Potassium Channel
Potassium Channel(钾离子通道)
Potassium channels are voltage-gated ion channels that selectively permeate potassium ion through the excitable membrane. It regulates the release of neurotransmitters, insulin secretion, smooth muscle contraction and heart rate etc.
Potassium Channel 相关产品(302)
- GC73927KIO-301 chloride (hydrochloride)纯度: >99.00%
KIO-301 chloride (hydrochloride)是一种偶氮苯光开关化合物,可阻断电压门控离子通道,包括过极化激活的环核苷酸门控和电压门控钾通道。
- GC743846-FAM-AEEAc-Stichodactyla helianthus Neurotoxin (ShK) (TFA)纯度: >95.00%
6-FAM-AEEAc-Stichodactyla helianthus Neurotoxin (ShK) (TFA) 6-FAM-AEEAC-SHK TFA是一种结合荧光标记物的肽神经毒素。
- GN1079920(S)-Ginsenoside Rg3CAS: 14197-60-5纯度: >98.00%
20(S)-Ginsenoside Rg3是从人参中提取的稀有人参皂苷(Na + :IC 50 = 32.2±4.5μM;hKv1.4:IC 50 = 32.6±2.2μM)。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC72302 | Spinoxin | 752984-66-0 | >98.00% | |
Spinoxin从刺异尾蝎毒液中分离出的一种由四个二硫键交联的34个残基的肽神经毒素。 | ||||
| GC72973 | AVE1231 | 767334-89-4 | 不显示 | |
AVE1231(A293)是一种具有抗心律失常活性的双孔钾通道TASK-1抑制剂。 | ||||
| GC73796 | CVN293 | 2815296-08-1 | >99.00% | |
CVN293是一种选择性和脑渗透性钾离子(K+)通道KCNK13抑制剂,对hKCNK13和mKCNK13的ic50分别为41 nM和28 nM。 | ||||
| GC73927 | KIO-301 chloride (hydrochloride) | - | >99.00% | |
KIO-301 chloride (hydrochloride)是一种偶氮苯光开关化合物,可阻断电压门控离子通道,包括过极化激活的环核苷酸门控和电压门控钾通道。 | ||||
| GC73985 | VU0542270 | 1396814-79-1 | >98.00% | |
VU0542270是一种选择性血管Kir6.1/SUR2B KATP通道抑制剂,IC50值为100nM。 | ||||
| GC74004 | CPK20 | 2397708-22-2 | >98.00% | |
CPK20是一种有效的高选择性KCNT1通道阻滞剂,CPK20可用于癫痫的研究。 | ||||
| GC74190 | Hydrochlorothiazide-13C6 | 1261396-79-5 | >99.00% | |
Hydrochlorothiazide-13C6是13C标记的屈氯噻嗪。 | ||||
| GC74384 | 6-FAM-AEEAc-Stichodactyla helianthus Neurotoxin (ShK) (TFA) | - | >95.00% | |
6-FAM-AEEAc-Stichodactyla helianthus Neurotoxin (ShK) (TFA) 6-FAM-AEEAC-SHK TFA是一种结合荧光标记物的肽神经毒素。 | ||||
| GC74396 | Tamapin TFA | - | >98.00% | |
Tamapin TFA是一种毒液肽,靶向小电导Ca(2+)激活的K(+)(SK)通道。 | ||||
| GN10267 | Loureirin B | 119425-90-0 | >99.00% | |
A flavonoid with diverse biological activities | ||||
| GN10446 | Tetrandrine | 518-34-3 | >99.50% | |
An alkaloid with diverse biological activities | ||||
| GN10799 | 20(S)-Ginsenoside Rg3 | 14197-60-5 | >98.00% | |
20(S)-Ginsenoside Rg3是从人参中提取的稀有人参皂苷(Na + :IC 50 = 32.2±4.5μM;hKv1.4:IC 50 = 32.6±2.2μM)。 | ||||
| GN10812 | Acacetin | 480-44-4 | >99.50% | |
A flavonoid | ||||
| GC17469 | 4-Aminopyridine | 504-24-5 | >98.00% | |
potassium channel-blocking agent | ||||
