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Home >> Signaling Pathways >> GPCR/G protein >> 5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC13583 CJ 033466 CJ 033466 是一种新型选择性 5-HT4 受体部分激动剂，EC50 为 9 nM，具有促胃动力作用。
  3. GC12657 LY 334370 hydrochloride A 5-HT1F receptor agonist
  4. GC10919 LY 272015 hydrochloride

    1-(3,4-二甲氧基苄基)-6-甲基-2,3,4,9-四氢-1H-吡啶并[3,4-B]吲哚盐酸盐

     A 5-HT2B receptor antagonist
  5. GC14607 1-Methylpsilocin 5-HT2C agonist,potent and selective
  6. GC14195 LP 12 hydrochloride LP 12 hydrochloride (compound 21) 是一种有效的选择性 5-HT7 受体激动剂，Ki 为 0.13 nM。
  7. GC17260 Ro 04-6790

    4-氨基-N-[2,6-双(甲基氨基)-4-嘧啶基]苯磺酰胺

     A 5-HT6 receptor antagonist
  8. GC16324 Nefazodone hydrochloride

    萘法唑酮盐酸盐,BMY-13754; MJ-13754-1

     A serotonin, norepinephrine, and dopamine reuptake inhibitor
  9. GC13109 Fananserin

    法南色林,RP 62203

     Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。
  10. GC11308 L-703,664 succinate 5-HT1D receptor agonist
  11. GC11490 TCB-2 5-HT2A受体激动剂
  12. GC18112 LP 44 A selective 5-HT7 receptor agonist
  13. GC11929 Melperone hydrochloride

    1-[3-(对氟苯甲酰基)丙基]-4-甲基哌嗪氯化物

     An atypical antipsychotic
  14. GC16045 EMD 386088 hydrochloride EMD 386088 hydrochloride 是一种有效的血清素 6 受体 (5-HT6R) 激动剂。
  15. GC17714 PNU 22394 hydrochloride 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
  16. GC14583 R 59-022

    DKGI-I; Diacylglycerol kinase inhibitor I

     R 59-022是一种二酰甘油激酶抑制剂（IC50 = 2.8µM）。
  17. GC12300 WAY 629 hydrochloride

    5-HT2C agonist
  18. GC17219 SDZ 205-557 hydrochloride 5-HT3/5-HT4 receptor antagonist
  19. GC17525 AS 19

    A 5-HT7 receptor agonist
  20. GC12383 SB 258585 hydrochloride A selective 5-HT6 receptor antagonist
  21. GC13883 Ritanserin

    利坦丝林,R 55667

     A potent 5-HT2A receptor antagonist
  22. GC15135 Ro 60-0175 fumarate A 5-HT2 receptor agonist
  23. GC14030 Altanserin hydrochloride 5-HT2A receptor antagonist
  24. GC11980 WAY 161503 hydrochloride A 5-HT2C receptor agonist
  25. GC17343 Zacopride hydrochloride

    查可必利盐酸盐

     Zacopride hydrochloride 是一种高效的 5-HT3 受体拮抗剂，对 5-HT3 和 5-HT4 受体的 Kis 分别为 0.38 和 373 nM。
  26. GC17706 R-96544 hydrochloride

    R-96544盐酸盐

     5-HT2 receptor antagonist
  27. GC10310 SB 206553 hydrochloride A 5-HT2C and 5-HT2B receptor antagonist
  28. GC15248 GR 125487 sulfamate 5-HT4 receptor antagonist
  29. GC14516 Mesulergine hydrochloride 5-HT2A and 2C receptor antagonist
  30. GC13607 LY 215840 5-HT2/5-HT7 receptor antagonist
  31. GC17140 GR 127935 hydrochloride GR 127935 hydrochloride是一种5-HT1B/1D受体拮抗剂，可抑制降压反应。
  32. GC13298 NAS-181 NAS181 是一种有效的、选择性的大鼠 5-HT1B 受体拮抗剂，Ki 为 47 nM。
  33. GC16556 SB 221284 SB 221284 是一种选择性 5-HT2C/2B 受体拮抗剂，对 5-HT2A、5-HT2B 和 5-HT2C 受体的 pKi 值分别为 6.4、7.9 和 8.6。
  34. GC14347 SB 228357 SB 228357 是一种选择性、有效的口服活性 5-HT2C/2B 受体拮抗剂，5-HT2A、5-HT2B 和 5-HT2C 的 pKi 值分别为 6.9、8.0 和 9.0。
  35. GC12803 SB 204741 SB 204741是一种选择性且高亲和力的5-HT2B受体拮抗剂，其pKi值为7.1。
  36. GC11624 GR 113808 GR 113808是一种有效和选择性的5-HT4受体拮抗剂，pKb=8.8。
  37. GC16653 CP 94253 hydrochloride A 5-HT1B receptor agonist
  38. GC12735 SDZ SER 082 fumarate

    SDZSER082富马酸盐

     5-HT2B/2C receptor antagonist
  39. GC15551 SB 216641 hydrochloride A 5-HT1B receptor antagonist
  40. GC13438 SB 224289 hydrochloride

    SB-224289A

     A 5-HT1B receptor inverse agonist
  41. GC15630 SR 57227 hydrochloride

    SR57227盐酸盐

     SR 57227 hydrochloride是一种强效的serotonin type-3 (5-HT3)受体激动剂，能够穿过血脑屏障。
  42. GC11231 BW 723C86 hydrochloride

    BW723C86盐酸盐

     A selective HT2B receptor agonist
  43. GC17524 GR 55562 dihydrochloride 5-HT1B (5-HT1Dβ) silent antagonist
  44. GC10068 CP 93129 dihydrochloride A 5-HT1B receptor agonist
  45. GC15979 RS 16566 dihydrochloride (R)-zacopride 结合位点的配体
  46. GC16553 N-Desmethylclozapine

    N-去甲基氯氮平; Norclozapine; Desmethylclozapine; Normethylclozapine

     An active metabolite of clozapine
  47. GC14696 RS 67506 hydrochloride potent and selective 5-HT4 partial agonist
  48. GC15137 RS 56812 hydrochloride

    5-HT3 partial agonist
  49. GC17745 MK 212 hydrochloride

    2-氯-6-哌嗪吡嗪盐酸盐,CPP monohydrochloride

     A 5-HT2C receptor agonist
  50. GC11119 MDL 11,939

    MDL11939

     A potent 5-HT2A receptor antagonist
  51. GC14959 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor

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