GlpBio

5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

5-HT Receptor 相关产品(419)

  • GC17808 structure
    GC17808Zolmitriptan
    CAS: 139264-17-8
    纯度: >99.50% / >98.00%

    An agonist of 5-HT 1B and 5-HT 1D receptors

  • GC17917 structure
    GC17917Palonosetron HCl
    CAS: 135729-62-3
    纯度: >99.50%

    A 5-HT 3 receptor antagonist

  • GC17981 structure
    GC17981Agomelatine
    CAS: 138112-76-2
    纯度: >98.50%

    Agomelatine是一种褪黑素（MT）受体激动剂，对MT1和MT2的K i 值分别为0.1 nM和0.12 nM。Agomelatine也是一种5-羟色胺（5-HT）受体拮抗剂，对5-HT 2C 和5-HT 2B 的K i 值分别为631 nM和660 nM。

  • GC18006 structure
    GC18006Sumatriptan Succinate
    CAS: 103628-48-4
    纯度: >99.50%

    Sumatriptan Succinate是一种具有口服活性的5-HT1受体激动剂，对5-HT1D、5-HT1B和5-HT1F受体的IC 50 值分别为7.3nM、9.3nM和17.8nM。

  • GC18013 structure
    GC18013S 14506 hydrochloride
    CAS: 286369-38-8

    A 5-HT 1A receptor agonist

  • GC18102 structure
    GC18102Paroxetine maleate
    CAS: 64006-44-6

    5-HT uptake inhibitor

  • GC10051 structure
    GC10051MDL 100907
    CAS: 139290-65-6
    纯度: >98.00%

    Selective antagonist of the serotonin receptor 5-HT 2A

  • GC10117 structure
    GC10117Aripiprazole
    CAS: 129722-12-9
    纯度: >99.50%

    An atypical antipsychotic

  • GC10242 structure
    GC10242Loxapine Succinate
    CAS: 27833-64-3
    纯度: >99.50%

    An atypical antipsychotic drug

  • GC10357 structure
    GC10357Metergoline
    CAS: 17692-51-2
    纯度: >99.50%

    A serotonin receptor antagonist

  • GC10614 structure
    GC10614Rotigotine
    CAS: 99755-59-6
    纯度: >99.50%

    A non-selective dopamine receptor agonist

  • GC10670 structure
    GC10670RS 127445 HCl

    5-HT2B receptor antagonist,high affinity

  • GC10698 structure
    GC10698Cyproheptadine hydrochloride
    CAS: 969-33-5
    纯度: >99.50%

    An antihistamine with antiserotonergic and anticholinergic activities

  • GC10743 structure
    GC10743Cyclobenzaprine HCl
    CAS: 6202-23-9
    纯度: >99.50%

    An Analytical Reference Material

  • GC10891 structure
    GC10891Alverine Citrate
    CAS: 5560-59-8
    纯度: >99.00%

    An antispasmodic agent

  • GC11033 structure
    GC11033Rupatadine Fumarate
    CAS: 182349-12-8
    纯度: >99.50%

    A histamine H 1 and PAF receptor antagonist

  • GC11100 structure
    GC11100Flibanserin
    CAS: 167933-07-5
    纯度: >99.00%

    A 5-HT 1A receptor agonist and 5-HT 2A receptor antagonist

  • GC11176 structure
    GC111762-Methyl-5-hydroxytryptamine hydrochloride
    CAS: 845861-49-6

    2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。

  • GC11186 structure
    GC11186Brexpiprazole
    CAS: 913611-97-9
    纯度: >97.00%

    Brexpiprazole是一种口服非典型抗精神病药物，是5-HT1A（K i =0.12nM）和dopamine D2L（K i =0.3nM）受体的强效部分激动剂，以及5-HT2A受体（K i =0.47nM）的拮抗剂。

  • GC11191 structure
    GC11191Buspirone HCl
    CAS: 33386-08-2
    纯度: >99.50% / >99.00%

    An Analytical Reference Standard

  • GC11447 structure
    GC11447Mirtazapine
    CAS: 85650-52-8
    纯度: >99.50%

    Mirtazapine是一种去甲肾上腺素能和特异性血清素抗抑郁药（NaSSA），可抑制5-HT 2A 、5-HT 2B 、5-HT 2C 和5-HT 3 受体，pK i 值分别为8.2、6.7、7.9和8.1。

  • GC11556 structure
    GC11556AL 34662
    CAS: 210580-75-9

    A potent 5-HT 2 receptor agonist

  • GC11624 structure
    GC11624GR 113808
    CAS: 144625-51-4
    纯度: >98.00% / >99.50%

    GR 113808是一种有效和选择性的5-HT4受体拮抗剂，pK b =8.8。

  • GC11814 structure
    GC11814Ondansetron HCl
    CAS: 99614-01-4
    纯度: >98.00%

    A Certified Reference Material