Home >> Proteins

Proteins(蛋白质)

  1. Cat.No. 产品名称 Information
  2. GC70181 α-Glucosidase-IN-22 α-Glucosidase-IN-22 (compound 7i) 是一种苯并咪唑,一种有效的 α-葡萄糖苷酶 (α-glucosidase) 抑制剂,IC50 为 0.64 μM。α-Glucosidase-IN-22 是一种有效的抗糖尿病活性分子,具有用于 2 型糖尿病 (T2DM) 研究的潜力。
  3. GC72710 α-Glucosidase-IN-35 α-Glucosidase-IN-35(化合物1)是一种苯并二氢吡喃。
  4. GC48292 α-MSH (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)

    Α-促黑激素,α-Melanocyte-Stimulating Hormone TFA

    A peptide hormone
  5. GC92108 α-MSH Acid (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)

    N-acetyl ACTH (1-13); N-acetyl Adrenocorticotropic Hormone (1-13); α-Melanocyte-stimulating Hormone Acid

    α-MSH Acid (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)α-MSH酸是α-MSH的酸形式。
  6. GC68390 α5β1 integrin agonist-1 α5β1 integrin agonist-1 作为 α5β1 integrin 激动剂,能够选择性地将 5-FU 输送到肿瘤细胞中,成功地导致肿瘤细胞死亡。
  7. GC62380 αvβ1 integrin-IN-1 αvβ1 integrin-IN-1 (Compound C8) 是一种有效的选择性 αvβ1 整合素抑制剂,IC50 为 0.63 nM。具有抗纤维化作用。
  8. GC62566 αvβ1 integrin-IN-1 TFA αvβ1 integrin-IN-1 TFA (Compound C8) 是一种有效的选择性 αvβ1 整合素抑制剂,IC50 为 0.63 nM。具有抗纤维化作用。
  9. GC64932 αvβ5 integrin-IN-1 αvβ5 integrin-IN-1 是第一个有效和选择性 αvβ5 整合素抑制剂(pIC50 = 8.2)。
  10. GC48920 β-Carboline-1-carboxylic Acid

    1-Formic Acid-β-carboline

    An alkaloid with diverse biological activities
  11. GC62551 β-Hydroxypropiovanillone

    3,4'-二羟基-3'-甲氧基苯丙酮

    β-Hydroxypropiovanillone 是一种天然化合物,对 α-葡萄糖苷酶 (α-glucosidase) 具有明显的浓度依赖性抑制作用 (IC50=257.8 μg/mL)。
  12. GC41502 β-Myrcene

    月桂烯; β-Myrcene

    A terpene with antioxidative properties
  13. GC92102 γ1-MSH (human, mouse, rat, bovine) (acetate)

    γ1-Melanocyte-stimulating Hormone

    γ1-MSH (human, mouse, rat, bovine) (acetate)是一种肽激素,由垂体中的前皮黑皮质素(POMC)翻译后加工产生。
  14. GC92101 γ1-MSH (human, mouse, rat, bovine) (trifluoroacetate salt)

    γ1-Melanocyte-stimulating Hormone

    γ1-MSH (human, mouse, rat, bovine) (trifluoroacetate salt)是一种肽激素,由垂体中的前皮黑皮质素(POMC)翻译后加工产生。
  15. GC45270 (±)10(11)-EDP Ethanolamide

    10,11-EDP-EA, 10,11-EDP epoxide, 10,11-epoxy Docosapentaenoic Ethanolamide

    An ω-3 endocannabinoid epoxide and CB receptor agonist
  16. GC40802 (±)12(13)-DiHOME

    Isoleukotoxin diol

    A diol form of (±)12,13-EpOME
  17. GC41648 (±)13(14)-DiHDPA

    13(14)-DiHDPA, 13(14)-DiHDoPE, 13,14-DiHDPE

    A metabolite of DHA
  18. GC41653 (±)16(17)-DiHDPA An epoxygenase metabolite of DHA
  19. GC41655 (±)19(20)-EDP Ethanolamide

    19,20-DHEA epoxide, 19,20-epoxy Docosapentaenoic Acid Ethanolamide, 19,20-EDP-EA, 19,20-EDP epoxide

    An ω-3 endocannabinoid epoxide and CB receptor agonist
  20. GC40801 (±)9(10)-DiHOME

    (±)-苏式-9,10-二羟基-12(Z)-十八碳烯酸

    A diol form of (±)9(10)-EpOME
  21. GC18516 (+)-Aeroplysinin-1

    (+)-Aeroplysinin-1

    A sea sponge metabolite with diverse biological activities
  22. GC39795 (+)-Afzelechin

    (+)-阿夫儿茶精

    (+)-Afzelechin 是从佛手根的根茎中分离出来的,是一种 α-葡萄糖苷酶 (alpha-glucosidase) 活性抑制剂,ID50 值为 0.13 mM。(+)-Afzelechin 可以延迟食物中碳水化合物的吸收,从而抑制餐后高血糖和高胰岛素血症。
  23. GC45266 (+)-Macrosphelide A A fungal metabolite
  24. GC18749 (+)-Rugulosin

    细皱青霉素+FORM,(+)-Rugulosin

    A mycotoxin
  25. GC17102 (-)-Tetramisole

    盐酸左旋咪唑

    An Analytical Reference Material
  26. GC65363 (1R)-Tenofovir amibufenamide

    (1R)-HS-10234

    (1R)-Tenofovir amibufenamide ((1R)-HS-10234) 是 Tenofovir amibufenamide 的异构体,是一种口服活性抗病毒药物。(1R)-Tenofovir amibufenamide ((1R)-HS-10234) 是一个 HIV 病毒感染的抑制剂和乙型肝炎病毒的抑制剂 ( HBV )。(1R)-Tenofovir amibufenamide ((1R)-HS-10234) 可用于 HIV 感染、乙肝研究。
  27. GC65547 (1S,2R)-Alicapistat

    (1S,2R)-ABT-957

    (1S,2R)-Alicapistat ((1S,2R)-ABT-957) 是一种具有口服活性的人钙激活中性蛋白酶 (calpains 1 和 2) 的选择性抑制剂,可能用于阿尔茨海默病 (AD) 的研究。 Alicapistat 可减轻羰基还原的代谢倾向,对 calpain 1 的 IC50 为 395 nM。
  28. GC62193 (1S,2S)-Bortezomib

    硼替佐米杂质E

    (1S,2S)-Bortezomib 是 Bortezomib 的对映异构体。Bortezomib 是一种细胞渗透性、可逆性和选择性的蛋白酶体抑制剂,通过靶向苏氨酸残基有效抑制 20S 蛋白酶体 (Ki 为 0.6 nM)。Bortezomib 破坏细胞周期、诱导细胞凋亡以及抑制核因子 NF-κB。Bortezomib 是一种抗癌药物,也是第一种用于人类的蛋白酶体抑制剂。
  29. GC68525 (2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid (2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid 是一种可从 Rubus ellipticus var. obcordatus 中分离得到的皂苷。(2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid 抑制 α-Glucosidase,其 IC50 为 1.68 mM。
  30. GC64260 (2S,5S)-Censavudine

    (2S,5S)-OBP-601; (2S,5S)-BMS-986001

    (2S,5S)-Censavudine ((2S,5S)-OBP-601) 是 Censavudine 的 (2S,5S)-对映异构体。Censavudine 是一种核苷类逆转录酶抑制剂,是一种有效的 HIV 抑制剂。
  31. GC40444 (5Z,11Z,15R)-15-Hydroxyeicosa-5,11-dien-13-ynoic Acid

    HETE Analog 1, Hydroxyeicosatetraenoic Acid Analog 1

    A stable isomer of 15(S)-HETE
  32. GC92107 (D-Phe7)-α-MSH (trifluoroacetate salt)

    (D-Phe7)-α-Melanocyte-stimulating Hormone

    (D-Phe7)-α-MSH (trifluoroacetate salt) ((D-Phe7)-α-MSH)是α-MSH的肽衍生物,是合成α-MSH环类似物的中间体。
  33. GC41699 (Des-octanoyl)-Ghrelin (human) (trifluoroacetate salt) A peptide hormone
  34. GC41700 (E)-2-(2-Chlorostyryl)-3,5,6-trimethylpyrazine

    CSTMP

    A stilbene derivative with antioxidant and anticancer activities
  35. GC62735 (E/Z)-GO289 (E/Z)-GO289 potently and selectively inhibits casein kinase 2 (CK2) at an IC50 of 7 nM in vitro kinase assay.
  36. GC49167 (R)-(+)-Trityl glycidyl ether

    三苯甲基-(R)-缩水甘油醚

    A synthetic precursor
  37. GC41620 (R)-(-)-Mellein

    (R)-蜂蜜曲菌素,以及(S)-蜂蜜曲菌素,(R)-Mellein

    A dihydroisocoumarin compound with antibacterial, antimalarial, antifungal , and anticancer effects
  38. GC74184 (R)-Azasetron besylate

    SENS-401

    (R)-Azasetron besylateSENS-401是一种口服活性钙调神经磷酸酶抑制剂。
  39. GC69837 (R/S)-Alicaforsen

    (R/S)-ISIS-2302

    (R/S)-Alicaforsen 是由R和S构型组成的 Alicaforsen 的消旋体。Alicaforsen是一种20个碱基长度的反义寡核苷酸,抑制 ICAM-1 的产生,ICAM-1 是一种重要的粘附分子,参与白细胞向炎症部位迁移和转运的过程。
  40. GC46351 (S)-CR8 An inhibitor of cyclin-dependent kinases
  41. GC64535 (S,S)-TAPI-1

    TAPI

    A TACE inhibitor
  42. GC45978 1,10-Phenanthroline (hydrate)

    邻菲罗啉,1,10-Phenanthroline monohydrate

    A metal chelator and inhibitor of metalloproteases
  43. GC41774 1,2,3-Trimyristoyl-rac-glycerol

    三肉豆蔻酸甘油酯

    A triacylglycerol
  44. GC90744 1,2-Dioleoyl-3(R)-trimethylammoniumpropane (chloride)

    R-DOTAP

    一个阳离子脂质

  45. GC49294 1-(4-Chlorobenzhydryl)piperazine

    1-(4-氯二苯甲基)哌嗪

    An inactive metabolite of meclizine and chlorcyclizine
  46. GC41992 1-Deoxynojirimycin (hydrochloride)

    去氧野艽霉素盐酸盐,Duvoglustat hydrochloride

    An iminosugar with diverse biological activities
  47. GC41998 1-Methyl-4-imidazoleacetic Acid (hydrochloride)

    1-甲基-4-羧酸咪唑盐酸盐

    A stable metabolite of histamine
  48. GC25005 1-Naphthyl phosphate potassium salt

    α-Naphthyl acid phosphate monopotassium salt

    1-Naphthyl phosphate potassium salt (α-Naphthyl acid phosphate monopotassium salt) is a non-specific phosphatase inhibitor which acts on acid, alkaline, and protein phosphatases.
  49. GC42026 1-Palmitoyl-2-hydroxy-sn-glycero-3-PC

    1-十六酰-SN-丙三醇-磷酸胆碱

    A product of PLA2-mediated hydrolysis of phosphatidylcholine
  50. GC46490 1-Palmitoyl-d3-2-hydroxy-sn-glycero-3-PC

    1-Hexadecanoyl-sn-glycero-3-Phosphatidylcholine-d3, 1-Hexadecanoyl-sn-glycero-3-Phosphocholine-d3, LPC-d3, 16:0/0:0(d3) Lyso-PC, 1-Palmitoyl-sn-glycero-3-Phosphocholine-d3, PC(16:0/0:0)-d3, 16:0/0:0-PC-d3

    A neuropeptide with diverse biological activities
  51. GC45693 1-Palmitoyl-d9-2-hydroxy-sn-glycero-3-PC

    1-Hexadecanoyl-d9-sn-glycero-3-Phosphatidylcholine, 1-Hexadecanoyl-d9-sn-glycero-3-Phosphocholine, 16:0(d9) Lyso-PC, PC(16:0-d9/0:0), 16:0-d9/0:0-PC

    An internal standard for the quantification of 1-palmitoyl-2-hydroxy-sn-glycero-3-PC

Items 1 to 50 of 6998 total

per page
  1. 1
  2. 2
  3. 3
  4. 4
  5. 5

Set Descending Direction