关于 "Dopamine Receptor" 的结果56+ 个结果
- Dopamine serotonin antagonist-1CAS: 1977-07-7
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.
- N-Arachidonoyl Dopamine-d8CAS: 1159908-42-5
An internal standard for the quantification of N-arachidonoyl dopamine
- GABAA receptor agent 1CAS: 1571-87-5
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity.
- H4 Receptor antagonist 1CAS: 848217-00-5
H4Receptorantagonist1是一种有效的、有选择性的组胺H4受体(H4R)的反向激动剂，其IC50值为19nM。
- CCK-B Receptor Antagonist 2CAS: 155412-88-7
CCK-B Receptor Antagonist 2，化合物 15b，是有效的口服活性 Gastrin/CCK-B 拮抗剂，IC50 值为 0.43 nM。 CCK-B Receptor Antagonist 2 还抑制 Gastrin/CCK-A 活性，IC50 为 1.82 μM。
- AMPA receptor modulator-2CAS: 2034181-36-5
AMPA receptor modulator-2 (Example 134) 是 AMPA 受体的调节剂，对TARPγ2 依赖的AMPA 受体的 pIC50 值为 10.1。
- AMPA receptor modulator-3CAS: 211311-39-6
AMPA receptor modulator-3 是一种变构的 AMPA 受体调节剂 (EC50: 4.4 μM)。AMPA receptor modulator-3 可用于哺乳动物神经系统的研究，如学习和记忆能力。
- CCK-A receptor inhibitor 1CAS: 137004-80-9
CCK-Areceptorinhibitor1是一种缩胆囊素A(cholecystokininA,CCK-A)受体抑制剂，IC50为340nM。
- α7 Nicotinic receptor agonist-1CAS: 220100-05-0
α7 Nicotinic receptor agonist-1 (Preparation 5) 是一种 α7 nAChR 激动剂。α7 Nicotinic receptor agonist-1 可用于精神障碍 (如精神分裂症、躁狂或躁狂抑郁症和焦虑症) 和智力障碍 (如阿尔茨海默氏病、学习缺陷、认知缺陷、注意力缺陷、记忆丧失、路易体痴呆和注意力缺陷多动症) 的研究。
- CCK-B Receptor Antagonist 1CAS: 168161-71-5
CCK-B Receptor Antagonist 1 是胆囊收缩素 B (CCK-B) 受体的拮抗剂，具有减少胃酸分泌的潜力。
- NK1 receptor antagonist 2CAS: 579475-17-5
NK1 receptor antagonist 2 是一种 NK1 受体拮抗剂。NK1 receptor antagonist 2 可用于耳鸣和听力损失的研究。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC62940 | Dopamine | 51-61-6 | Dopamine Receptor | ||
An endogenous catecholamine | |||||
| GC11028 | Dopamine HCl | 62-31-7 | Dopamine Receptor | ||
An endogenous catecholamine | |||||
| GC18506 | N-Arachidonoyl Dopamine | 199875-69-9 | Cancer Biology | ||
An arachidonoyl amino acid and CB1 receptor agonist | |||||
| GC44706 | Prostaglandin D2 Dopamine | - | Prostaglandins | ||
A neurotransmitter/fatty acid conjugate | |||||
| GC49497 | Dopamine-d4 (hydrochloride) | 203633-19-6 | Analytical Standards | ||
An internal standard for the quantification of dopamine | |||||
| GC30772 | Dopamine serotonin antagonist-1 | 1977-07-7 | Serotonin Transporter | ||
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively. | |||||
| GC47748 | N-Arachidonoyl Dopamine-d8 | 1159908-42-5 | Cancer Biology | ||
An internal standard for the quantification of N-arachidonoyl dopamine | |||||
| GC49516 | Dopamine 4-O-Sulfate | 38339-02-5 | Neuroscience | ||
An inactive metabolite of dopamine | |||||
| GC49166 | Dopamine 3-O-Sulfate | 51317-41-0 | Neuroscience | ||
A metabolite of dopamine | |||||
| GC43083 | C3a Receptor Agonist | 944997-60-8 | Neuroscience | ||
C3a Receptor Agonist是一种选择性的补体3a受体（C3aR）特异性激动剂。 | |||||
| GC60862 | GABAA receptor agent 1 | 1571-87-5 | GABA Receptor | ||
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity. | |||||
| GC39554 | AT2 receptor agonist C21 | 477775-14-7 | Cardiomyopathy | ||
An AT2 receptor agonist | |||||
| GC30759 | H3 receptor-MO-1 | 1240914-03-7 | Histamine Receptor | ||
H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。 | |||||
| GC31310 | H3 receptor antagonist 1 | 935840-13-4 | Histamine Receptor | ||
H3receptorantagonist1是组胺H3(histamineH3)受体拮抗剂，可用于神经疾病的研究。 | |||||
| GC31984 | M3 receptor antagonist 1 | 1004312-94-0 | mAChR | ||
M3 受体拮抗剂 1 是一种选择性、长效和竞争性毒蕈碱 M3 受体拮抗剂。 | |||||
| GC31232 | H4 Receptor antagonist 1 | 848217-00-5 | Histamine Receptor | ||
H4Receptorantagonist1是一种有效的、有选择性的组胺H4受体(H4R)的反向激动剂，其IC50值为19nM。 | |||||
| GC38746 | CCK-B Receptor Antagonist 2 | 155412-88-7 | Cholecystokinin Receptor | ||
CCK-B Receptor Antagonist 2，化合物 15b，是有效的口服活性 Gastrin/CCK-B 拮抗剂，IC50 值为 0.43 nM。 CCK-B Receptor Antagonist 2 还抑制 Gastrin/CCK-A 活性，IC50 为 1.82 μM。 | |||||
| GC62840 | AMPA receptor modulator-2 | 2034181-36-5 | iGluR | ||
AMPA receptor modulator-2 (Example 134) 是 AMPA 受体的调节剂，对TARPγ2 依赖的AMPA 受体的 pIC50 值为 10.1。 | |||||
| GC68438 | AMPA receptor modulator-3 | 211311-39-6 | iGluR | ||
AMPA receptor modulator-3 是一种变构的 AMPA 受体调节剂 (EC50: 4.4 μM)。AMPA receptor modulator-3 可用于哺乳动物神经系统的研究，如学习和记忆能力。 | |||||
| GC31558 | CCK-A receptor inhibitor 1 | 137004-80-9 | Cholecystokinin Receptor | ||
CCK-Areceptorinhibitor1是一种缩胆囊素A(cholecystokininA,CCK-A)受体抑制剂，IC50为340nM。 | |||||
| GC70179 | α7 Nicotinic receptor agonist-1 | 220100-05-0 | nAChR | ||
α7 Nicotinic receptor agonist-1 (Preparation 5) 是一种 α7 nAChR 激动剂。α7 Nicotinic receptor agonist-1 可用于精神障碍 (如精神分裂症、躁狂或躁狂抑郁症和焦虑症) 和智力障碍 (如阿尔茨海默氏病、学习缺陷、认知缺陷、注意力缺陷、记忆丧失、路易体痴呆和注意力缺陷多动症) 的研究。 | |||||
| GC30752 | CCK-B Receptor Antagonist 1 | 168161-71-5 | Cholecystokinin Receptor | ||
CCK-B Receptor Antagonist 1 是胆囊收缩素 B (CCK-B) 受体的拮抗剂，具有减少胃酸分泌的潜力。 | |||||
| GC30836 | MK-7622 (M1 receptor modulator) | 1227923-29-6 | mAChR | ||
A positive allosteric modulator of M1 mAChRs | |||||
| GC69568 | NK1 receptor antagonist 2 | 579475-17-5 | Neurokinin Receptor | ||
NK1 receptor antagonist 2 是一种 NK1 受体拮抗剂。NK1 receptor antagonist 2 可用于耳鸣和听力损失的研究。 | |||||