GlpBio

Prostaglandin Receptor

Prostaglandin Receptor(前列腺素受体)

Prostaglandin receptors are a group of g-protein coupled receptor that exhibited a variety of functions in regulation of blood pressure and renal function; smooth muscle contraction; inhibition of plate aggregation; immune response etc.

Prostaglandin Receptor 相关产品(170)

  • GC17348 structure
    GC17348BW A868C
    CAS: 118675-50-6
    纯度: >98.00%

    A DP receptor antagonist

  • GC17367 structure
    GC17367Rebamipide
    CAS: 90098-04-7
    纯度: >99.50%

    A gastroprotective agent and mucin secretagogue

  • GC17410 structure
    GC17410S18886
    CAS: 165538-40-9
    纯度: >98.00%

    A TP receptor antagonist

  • GC17719 structure
    GC177195-trans U-46619
    CAS: 330796-58-2

    An isomer of U-46619

  • GC17861 structure
    GC17861Sulprostone
    CAS: 60325-46-4
    纯度: >98.00%

    Selective EP 3 receptor agonist

  • GC18111 structure
    GC18111Seratrodast
    CAS: 112665-43-7
    纯度: >98.00%

    A thromboxane A 2 receptor antagonist

  • GC18132 structure
    GC18132U-44069
    CAS: 56985-32-1

    A TP receptor agonist

  • GC18318 structure
    GC18318CAY10441
    CAS: 221529-58-4
    纯度: >98.00%

    An IP receptor antagonist

  • GC18678 structure
    GC18678CAY10595
    CAS: 916047-16-0

    A potent CRTH2/DP 2 receptor antagonist

  • GC19147 structure
    GC19147Evatanepag
    CAS: 223488-57-1
    纯度: >99.00%

    Evatanepag (CP-533536) 是一种非前列腺素、强效和选择性 EP2 受体激动剂。

  • GC19153 structure
    GC19153Fevipiprant
    CAS: 872365-14-5
    纯度: >99.50%

    A DP 2 /CRTH 2 antagonist

  • GC19327 structure
    GC19327Setipiprant
    CAS: 866460-33-5
    纯度: >98.00%

    Setipiprant是一种选择性、口服可用的前列腺素 D2 受体 2（DP2，也称为 CRTH2）拮抗剂，是γ-咔啉衍生物，其IC₅₀为6nM。

  • GC19354 structure
    GC19354TG6-10-1
    CAS: 1415716-58-3
    纯度: >99.50%

    A potent EP 2 receptor antagonist

  • GC19395 structure
    GC19395MK-7246
    CAS: 1218918-62-7
    纯度: >98.50%

    A CRTH 2 /DP 2 receptor antagonist

  • GC30068 structure
    GC30068Taprenepag (CP-544326)
    CAS: 752187-80-7
    纯度: >99.50%

    A potent EP 2 receptor agonist

  • GC30299 structure
    GC30299GSK726701A
    CAS: 945721-87-9
    纯度: >98.50%

    GSK726701A是前列腺素E2受体4(EP4)的部分激动剂，pEC50为7.4。

  • GC30307 structure
    GC30307GSK-269984A
    CAS: 892664-04-9

    GSK-269984A是前列腺素E2受体1(ProstaglandinE2Receptor1(EP1))的拮抗剂，pIC50值为7.9。

  • GC30370 structure
    GC30370Dinoprost (Prostaglandin F2a)
    CAS: 551-11-1
    纯度: >99.00% / >96.50%

    Dinoprost (Prostaglandin F2a)是一种口服有效的强效前列腺素受体 （FP 受体） 激动剂。Dinoprost刺激子宫肌层活动，放松宫颈，抑制黄体类固醇生成，并通过直接作用诱导黄体溶解。

  • GC30561 structure
    GC305612-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
    CAS: 137089-36-2

    2-(E-2-decenoylamino)ethyl2-(cyclohexylethyl)sulfide是一种由压力诱发的溃疡和低毒性抑制剂，可以在压力引起的溃疡大鼠中，维持磷脂酶A2(phospholipaseA2)和前列腺素E2(prostaglandinE2)的含量水平。

  • GC30572 structure
    GC30572Aganepag (AGN 210937)
    CAS: 910562-18-4

    Aganepag (AGN 210937) 是一种有效的 Prostanoid EP2 受体激动剂，EC50 为 0.19 nM，对 EP4 受体没有活性。

  • GC30604 structure
    GC30604Darbufelone mesylate (CI-1004 mesylate)
    CAS: 139340-56-0
    纯度: >98.00%

    Darbufelone mesylate (CI-1004 mesylate) (CI-1004 mesylate) 是细胞 PGF2α 的双重抑制剂；和 LTB4 生产。

  • GC30743 structure
    GC30743(+)-Cloprostenol (D-Cloprostenol)
    CAS: 54276-21-0
    纯度: >98.00%

    A FP receptor agonist and potent luteolytic agent

  • GC31202 structure
    GC31202EP1-antanoist-1
    CAS: 851204-35-8

    EP1-antanoist-1 是一种 EP1 拮抗剂，pKi 为 7.54，pIC50 为 8.5。

  • GC31445 structure
    GC31445Tiaprost (Iliren)
    CAS: 71116-82-0

    A synthetic analog of PGF 2α