Dihydroxy VD2 是一种维生素D2的羟基化代谢产物，是合成的维生素D类似物。 | ||||
| GC35090 | 2-Hydroxy atorvastatin calcium salt | 265989-46-6 | >98.00% | |
An active metabolite of atorvastatin | ||||
| GC35219 | Abiraterone metabolite 1 | 1940176-03-3 | >99.50% | |
Abiraterone metabolite 1 是 abiraterone 的 5β-还原代谢物。Abiraterone 是一种甾体药物，可抑制 CYP17A1，阻断雄激素的合成，延长前列腺癌的生存期。 | ||||
| GC35295 | Allopurinol riboside | 16220-07-8 | >98.00% | |
A ribonucleoside | ||||
| GC35780 | Cycloguanil | 516-21-2 | - | |
Cycloguanil hydrochloride, an active metabolite of proguanil, acts on malaria schizonts in erythrocytes and hepatocytes. | ||||
| GC35990 | Endoxifen hydrochloride | 1197194-41-4 | >98.00% | |
Endoxifen hydrochloride 是 Tamoxifen 的活性代谢物，是有效的雌激素受体 (estrogen receptor) 拮抗剂。 | ||||