COX
COX(环氧合酶)
COX (cyclooxygenase) is an enzyme that is responsible for formation of important biological mediators called prostanoids, including prostaglandins, prostacyclin and thromboxane.
COX 相关产品(291)
- GC16294Ibuprofen LysineCAS: 57469-77-9
Ibuprofen ((±)-Ibuprofen) L-lysine 是一种有效的具有口服活性的选择性 COX-1 抑制剂,IC50 值为 13 μM.
- GC17556IndomethacinCAS: 53-86-1纯度: >99.50% / >99.00%
Indomethacin(吲哚美辛)是一种有效的口服活性 COX1/2 抑制剂,COX-1 和 COX-2 的IC50 值分别为 18 nM 和 26 nM。
- GC17776AsaraldehydeCAS: 4460-86-0纯度: >99.50%
Asarylaldehyde (Asaronaldehyde) 是一种 COX-2 抑制剂,可显着抑制环氧合酶 II (COX-2) 的活性,IC50 值为 100 μg/mL。
- GC10603(-)-epicatechin gallateCAS: 1257-08-5纯度: >98.00%
(-)-epicatechin gallate是一种天然黄烷醇,属于茶多酚中的酯型儿茶素类化合物,(-)-epicatechin gallate通过抑制环加氧酶-1(COX-1)发挥抗炎作用(IC₅₀=7.5μM)。
- GC10611N-(4-acetamidophenyl)-Indomethacin amideCAS: 261766-23-8
Potent and selective reversible inhibitor of COX-2
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15634 | SC 560 | 188817-13-2 | >99.50% | |
A selective inhibitor of COX-1 | ||||
| GC15928 | Phenacetin | 62-44-2 | >99.50% | |
An Analytical Reference Standard | ||||
| GC16077 | Deracoxib | 169590-41-4 | >99.50% | |
An NSAID and selective COX-2 inhibitor | ||||
| GC16294 | Ibuprofen Lysine | 57469-77-9 | - | |
Ibuprofen ((±)-Ibuprofen) L-lysine 是一种有效的具有口服活性的选择性 COX-1 抑制剂,IC50 值为 13 μM. | ||||
| GC16508 | Salicylic acid | 69-72-7 | >98.00% | |
An Analytical Reference Standard | ||||
| GC16594 | Ketorolac tromethamine salt | 74103-07-4 | >99.50% | |
An NSAID and COX inhibitor | ||||
| GC16662 | Etodolac | 41340-25-4 | >99.00% | |
An NSAID | ||||
| GC16716 | Sulindac | 38194-50-2 | >99.50% | |
A non-selective COX inhibitor | ||||
| GC16721 | Licofelone | 156897-06-2 | >98.00% | |
A dual inhibitor of COX-1/COX-2 and 5-LO | ||||
| GC16790 | Piroxicam | 36322-90-4 | >99.50% | |
A COX inhibitor and NSAID | ||||
| GC16881 | FR 122047 hydrochloride | 130717-51-0 | - | |
A selective COX-1 inhibitor | ||||
| GC17051 | Parecoxib Sodium | 198470-85-8 | >99.50% | |
A prodrug form of valdecoxib | ||||
| GC17556 | Indomethacin | 53-86-1 | >99.50% / >99.00% | |
Indomethacin(吲哚美辛)是一种有效的口服活性 COX1/2 抑制剂,COX-1 和 COX-2 的IC50 值分别为 18 nM 和 26 nM。 | ||||
| GC17776 | Asaraldehyde | 4460-86-0 | >99.50% | |
Asarylaldehyde (Asaronaldehyde) 是一种 COX-2 抑制剂,可显着抑制环氧合酶 II (COX-2) 的活性,IC50 值为 100 μg/mL。 | ||||
| GC17817 | SC 58125 | 162054-19-5 | - | |
A selective COX-2 inhibitor | ||||
| GC17863 | Ibuprofen | 15687-27-1 | >99.50% | |
An NSAID and non-selective COX inhibitor | ||||
| GC18084 | Nimesulide | 51803-78-2 | >99.50% | |
An NSAID and COX2 inhibitor | ||||
| GC10006 | Tenoxicam | 59804-37-4 | >99.50% | |
An NSAID and COX-1 inhibitor | ||||
| GC10335 | Valeroyl Salicylate | 64206-54-8 | - | |
A selective, irreversible inhibitor of COX-1 | ||||
| GC10429 | Etoricoxib | 202409-33-4 | >99.00% | |
A selective COX-2 inhibitor | ||||
| GC10603 | (-)-epicatechin gallate | 1257-08-5 | >98.00% | |
(-)-epicatechin gallate是一种天然黄烷醇,属于茶多酚中的酯型儿茶素类化合物,(-)-epicatechin gallate通过抑制环加氧酶-1(COX-1)发挥抗炎作用(IC₅₀=7.5μM)。 | ||||
| GC10611 | N-(4-acetamidophenyl)-Indomethacin amide | 261766-23-8 | - | |
Potent and selective reversible inhibitor of COX-2 | ||||
| GC10873 | α-Spinasterol | 481-18-5 | >99.00% | |
A TRPV1 antagonist | ||||
| GC11049 | (+/-)-Sulfinpyrazone | 57-96-5 | >99.00% | |
An inhibitor of uric acid reabsorption | ||||
