Proteins(蛋白质)
- Chemokines(173)
- Cytokines(632)
- Enzymes(1726)
- Growth Factors(507)
- Hormones(214)
- Natural Proteins(58)
- Neurotrophins(74)
- Recombinant Proteins(2695)
- Viral Antigens(718)
- CD Antigens(200)
- Cat.No. 产品名称 Information
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GC70181
α-Glucosidase-IN-22
α-Glucosidase-IN-22 (compound 7i) 是一种苯并咪唑,一种有效的 α-葡萄糖苷酶 (α-glucosidase) 抑制剂,IC50 为 0.64 μM。α-Glucosidase-IN-22 是一种有效的抗糖尿病活性分子,具有用于 2 型糖尿病 (T2DM) 研究的潜力。
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GC72710
α-Glucosidase-IN-35
α-Glucosidase-IN-35(化合物1)是一种苯并二氢吡喃。
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GC48292
α-MSH (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)
Α-促黑激素,α-Melanocyte-Stimulating Hormone TFA
A peptide hormone -
GC92108
α-MSH Acid (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)
N-acetyl ACTH (1-13); N-acetyl Adrenocorticotropic Hormone (1-13); α-Melanocyte-stimulating Hormone Acid
α-MSH Acid (human, mouse, rat, porcine, bovine, ovine) (trifluoroacetate salt)α-MSH酸是α-MSH的酸形式。 -
GC68390
α5β1 integrin agonist-1
α5β1 integrin agonist-1 作为 α5β1 integrin 激动剂,能够选择性地将 5-FU 输送到肿瘤细胞中,成功地导致肿瘤细胞死亡。
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GC62380
αvβ1 integrin-IN-1
αvβ1 integrin-IN-1 (Compound C8) 是一种有效的选择性 αvβ1 整合素抑制剂,IC50 为 0.63 nM。具有抗纤维化作用。
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GC62566
αvβ1 integrin-IN-1 TFA
αvβ1 integrin-IN-1 TFA (Compound C8) 是一种有效的选择性 αvβ1 整合素抑制剂,IC50 为 0.63 nM。具有抗纤维化作用。
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GC64932
αvβ5 integrin-IN-1
αvβ5 integrin-IN-1 是第一个有效和选择性 αvβ5 整合素抑制剂(pIC50 = 8.2)。
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GC48920
β-Carboline-1-carboxylic Acid
1-Formic Acid-β-carboline
An alkaloid with diverse biological activities -
GC62551
β-Hydroxypropiovanillone
3,4'-二羟基-3'-甲氧基苯丙酮
β-Hydroxypropiovanillone 是一种天然化合物,对 α-葡萄糖苷酶 (α-glucosidase) 具有明显的浓度依赖性抑制作用 (IC50=257.8 μg/mL)。 -
GC41502
β-Myrcene
月桂烯; β-Myrcene
A terpene with antioxidative properties -
GC92102
γ1-MSH (human, mouse, rat, bovine) (acetate)
γ1-Melanocyte-stimulating Hormone
γ1-MSH (human, mouse, rat, bovine) (acetate)是一种肽激素,由垂体中的前皮黑皮质素(POMC)翻译后加工产生。 -
GC92101
γ1-MSH (human, mouse, rat, bovine) (trifluoroacetate salt)
γ1-Melanocyte-stimulating Hormone
γ1-MSH (human, mouse, rat, bovine) (trifluoroacetate salt)是一种肽激素,由垂体中的前皮黑皮质素(POMC)翻译后加工产生。 -
GC45270
(±)10(11)-EDP Ethanolamide
10,11-EDP-EA, 10,11-EDP epoxide, 10,11-epoxy Docosapentaenoic Ethanolamide
An ω-3 endocannabinoid epoxide and CB receptor agonist -
GC40802
(±)12(13)-DiHOME
Isoleukotoxin diol
A diol form of (±)12,13-EpOME -
GC41648
(±)13(14)-DiHDPA
13(14)-DiHDPA, 13(14)-DiHDoPE, 13,14-DiHDPE
A metabolite of DHA -
GC41653
(±)16(17)-DiHDPA
An epoxygenase metabolite of DHA
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GC41655
(±)19(20)-EDP Ethanolamide
19,20-DHEA epoxide, 19,20-epoxy Docosapentaenoic Acid Ethanolamide, 19,20-EDP-EA, 19,20-EDP epoxide
An ω-3 endocannabinoid epoxide and CB receptor agonist -
GC40801
(±)9(10)-DiHOME
(±)-苏式-9,10-二羟基-12(Z)-十八碳烯酸
A diol form of (±)9(10)-EpOME -
GC18516
(+)-Aeroplysinin-1
(+)-Aeroplysinin-1
A sea sponge metabolite with diverse biological activities -
GC39795
(+)-Afzelechin
(+)-阿夫儿茶精
(+)-Afzelechin 是从佛手根的根茎中分离出来的,是一种 α-葡萄糖苷酶 (alpha-glucosidase) 活性抑制剂,ID50 值为 0.13 mM。(+)-Afzelechin 可以延迟食物中碳水化合物的吸收,从而抑制餐后高血糖和高胰岛素血症。 -
GC45266
(+)-Macrosphelide A
A fungal metabolite
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GC18749
(+)-Rugulosin
细皱青霉素+FORM,(+)-Rugulosin
A mycotoxin -
GC17102
(-)-Tetramisole
盐酸左旋咪唑
An Analytical Reference Material -
GC65363
(1R)-Tenofovir amibufenamide
(1R)-HS-10234
(1R)-Tenofovir amibufenamide ((1R)-HS-10234) 是 Tenofovir amibufenamide 的异构体,是一种口服活性抗病毒药物。(1R)-Tenofovir amibufenamide ((1R)-HS-10234) 是一个 HIV 病毒感染的抑制剂和乙型肝炎病毒的抑制剂 ( HBV )。(1R)-Tenofovir amibufenamide ((1R)-HS-10234) 可用于 HIV 感染、乙肝研究。 -
GC65547
(1S,2R)-Alicapistat
(1S,2R)-ABT-957
(1S,2R)-Alicapistat ((1S,2R)-ABT-957) 是一种具有口服活性的人钙激活中性蛋白酶 (calpains 1 和 2) 的选择性抑制剂,可能用于阿尔茨海默病 (AD) 的研究。 Alicapistat 可减轻羰基还原的代谢倾向,对 calpain 1 的 IC50 为 395 nM。 -
GC62193
(1S,2S)-Bortezomib
硼替佐米杂质E
(1S,2S)-Bortezomib 是 Bortezomib 的对映异构体。Bortezomib 是一种细胞渗透性、可逆性和选择性的蛋白酶体抑制剂,通过靶向苏氨酸残基有效抑制 20S 蛋白酶体 (Ki 为 0.6 nM)。Bortezomib 破坏细胞周期、诱导细胞凋亡以及抑制核因子 NF-κB。Bortezomib 是一种抗癌药物,也是第一种用于人类的蛋白酶体抑制剂。 -
GC68525
(2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid
(2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid 是一种可从 Rubus ellipticus var. obcordatus 中分离得到的皂苷。(2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid 抑制 α-Glucosidase,其 IC50 为 1.68 mM。
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GC64260
(2S,5S)-Censavudine
(2S,5S)-OBP-601; (2S,5S)-BMS-986001
(2S,5S)-Censavudine ((2S,5S)-OBP-601) 是 Censavudine 的 (2S,5S)-对映异构体。Censavudine 是一种核苷类逆转录酶抑制剂,是一种有效的 HIV 抑制剂。 -
GC40444
(5Z,11Z,15R)-15-Hydroxyeicosa-5,11-dien-13-ynoic Acid
HETE Analog 1, Hydroxyeicosatetraenoic Acid Analog 1
A stable isomer of 15(S)-HETE -
GC92107
(D-Phe7)-α-MSH (trifluoroacetate salt)
(D-Phe7)-α-Melanocyte-stimulating Hormone
(D-Phe7)-α-MSH (trifluoroacetate salt) ((D-Phe7)-α-MSH)是α-MSH的肽衍生物,是合成α-MSH环类似物的中间体。 -
GC41699
(Des-octanoyl)-Ghrelin (human) (trifluoroacetate salt)
A peptide hormone
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GC41700
(E)-2-(2-Chlorostyryl)-3,5,6-trimethylpyrazine
CSTMP
A stilbene derivative with antioxidant and anticancer activities -
GC62735
(E/Z)-GO289
(E/Z)-GO289 potently and selectively inhibits casein kinase 2 (CK2) at an IC50 of 7 nM in vitro kinase assay.
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GC49167
(R)-(+)-Trityl glycidyl ether
三苯甲基-(R)-缩水甘油醚
A synthetic precursor -
GC41620
(R)-(-)-Mellein
(R)-蜂蜜曲菌素,以及(S)-蜂蜜曲菌素,(R)-Mellein
A dihydroisocoumarin compound with antibacterial, antimalarial, antifungal , and anticancer effects -
GC74184
(R)-Azasetron besylate
SENS-401
(R)-Azasetron besylateSENS-401是一种口服活性钙调神经磷酸酶抑制剂。 -
GC69837
(R/S)-Alicaforsen
(R/S)-ISIS-2302
(R/S)-Alicaforsen 是由R和S构型组成的 Alicaforsen 的消旋体。Alicaforsen是一种20个碱基长度的反义寡核苷酸,抑制 ICAM-1 的产生,ICAM-1 是一种重要的粘附分子,参与白细胞向炎症部位迁移和转运的过程。 -
GC46351
(S)-CR8
An inhibitor of cyclin-dependent kinases
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GC64535
(S,S)-TAPI-1
TAPI
A TACE inhibitor -
GC45978
1,10-Phenanthroline (hydrate)
邻菲罗啉,1,10-Phenanthroline monohydrate
A metal chelator and inhibitor of metalloproteases -
GC41774
1,2,3-Trimyristoyl-rac-glycerol
三肉豆蔻酸甘油酯
A triacylglycerol -
GC90744
1,2-Dioleoyl-3(R)-trimethylammoniumpropane (chloride)
R-DOTAP
一个阳离子脂质
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GC49294
1-(4-Chlorobenzhydryl)piperazine
1-(4-氯二苯甲基)哌嗪
An inactive metabolite of meclizine and chlorcyclizine -
GC41992
1-Deoxynojirimycin (hydrochloride)
去氧野艽霉素盐酸盐,Duvoglustat hydrochloride
An iminosugar with diverse biological activities -
GC41998
1-Methyl-4-imidazoleacetic Acid (hydrochloride)
1-甲基-4-羧酸咪唑盐酸盐
A stable metabolite of histamine -
GC25005
1-Naphthyl phosphate potassium salt
α-Naphthyl acid phosphate monopotassium salt
1-Naphthyl phosphate potassium salt (α-Naphthyl acid phosphate monopotassium salt) is a non-specific phosphatase inhibitor which acts on acid, alkaline, and protein phosphatases. -
GC42026
1-Palmitoyl-2-hydroxy-sn-glycero-3-PC
1-十六酰-SN-丙三醇-磷酸胆碱
A product of PLA2-mediated hydrolysis of phosphatidylcholine -
GC46490
1-Palmitoyl-d3-2-hydroxy-sn-glycero-3-PC
1-Hexadecanoyl-sn-glycero-3-Phosphatidylcholine-d3, 1-Hexadecanoyl-sn-glycero-3-Phosphocholine-d3, LPC-d3, 16:0/0:0(d3) Lyso-PC, 1-Palmitoyl-sn-glycero-3-Phosphocholine-d3, PC(16:0/0:0)-d3, 16:0/0:0-PC-d3
A neuropeptide with diverse biological activities -
GC45693
1-Palmitoyl-d9-2-hydroxy-sn-glycero-3-PC
1-Hexadecanoyl-d9-sn-glycero-3-Phosphatidylcholine, 1-Hexadecanoyl-d9-sn-glycero-3-Phosphocholine, 16:0(d9) Lyso-PC, PC(16:0-d9/0:0), 16:0-d9/0:0-PC
An internal standard for the quantification of 1-palmitoyl-2-hydroxy-sn-glycero-3-PC