Drug Metabolite
Drug Metabolite(药物代谢物)
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Drug Metabolite 相关产品(498)
- GC44299N-Acetyl-4-benzoquinone imineCAS: 50700-49-7纯度: >90.00%
A reactive CYP450 metabolite of acetaminophen
- GC44451Norfluoxetine (hydrochloride)CAS: 57226-68-3纯度: >98.00%
Norfluoxetine (hydrochloride)是Fluoxetine在肝脏中通过N-去甲基化产生的活性代谢物，具有口服活性。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC43743 | Gemfibrozil 1-O-β-Glucuronide | 91683-38-4 | >99.5% | |
A major metabolite of gemfibrozil | ||||
| GC43878 | Hydroxy Dimetridazole | 936-05-0 | >98.50% | |
A metabolite of dimetridazole | ||||
| GC43879 | Hydroxy Ebastine | 210686-41-2 | >87.00% | |
An ebastine metabolite | ||||
| GC43881 | Hydroxy Varenicline | 357424-21-6 | >95.00% | |
A metabolite of varenicline | ||||
| GC43895 | Iloperidone metabolite P88 | 133454-55-4 | >99.50% | |
An active metabolite of iloperidone | ||||
| GC43896 | Iloperidone metabolite P95 | 475110-48-6 | >98.00% | |
A metabolite of iloperidone | ||||
| GC44033 | Lansoprazole sulfone | 131926-99-3 | >98.00% | |
A metabolite of lansoprazole | ||||
| GC44246 | Moxifloxacin N-Sulfate (sodium salt) | - | >95.00% | |
A metabolite of moxifloxacin | ||||
| GC44294 | N-acetyl Dapsone | 565-20-8 | >95.00% | |
A metabolite of dapsone | ||||
| GC44299 | N-Acetyl-4-benzoquinone imine | 50700-49-7 | >90.00% | |
A reactive CYP450 metabolite of acetaminophen | ||||
| GC44304 | N-Acetyl-S-allyl-L-cysteine | 23127-41-5 | >98.00% | |
A primary metabolite of L-deoxyalliin | ||||
| GC44345 | N-Desethyl Vardenafil | 448184-46-1 | >98.00% | |
A vardenafil metabolite | ||||
| GC44348 | N-desmethyl Bendamustine | 41515-13-3 | >95.00% | |
An active metabolite of bendamustine | ||||
| GC44349 | N-desmethyl Levofloxacin | 117707-40-1 | >98.00% | |
An active metabolite of levofloxacin | ||||
| GC44350 | N-Desmethyl Sildenafil | 139755-82-1 | >98.00% | |
A major metabolite of sildenafil | ||||
| GC44351 | N-Desmethyl Sildenafil (citrate) | - | >98.00% | |
A major metabolite of sildenafil | ||||
| GC44358 | Nebivolol O-β-D-Glucuronide | - | >95.00% | |
An active metabolite of nebivolol | ||||
| GC44451 | Norfluoxetine (hydrochloride) | 57226-68-3 | >98.00% | |
Norfluoxetine (hydrochloride)是Fluoxetine在肝脏中通过N-去甲基化产生的活性代谢物，具有口服活性。 | ||||
| GC44492 | O-Desmethyl Metoprolol | 62572-94-5 | >99.00% | |
A major active metabolite of metoprolol | ||||
| GC44509 | Omeprazole sulfide | 73590-85-9 | >99.50% | |
An intermediate for omeprazole synthesis | ||||
| GC44527 | p,p'-DDE | 72-55-9 | >99.50% | |
A metabolite and degradation product of the pesticide DDT | ||||
| GC44554 | Pantoprazole Sulfide | 102625-64-9 | >98.00% | |
A pantoprazole metabolite | ||||
| GC44555 | Pantoprazole sulfone | 127780-16-9 | >98.00% | |
A pantoprazole metabolite | ||||
| GC44599 | Perindoprilat | 95153-31-4 | >95.00% | |
An active ACE inhibitor | ||||