GlpBio

5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

5-HT Receptor 相关产品(419)

  • GC11844 structure
    GC11844Pimavanserin
    CAS: 706779-91-1
    纯度: >99.50%

    A 5-HT 2A inverse agonist

  • GC11962 structure
    GC11962Lu AE58054 Hydrochloride
    CAS: 467458-02-2
    纯度: >99.50%

    A 5-HT 6 receptor antagonist

  • GC11977 structure
    GC11977Thioridazine HCl
    CAS: 130-61-0
    纯度: >99.50%

    A typical antipsychotic

  • GC11989 structure
    GC11989Nortriptyline (hydrochloride)
    CAS: 894-71-3
    纯度: >99.50%

    A tricyclic antidepressant

  • GC12293 structure
    GC12293Perphenazine
    CAS: 58-39-9
    纯度: >99.50%

    A typical antipsychotic

  • GC12535 structure
    GC12535Flopropione
    CAS: 2295-58-1
    纯度: >98.50%

    Flopropione 是一种 5-HT 受体拮抗剂，也是一种儿茶酚-邻甲基转移酶 (COMT) 抑制剂。

  • GC12885 structure
    GC12885Imipramine (hydrochloride)
    CAS: 113-52-0
    纯度: >99.50% / >98.00%

    A tricyclic antidepressant

  • GC13109 structure
    GC13109Fananserin
    CAS: 127625-29-0
    纯度: >99.50%

    Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。

  • GC13291 structure
    GC13291Prucalopride Succinat
    CAS: 179474-85-2
    纯度: >99.50%

    A selective 5-HT 4 receptor agonist

  • GC13438 structure
    GC13438SB 224289 hydrochloride
    CAS: 180084-26-8
    纯度: >99.00%

    A 5-HT 1B receptor inverse agonist

  • GC13549 structure
    GC13549Setiptiline maleate
    CAS: 85650-57-3
    纯度: >98.00%

    Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。

  • GC13883 structure
    GC13883Ritanserin
    CAS: 87051-43-2
    纯度: >99.50%

    A potent 5-HT 2A receptor antagonist

  • GC13990 structure
    GC13990Setiptiline
    CAS: 57262-94-9

    Setiptiline (Org-8282) 是一种血清素受体拮抗剂。

  • GC14000 structure
    GC140006-fluoro-DL-Tryptophan
    CAS: 7730-20-3

    A serotonin synthesis inhibitor

  • GC14083 structure
    GC14083MDL 72222
    CAS: 40796-97-2
    纯度: >99.00%

    MDL 72222 (MDL 72222) 是一种选择性 5-HT3 受体拮抗剂，IC50 为 0.33 nM。

  • GC14105 structure
    GC14105Alprenolol hydrochloride
    CAS: 13707-88-5
    纯度: >98.00%

    A non-selective β-AR and 5-HT receptor antagonist

  • GC14167 structure
    GC14167Quetiapine
    CAS: 111974-69-7
    纯度: >98.00%

    Quetiapine是一种5-HT受体激动剂，对人类5-HT1A受体的 pEC 50 为4.77。Quetiapine是一种多巴胺受体拮抗剂，对人类D2受体的pIC 50 为6.33。Quetiapine是一种非典型抗精神病药，用于治疗精神分裂症、躁郁症和重度抑郁症。

  • GC14216 structure
    GC14216Chlorpromazine HCl
    CAS: 69-09-0
    纯度: >99.50%

    Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药，能够有效抑制D2多巴胺受体和5-HT 2A ，具有很强的镇静作用。

  • GC14343 structure
    GC143433,4-dihydro Naratriptan
    CAS: 121679-20-7

    An impurity in the preparation of naratriptan

  • GC14392 structure
    GC14392SB 242084
    CAS: 181632-25-7
    纯度: >98.00%

    Specific antagonist of 5-HT 2C

  • GC14558 structure
    GC14558Dihydroergotamine mesylate
    CAS: 6190-39-2
    纯度: >99.50%

    An agonist of 5-HT 1B and 5-HT 1D receptors

  • GC14583 structure
    GC14583R 59-022
    CAS: 93076-89-2
    纯度: 不显示

    R 59-022是一种二酰甘油激酶抑制剂（IC 50 = 2.8µM）。

  • GC14657 structure
    GC14657Rotundine
    CAS: 483-14-7
    纯度: >99.50%

    An antinociceptive alkaloid

  • GC14843 structure
    GC14843Serotonin HCl
    CAS: 153-98-0
    纯度: >99.50% / >98.00%

    Serotonin HCl是一种神经递质，是介导人体多种中枢和外周功能的关键信使。