5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(481)
- GC12744NPS ALX Compound 4a dihydrochlorideCAS: 299433-10-6纯度: >99.00%
NPS ALX Compound 4a dihydrochloride 是一种有效的选择性 5-hydroxytryptamine6 (5-HT6) 受体拮抗剂，IC50 为 7.2 nM，Ki 为 0.2 nM。
- GC12798SB 258719 hydrochlorideCAS: 1217674-10-6
SB 258719 hydrochloride 是一种选择性 5-HT7 受体拮抗剂，对受体具有高亲和力 (pKi=7.5)。
- GC13109FananserinCAS: 127625-29-0纯度: >99.50%
Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。
- GC13549Setiptiline maleateCAS: 85650-57-3纯度: >98.00%
Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。
- GC14052SB 200646 hydrochlorideCAS: 143797-62-0纯度: >99.00%
A dual antagonist of 5-HT 2C and 5-HT 2B receptors
- GC14105Alprenolol hydrochlorideCAS: 13707-88-5纯度: >98.00%
A non-selective β-AR and 5-HT receptor antagonist
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC12735 | SDZ SER 082 fumarate | 141474-54-6 | - | |
5-HT2B/2C receptor antagonist | ||||
| GC12744 | NPS ALX Compound 4a dihydrochloride | 299433-10-6 | >99.00% | |
NPS ALX Compound 4a dihydrochloride 是一种有效的选择性 5-hydroxytryptamine6 (5-HT6) 受体拮抗剂，IC50 为 7.2 nM，Ki 为 0.2 nM。 | ||||
| GC12798 | SB 258719 hydrochloride | 1217674-10-6 | - | |
SB 258719 hydrochloride 是一种选择性 5-HT7 受体拮抗剂，对受体具有高亲和力 (pKi=7.5)。 | ||||
| GC12803 | SB 204741 | 152239-46-8 | >99.50% | |
SB 204741是一种选择性且高亲和力的5-HT2B受体拮抗剂，其pK i 值为7.1。 | ||||
| GC13109 | Fananserin | 127625-29-0 | >99.50% | |
Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。 | ||||
| GC13135 | NBOH-2C-CN hydrochloride | 1539266-32-4 | - | |
5-HT2A agonist | ||||
| GC13265 | Donitriptan hydrochloride | 170911-68-9 | - | |
5-HT1B/1D receptors agonist, potent and selective | ||||
| GC13291 | Prucalopride Succinat | 179474-85-2 | >99.50% | |
A selective 5-HT 4 receptor agonist | ||||
| GC13298 | NAS-181 | 1217474-40-2 | - | |
NAS181 是一种有效的、选择性的大鼠 5-HT1B 受体拮抗剂，Ki 为 47 nM。 | ||||
| GC13369 | R 1485 dihydrochloride | - | - | |
5-HT6 antagonist,selective and high affinity | ||||
| GC13438 | SB 224289 hydrochloride | 180084-26-8 | >99.00% | |
A 5-HT 1B receptor inverse agonist | ||||
| GC13549 | Setiptiline maleate | 85650-57-3 | >98.00% | |
Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。 | ||||
| GC13583 | CJ 033466 | 519148-48-2 | - | |
CJ 033466 是一种新型选择性 5-HT4 受体部分激动剂，EC50 为 9 nM，具有促胃动力作用。 | ||||
| GC13607 | LY 215840 | 137328-52-0 | - | |
5-HT2/5-HT7 receptor antagonist | ||||
| GC13627 | Ziprasidone hydrochloride monohydrate | 138982-67-9 | >99.50% | |
An atypical antipsychotic | ||||
| GC13654 | Alosetron | 122852-42-0 | - | |
A 5-HT 3 receptor antagonist | ||||
| GC13883 | Ritanserin | 87051-43-2 | >99.50% | |
A potent 5-HT 2A receptor antagonist | ||||
| GC13977 | MS 245 oxalate | 275363-58-1 | - | |
A 5-HT 6 receptor antagonist | ||||
| GC13990 | Setiptiline | 57262-94-9 | - | |
Setiptiline (Org-8282) 是一种血清素受体拮抗剂。 | ||||
| GC14030 | Altanserin hydrochloride | 1135280-78-2 | - | |
5-HT2A receptor antagonist | ||||
| GC14052 | SB 200646 hydrochloride | 143797-62-0 | >99.00% | |
A dual antagonist of 5-HT 2C and 5-HT 2B receptors | ||||
| GC14083 | MDL 72222 | 40796-97-2 | >99.00% | |
MDL 72222 (MDL 72222) 是一种选择性 5-HT3 受体拮抗剂，IC50 为 0.33 nM。 | ||||
| GC14088 | Zotepine | 26615-21-4 | - | |
An atypical antipsychotic | ||||
| GC14105 | Alprenolol hydrochloride | 13707-88-5 | >98.00% | |
A non-selective β-AR and 5-HT receptor antagonist | ||||