5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(481)
- GC15138SB 243213 dihydrochlorideCAS: 200940-23-4
SB 243213 dihydrochloride 是一种具有口服活性、选择性和高亲和力的 5-HT2C 受体拮抗剂，对人 5-HT2C 受体的 pKi 为 9.37，pKb 为 9.8。
- GC15235NAN-190 hydrobromideCAS: 115338-32-4纯度: >99.00%
A 5-HT1A receptor mixed antagonist and partial agonist
- GC15630SR 57227 hydrochlorideCAS: 77145-61-0纯度: >98.00%
SR 57227 hydrochloride是一种强效的serotonin type-3 (5-HT 3 )受体激动剂，能够穿过血脑屏障。
- GC160311-(3-Chlorophenyl)piperazine (hydrochloride)CAS: 13078-15-4纯度: >98.00%
An Analytical Reference Standard
- GC16045EMD 386088 hydrochlorideCAS: 1171123-46-8
EMD 386088 hydrochloride 是一种有效的血清素 6 受体 (5-HT6R) 激动剂。
- GC16324Nefazodone hydrochlorideCAS: 82752-99-6纯度: >98.00%
A serotonin, norepinephrine, and dopamine reuptake inhibitor
- GC16439SB 203186 hydrochlorideCAS: 207572-69-8纯度: >99.50%
SB 203186 hydrochloride 是一种有效的、选择性的和竞争性的 5-HT4 拮抗剂。
- GC16470Methysergide maleateCAS: 129-49-7纯度: >95.00%
A 5-HT 1 receptor agonist and 5-HT 2 receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15137 | RS 56812 hydrochloride | 143339-12-2 | - | |
5-HT3 partial agonist | ||||
| GC15138 | SB 243213 dihydrochloride | 200940-23-4 | - | |
SB 243213 dihydrochloride 是一种具有口服活性、选择性和高亲和力的 5-HT2C 受体拮抗剂，对人 5-HT2C 受体的 pKi 为 9.37，pKb 为 9.8。 | ||||
| GC15235 | NAN-190 hydrobromide | 115338-32-4 | >99.00% | |
A 5-HT1A receptor mixed antagonist and partial agonist | ||||
| GC15248 | GR 125487 sulfamate | 859502-43-5 | - | |
5-HT4 receptor antagonist | ||||
| GC15268 | Org 12962 hydrochloride | 210821-63-9 | - | |
A 5-HT 2C receptor agonist | ||||
| GC15367 | EMDT oxalate | 263744-72-5 | - | |
EMDT 草酸盐是一种选择性 5-HT6 激动剂，具有抗抑郁作用。 | ||||
| GC15456 | m-Chlorophenylbiguanide hydrochloride | 2113-05-5 | - | |
A 5-HT 3 receptor agonist | ||||
| GC15551 | SB 216641 hydrochloride | 193611-67-5 | >98.00% | |
A 5-HT 1B receptor antagonist | ||||
| GC15569 | 3-AQC | 201216-42-4 | - | |
5-HT3 antagonist | ||||
| GC15630 | SR 57227 hydrochloride | 77145-61-0 | >98.00% | |
SR 57227 hydrochloride是一种强效的serotonin type-3 (5-HT 3 )受体激动剂，能够穿过血脑屏障。 | ||||
| GC15660 | SB 399885 hydrochloride | 402713-81-9 | >99.50% | |
A 5-HT 6 receptor antagonist | ||||
| GC15872 | NPEC-caged-serotonin | 1257326-22-9 | - | |
5-HT receptor agonist | ||||
| GC15979 | RS 16566 dihydrochloride | 1217788-97-0 | - | |
(R)-zacopride 结合位点的配体 | ||||
| GC15985 | Cariprazine | 839712-12-8 | >99.00% | |
An atypical antipsychotic | ||||
| GC16031 | 1-(3-Chlorophenyl)piperazine (hydrochloride) | 13078-15-4 | >98.00% | |
An Analytical Reference Standard | ||||
| GC16040 | 4F 4PP oxalate | 144734-36-1 | - | |
A 5-HT 2A receptor antagonist | ||||
| GC16045 | EMD 386088 hydrochloride | 1171123-46-8 | - | |
EMD 386088 hydrochloride 是一种有效的血清素 6 受体 (5-HT6R) 激动剂。 | ||||
| GC16135 | Cinanserin hydrochloride | 54-84-2 | >99.50% | |
A 5-HT receptor antagonist | ||||
| GC16324 | Nefazodone hydrochloride | 82752-99-6 | >98.00% | |
A serotonin, norepinephrine, and dopamine reuptake inhibitor | ||||
| GC16399 | N-Methylquipazine dimaleate | 171205-17-7 | - | |
5-HT3 agonist | ||||
| GC16439 | SB 203186 hydrochloride | 207572-69-8 | >99.50% | |
SB 203186 hydrochloride 是一种有效的、选择性的和竞争性的 5-HT4 拮抗剂。 | ||||
| GC16470 | Methysergide maleate | 129-49-7 | >95.00% | |
A 5-HT 1 receptor agonist and 5-HT 2 receptor antagonist | ||||
| GC16506 | Quipazine dimaleate | 150323-78-7 | - | |
5-HT3 receptor agonist | ||||
| GC16553 | N-Desmethylclozapine | 6104-71-8 | >99.50% | |
An active metabolite of clozapine | ||||