Androgen Receptor
Androgen Receptor(雄激素受体)
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
Androgen Receptor 相关产品(148)
- GC46775Abiraterone Acetate-d4CAS: 2122245-63-8纯度: >99.00%
醋酸阿比特龙-d4 (CB7630-d4) 是氘标记的醋酸阿比特龙。醋酸阿比特龙 (CB7630) 是一种口服的、有效的、选择性的、不可逆的 CYP17A1 抑制剂,具有抗雄激素活性。醋酸阿比特龙是阿比特龙 (CB7598) 的前药形式。
- GC46925Bicalutamide-d4CAS: 1185035-71-5纯度: >99.00%
An internal standard for the quantification of bicalutamide
- GC47215Dienogest-d8CAS: 2376035-92-4纯度: >99.00%
An internal standard for the quantification of dienogest
- GC47554Letrozole-d4CAS: 1133712-96-5纯度: >99.00%
An internal standard for the quantification of letrozole
- GC488085β-Androstane-3α,17β-diolCAS: 1851-23-6纯度: >95.00%
A metabolite of testosterone
- GC49055Tebuconazole-d9CAS: 1246818-83-6纯度: >99.00%
An internal standard for the quantification of tebuconazole
- GC49303Ganoderic Acid DMCAS: 173075-45-1纯度: >98.00%
A triterpenoid with diverse biological activities
- GC49648Enobosarm-d4CAS: 1202044-20-9纯度: >99.00%
An internal standard for the quantification of enobosarm
- GC60589Apalutamide D4CAS: 1638885-65-0纯度: >99.00%
ApalutamideD4(ARN-509D4)是Apalutamide的一种氘代化合物。Apalutamide是有效,竞争性的雄激素受体(AR)拮抗剂,IC50为16nM。
- GC61481PROTAC AR Degrader-4 TFA纯度: >98.00%
PROTACARDegrader-4包含cIAP1配体结合基团,linker和雄激素受体(AR)配体结合基团。基于cIAP1的降解剂也被称为SNIPER。
- GC61491(R)-BicalutamideCAS: 113299-40-4纯度: >99.50%
(R)-Bicalutamide是Bicalutamide的R型对映体。(R)-Bicalutamide是一种雄激素受体(AR)拮抗剂,具有抗肿瘤活性。(R)-Bicalutamide广泛用于前列腺癌的研究。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC46471 | 17β-hydroxy Exemestane-d3 | - | >99.00% | |
A neuropeptide with diverse biological activities | ||||
| GC46775 | Abiraterone Acetate-d4 | 2122245-63-8 | >99.00% | |
醋酸阿比特龙-d4 (CB7630-d4) 是氘标记的醋酸阿比特龙。醋酸阿比特龙 (CB7630) 是一种口服的、有效的、选择性的、不可逆的 CYP17A1 抑制剂,具有抗雄激素活性。醋酸阿比特龙是阿比特龙 (CB7598) 的前药形式。 | ||||
| GC46777 | AC-262536 | 870888-46-3 | >98.00% | |
A selective androgen receptor modulator | ||||
| GC46925 | Bicalutamide-d4 | 1185035-71-5 | >99.00% | |
An internal standard for the quantification of bicalutamide | ||||
| GC47159 | Cyprodinil | 121552-61-2 | >99.00% | |
An anilinopyrimidine fungicide | ||||
| GC47215 | Dienogest-d8 | 2376035-92-4 | >99.00% | |
An internal standard for the quantification of dienogest | ||||
| GC47231 | Dimethomorph | 110488-70-5 | >97.00% | |
A morpholine fungicide | ||||
| GC47554 | Letrozole-d4 | 1133712-96-5 | >99.00% | |
An internal standard for the quantification of letrozole | ||||
| GC47674 | Mifepristone-d3 | - | >99.00% | |
A neuropeptide with diverse biological activities | ||||
| GC48724 | Pregnanetriol | 1098-45-9 | >95.00% | |
A metabolite of 17α-hydroxyprogesterone | ||||
| GC48808 | 5β-Androstane-3α,17β-diol | 1851-23-6 | >95.00% | |
A metabolite of testosterone | ||||
| GC48831 | Flutamide-d7 | 223134-72-3 | >99.00% | |
Flutamide-d7 是氘标记的氟他胺。 | ||||
| GC48880 | 7-Methoxyflavone | 22395-22-8 | >98.00% | |
A flavone with diverse biological activities | ||||
| GC49055 | Tebuconazole-d9 | 1246818-83-6 | >99.00% | |
An internal standard for the quantification of tebuconazole | ||||
| GC49303 | Ganoderic Acid DM | 173075-45-1 | >98.00% | |
A triterpenoid with diverse biological activities | ||||
| GC49391 | 7α-Thiospironolactone | 38753-76-3 | >90.00% | |
An active metabolite of spironolactone | ||||
| GC49520 | (S)-Equol | 531-95-3 | >98.00% | |
(S)-Equol是一种由部分人群肠道微生物产生的异黄烷类化合物,主要来源于大豆中的大豆素在特定肠道菌群的作用下生成。(S)-Equol具有显著的雌激素样活性和抗氧化特性,能够与雌激素受体结合,对 ERβ的亲和力为Ki=0.73±0.2nM,对ERα的亲和力为Ki=6.41±1nM。 | ||||
| GC49542 | 5α-Androstan-3β-ol | 1224-92-6 | >98.00% | |
A steroidal androgen | ||||
| GC49563 | Fenhexamid | 126833-17-8 | >98.00% | |
A fungicide | ||||
| GC49648 | Enobosarm-d4 | 1202044-20-9 | >99.00% | |
An internal standard for the quantification of enobosarm | ||||
| GC49827 | 5-Androstenetriol | 4150-30-5 | >98.00% | |
An active metabolite of DHEA | ||||
| GC60589 | Apalutamide D4 | 1638885-65-0 | >99.00% | |
ApalutamideD4(ARN-509D4)是Apalutamide的一种氘代化合物。Apalutamide是有效,竞争性的雄激素受体(AR)拮抗剂,IC50为16nM。 | ||||
| GC61481 | PROTAC AR Degrader-4 TFA | - | >98.00% | |
PROTACARDegrader-4包含cIAP1配体结合基团,linker和雄激素受体(AR)配体结合基团。基于cIAP1的降解剂也被称为SNIPER。 | ||||
| GC61491 | (R)-Bicalutamide | 113299-40-4 | >99.50% | |
(R)-Bicalutamide是Bicalutamide的R型对映体。(R)-Bicalutamide是一种雄激素受体(AR)拮抗剂,具有抗肿瘤活性。(R)-Bicalutamide广泛用于前列腺癌的研究。 | ||||
