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Home >> Signaling Pathways >> GPCR/G protein >> 5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC11570 Desvenlafaxine

    去甲文拉法辛; O-Desmethylvenlafaxine

     An active metabolite of venlafaxine
  3. GC10848 BMY 7378

    BMY7378抑制剂

     BMY 7378是一种α1D-肾上腺素能受体（α1D-AR）的选择性拮抗剂，pki值为8.89，也是血清素1A受体（5-HT1A R）的混合激动剂和拮抗剂。
  4. GC13723 Amitriptyline HCl

    盐酸阿米替林

     A tricyclic antidepressant
  5. GC10891 Alverine Citrate

    枸橼酸阿尔维林,NSC 35459

     An antispasmodic agent
  6. GC17808 Zolmitriptan

    佐米曲普坦,BW-311C90; 311C90

     An agonist of 5-HT1B and 5-HT1D receptors
  7. GC11959 Naratriptan

    盐酸那拉曲坦,GR-85548A

     A potent 5-HT1B and 5-HT1D receptor agonist
  8. GC13428 Mosapride

    莫沙必利; TAK-370; AS-4370

     A 5-HT4 receptor agonist
  9. GC13478 Pizotifen Malate

    苯噻啶苹果酸盐,Pizotyline malate; BC-105 malate

     A triptan
  10. GC13053 Pizotifen

    苯噻啶; Pizotyline; BC-105

     A triptan
  11. GC13092 Fluvoxamine

    氟伏沙明; DU-23000

     Fluvoxamine是一种选择性血清素（5-HT）再摄取抑制剂（SSRI），具有抗抑郁活性。
  12. GC17593 Lurasidone HCl

    盐酸鲁拉西酮; SM-13496 Hydrochloride

     An atypical antipsychotic
  13. GC16891 Quetiapine Fumarate

    富马酸喹硫平

     An antagonist of diverse neurological receptors
  14. GC15223 Tropisetron Hydrochloride

    盐酸托烷司琼

     A 5-HT3 receptor antagonist
  15. GC11651 Ondansetron hydrochloride dihydrate

    盐酸昂丹司琼二水物; GR 38032 hydrochloride dihydrate; SN 307 hydrochloride dihydrate

     An Analytical Reference Material
  16. GC14512 Fenspiride HCl

    盐酸芬司必利

     A histamine H1 receptor antagonist
  17. GC17917 Palonosetron HCl

    盐酸帕洛诺司琼

     A 5-HT3 receptor antagonist
  18. GC17053 Eletriptan HBr

    依来曲普坦氢溴酸盐; Eletriptan HBr; UK-116044 hydrobromide

     An agonist of 5-HT1B and 5-HT1D receptors
  19. GC10799 Iloperidone hydrochloride

    盐酸伊潘立酮; HP 873 hydrochloride

     An atypical antipsychotic
  20. GC13081 Loxapine

    洛沙平

     洛沙平是一种口服活性多巴胺抑制剂、5-HT 受体拮抗剂，也是一种二苯并沙西平抗精神病药物。
  21. GC17981 Agomelatine

    阿戈美拉汀; S-20098

     Agomelatine是一种褪黑素（MT）受体激动剂，对MT1和MT2的Ki值分别为0.1 nM和0.12 nM。Agomelatine也是一种5-羟色胺（5-HT）受体拮抗剂，对5-HT2C 和5-HT2B 的Ki值分别为631 nM和660 nM。
  22. GC11186 Brexpiprazole

    依匹哌唑; OPC-34712

     Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（Ki=0.12nM）和dopamine D2L（Ki=0.3nM）受体的强效部分激动剂，以及5-HT2A受体（Ki=0.47nM）的拮抗剂。
  23. GC10450 PRX-08066 A 5-HT2B receptor antagonist
  24. GC10769 SB269970 HCl

    SB-269970A

     SB269970 HCl是一种强效且选择性的5-HT7受体拮抗剂，具有高亲和力 (pKi = 8.9)。
  25. GC15121 Lasmiditan

    拉米地坦

     An Analytical Reference Standard
  26. GC10945 Tandospirone

    坦度螺酮; SM-3997

     Tandospirone (SM-3997) 是一种有效的选择性 5-HT1A 受体部分激动剂，Ki 为 27 nM。
  27. GC10117 Aripiprazole

    阿立哌唑; OPC-14597

     An atypical antipsychotic
  28. GC12495 Olanzapine

    奥氮平; LY170053

     Olanzapine是一种单胺拮抗剂。
  29. GC12091 SB742457

    3-苯基磺酰基-8-(哌嗪-1-基)喹啉,SB-742457; GSK-742457; RVT-101

     A 5-HT6 receptor antagonist
  30. GC13533 Cisapride

    西沙比利; R 51619; (±)-Cisaprid

     A 5-HT4 receptor agonist
  31. GC17130 BRL-54443

    3-(1-甲基-4-哌啶基)-1H-吲哚-5-醇

     A potent agonist of 5-HT1E and 5-HT1F
  32. GC16226 BRL-15572 dihydrochloride

    BRL15572盐酸盐

     A 5-HT1D receptor antagonist
  33. GC10698 Cyproheptadine hydrochloride

    盐酸赛庚啶

     An antihistamine with antiserotonergic and anticholinergic activities
  34. GC13871 Duloxetine HCl

    盐酸度洛西汀; (S)-Duloxetine hydrochloride; LY-248686 hydrochloride

     A serotonin and norepinephrine reuptake inhibitor
  35. GC14160 Blonanserin

    布南色林; AD-5423

     A dopamine and serotonin receptor antagonist
  36. GC11977 Thioridazine HCl

    盐酸硫利达嗪；盐酸硫代利哒；甲硫达嗪盐酸盐；甲硫哒嗪盐酸盐

     A typical antipsychotic
  37. GC10460 Rizatriptan Benzoate

    苯甲酸利扎曲坦,MK 462

     A 5-HT1B and 5-HT1D receptor agonist
  38. GC12986 Risperidone

    利培酮; R 64 766

     Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂，对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。
  39. GC16788 PRX-08066 Maleic acid 5-HT2B receptor antagonist,potent and selective
  40. GC14437 Vortioxetine (Lu AA21004) HBr

    盐酸沃替西汀; Lu AA21004 hydrobromide

     A multimodal serotonergic agent
  41. GC15463 Iloperidone

    伊潘立酮; HP 873

     An atypical antipsychotic
  42. GC11521 Ziprasidone HCl

    盐酸齐拉西酮; CP-88059 hydrochloride

     An atypical antipsychotic
  43. GC18006 Sumatriptan Succinate

    舒马普坦琥珀酸盐; GR 43175

     Sumatriptan Succinate是一种具有口服活性的5-HT1受体激动剂，对5-HT1D、5-HT1B和5-HT1F受体的IC50值分别为7.3nM、9.3nM和17.8nM。
  44. GC10121 Tianeptine sodium

    噻奈普汀钠

     An atypical antidepressant
  45. GC10911 Venlafaxine hydrochloride

    盐酸文拉法辛; Wy 45030 hydrochloride

     Venlafaxine hydrochloride是一种具有口服活性的5-羟色胺和去甲肾上腺素再摄取抑制剂 （SNRIs; Serotonin-norepinephrine reuptake inhibitors），对配体与人NE和5-HT转运蛋白结合的Ki值分别为2480nM和82nM。
  46. GC11814 Ondansetron HCl

    盐酸昂丹司琼; GR 38032 hydrochloride; SN 307 hydrochloride

     A Certified Reference Material
  47. GC15025 Fluvoxamine maleate

    氟伏沙明马来酸盐; DU-23000 maleate

     A selective serotonin reuptake inhibitor
  48. GC11709 Fluoxetine HCl

    盐酸氟西汀; LY 110140

     An Analytical Reference Material
  49. GC11824 Asenapine

    阿塞那平; Org 5222

     An atypical antipsychotic
  50. GC17536 Mosapride Citrate

    莫沙必利柠檬酸盐; TAK-370 citrate; AS-4370 citrate

     A 5-HT4 receptor agonist
  51. GC16029 Granisetron HCl

    盐酸格拉司琼; BRL 43694A

     A 5-HT3 receptor antagonist with antiemetic activity

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