Histamine Receptor
Histamine Receptor(组胺受体)
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
Histamine Receptor 相关产品(236)
- GC18198CarebastineCAS: 90729-42-3纯度: >99.00%
An active metabolite of ebastine and a histamine H 1 receptor antagonist
- GC25060AmitriptylineCAS: 50-48-6
Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties, widely used to treat depression and neuropathic pain. Amitriptyline is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. Amitriptyline also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. This product is a waxy solid.
- GC25136Betazole DihydrochlorideCAS: 138-92-1纯度: >99.00%
Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function.
- GC25571LevocetirizineCAS: 130018-77-8
Levocetirizine (LCZ, (R)-Cetirizine), the R-enantiomer of cetirizine, is an antagonist of histamine H(1) receptor.
- GC25785PromethazineCAS: 60-87-7纯度: >98.00%
Promethazine is a potent histamine H1 receptor antagonist. Promethazine is a medication used in the management and treatment of allergic conditions, nausea and vomiting, motion sickness, and sedation. Promethazine exhibits antiparasitic properties.
- GC30902DimenhydrinateCAS: 523-87-5纯度: >99.50%
Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC17564 | VUF 8430 dihydrobromide | 100130-32-3 | >95.00% | |
A histamine H 4 receptor agonist | ||||
| GC17585 | VUF 10460 | 1028327-66-3 | >98.00% | |
A histamine H 4 receptor agonist | ||||
| GC17701 | Clemizole hydrochloride | 1163-36-6 | >99.50% | |
An antihistamine and TRPC5 channel blocker | ||||
| GC17743 | A 987306 | 1082954-71-9 | - | |
A 987306 是一种有效的、可口服的组胺 H4 拮抗剂，对大鼠 H4 和人 H4 的 Kis 分别为 3.4 nM 和 5.8 nM。 | ||||
| GC17869 | Histamine Phosphate | 51-74-1 | >98.00% | |
A biogenic amine | ||||
| GC17974 | Latrepirdine dihydrochloride | 97657-92-6 | >99.50% / >98.00% | |
A neuroprotective agent | ||||
| GC18198 | Carebastine | 90729-42-3 | >99.00% | |
An active metabolite of ebastine and a histamine H 1 receptor antagonist | ||||
| GC18282 | Lodoxamide | 53882-12-5 | >99.50% | |
A potent agonist of GPR35 and a mast cell stabilizer | ||||
| GC18463 | N-acetyl Histamine | 673-49-4 | >99.50% | |
A histamine metabolite | ||||
| GC19178 | GSK189254A | 720690-73-3 | >98.00% | |
A histamine H 3 receptor antagonist | ||||
| GC19441 | Levocabastine (hydrochloride) | 79547-78-7 | >98.00% | |
A histamine H 1 receptor antagonist | ||||
| GC25060 | Amitriptyline | 50-48-6 | - | |
Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties, widely used to treat depression and neuropathic pain. Amitriptyline is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. Amitriptyline also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. This product is a waxy solid. | ||||
| GC25136 | Betazole Dihydrochloride | 138-92-1 | >99.00% | |
Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function. | ||||
| GC25571 | Levocetirizine | 130018-77-8 | - | |
Levocetirizine (LCZ, (R)-Cetirizine), the R-enantiomer of cetirizine, is an antagonist of histamine H(1) receptor. | ||||
| GC25785 | Promethazine | 60-87-7 | >98.00% | |
Promethazine is a potent histamine H1 receptor antagonist. Promethazine is a medication used in the management and treatment of allergic conditions, nausea and vomiting, motion sickness, and sedation. Promethazine exhibits antiparasitic properties. | ||||
| GC30423 | CP-66948 | 101189-47-3 | - | |
CP-66948是histamineH2受体拮抗剂，能够抑制胃酸分泌，保护粘膜的作用。 | ||||
| GC30455 | Rocastine (AHR-11325) | 91833-49-7 | - | |
Rocastine (AHR-11325) 是一种选择性、非镇静 H1 拮抗剂，用作抗组胺药。 | ||||
| GC30496 | Doxylamine D5 succinate | 1216840-94-6 | - | |
DoxylamineD5琥珀酸盐是Doxylamine氘代化合物标准品。 | ||||
| GC30759 | H3 receptor-MO-1 | 1240914-03-7 | - | |
H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。 | ||||
| GC30775 | Histamine (Ergamine) | 51-45-6 | >99.00% / >98.00% | |
A biogenic amine | ||||
| GC30821 | JNJ-39758979 | 1046447-90-8 | >98.00% | |
JNJ-39758979是一个有选择性且具有高亲和性的组胺H4受体拮抗剂,其Ki值为12.5nM。 | ||||
| GC30902 | Dimenhydrinate | 523-87-5 | >99.50% | |
Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness. | ||||
| GC30948 | Chlorphenoxamine | 77-38-3 | - | |
Chlorphenoxamine是一种抗组胺剂和抗胆碱能药,用作抗帕金森氏病。 | ||||
| GC30999 | Pimethixene (Pimetixene) | 314-03-4 | - | |
Pimethixene (Pimetixene) 是抗组胺药和抗血清素能化合物，用作抗偏头痛剂。 | ||||