5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(419)
- GC11984Isamoltane hemifumarateCAS: 874882-92-5
Isamoltane hemifumarate 是 5-HT1B 受体的选择性拮抗剂，抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B 识别位点的结合，IC50 为 39 nM。
- GC12986RisperidoneCAS: 106266-06-2纯度: >98.00%
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂，对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11824 | Asenapine | 65576-45-6 | >98.50% | |
An atypical antipsychotic | ||||
| GC11959 | Naratriptan | 143388-64-1 | >98.00% | |
A potent 5-HT 1B and 5-HT 1D receptor agonist | ||||
| GC11984 | Isamoltane hemifumarate | 874882-92-5 | - | |
Isamoltane hemifumarate 是 5-HT1B 受体的选择性拮抗剂，抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B 识别位点的结合，IC50 为 39 nM。 | ||||
| GC12091 | SB742457 | 607742-69-8 | >98.00% | |
A 5-HT 6 receptor antagonist | ||||
| GC12276 | CGS 12066B dimaleate | 109028-10-6 | >98.00% | |
A 5-HT 1B receptor agonist | ||||
| GC12398 | Granisetron | 109889-09-0 | - | |
Granisetron (BRL 43694) 是一种血清素 5-HT3 受体拮抗剂，用作止吐剂，用于治疗化疗后的恶心和呕吐。 | ||||
| GC12427 | 8-Hydroxy-PIPAT oxalate | 159651-91-9 | - | |
5-HT1A receptor agonist | ||||
| GC12495 | Olanzapine | 132539-06-1 | >99.00% / >98.00% / >99.50% | |
Olanzapine是一种单胺拮抗剂。 | ||||
| GC12541 | Bilobalide | 33570-04-6 | >98.00% | |
A neuroprotective natural product | ||||
| GC12632 | Cyanopindolol hemifumarate | 106469-57-2 | - | |
5-HT1A/1B antagonist and β-adrenoceptor antagonist | ||||
| GC12782 | CP-809101 hydrochloride | 1215721-40-6 | >99.50% | |
A potent 5-HT 2C receptor agonist | ||||
| GC12986 | Risperidone | 106266-06-2 | >98.00% | |
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂，对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。 | ||||
| GC13053 | Pizotifen | 15574-96-6 | >98.00% | |
A triptan | ||||
| GC13081 | Loxapine | 1977-10-2 | >99.50% | |
洛沙平是一种口服活性多巴胺抑制剂、5-HT 受体拮抗剂，也是一种二苯并沙西平抗精神病药物。 | ||||
| GC13092 | Fluvoxamine | 54739-18-3 | - | |
Fluvoxamine是一种选择性血清素（5-HT）再摄取抑制剂（SSRI），具有抗抑郁活性。 | ||||
| GC13133 | Ipsapirone | 95847-70-4 | >99.00% | |
A partial agonist of serotonin 5-HT 1A receptors | ||||
| GC13428 | Mosapride | 112885-41-3 | - | |
A 5-HT 4 receptor agonist | ||||
| GC13478 | Pizotifen Malate | 5189-11-7 | - | |
A triptan | ||||
| GC13501 | VUF 10166 | 155584-74-0 | - | |
A 5-HT 3 receptor antagonist | ||||
| GC13533 | Cisapride | 81098-60-4 | >99.50% | |
A 5-HT 4 receptor agonist | ||||
| GC13627 | Ziprasidone hydrochloride monohydrate | 138982-67-9 | >99.50% | |
An atypical antipsychotic | ||||
| GC13654 | Alosetron | 122852-42-0 | - | |
A 5-HT 3 receptor antagonist | ||||
| GC13723 | Amitriptyline HCl | 549-18-8 | >99.50% | |
A tricyclic antidepressant | ||||
| GC13871 | Duloxetine HCl | 136434-34-9 | >99.50% | |
A serotonin and norepinephrine reuptake inhibitor | ||||