5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

5-HT Receptor 相关产品(419)

GC14940 5-Methoxytryptamine
CAS: 608-07-1
纯度: >99.00%
GC15367 EMDT oxalate
CAS: 263744-72-5
EMDT 草酸盐是一种选择性 5-HT6 激动剂，具有抗抑郁作用。
GC15639 Ramosetron Hydrochloride
CAS: 132907-72-3
纯度: >99.50%
A potent, selective 5-HT 3 receptor antagonist
GC15660 SB 399885 hydrochloride
CAS: 402713-81-9
纯度: >99.50%
A 5-HT 6 receptor antagonist
GC15985 Cariprazine
CAS: 839712-12-8
纯度: >99.00%
An atypical antipsychotic
GC16017 Rotigotine hydrochloride
CAS: 125572-93-2
纯度: >99.00%
A non-selective dopamine receptor agonist
GC16135 Cinanserin hydrochloride
CAS: 54-84-2
纯度: >99.50%
A 5-HT receptor antagonist
GC16202 Sarpogrelate hydrochloride
CAS: 135159-51-2
纯度: >98.00%
Sarpogrelate hydrochloride是一种高选择性5-羟色胺（5-HT）2受体拮抗剂（5-HT 2A : pK i = 8.52；5-HT 2B : pK i = 6.57；5-HT 2C : pK i = 7.43）。
GC16324 Nefazodone hydrochloride
CAS: 82752-99-6
纯度: >98.00%
A serotonin, norepinephrine, and dopamine reuptake inhibitor
GC16634 Sumatriptan
CAS: 103628-46-2
纯度: >98.00%
Sumatriptan是一种具有口服活性的5-HT1受体激动剂，对5-HT1D、5-HT1B和5-HT1F受体的IC 50 值分别为7.3nM、9.3nM和17.8nM。
GC16891 Quetiapine Fumarate
CAS: 111974-72-2
纯度: >98.00%
An antagonist of diverse neurological receptors
GC17488 Trimipramine (maleate)
CAS: 521-78-8
纯度: >99.50% / >98.00%
A tricyclic antidepressant
GC17525 AS 19
CAS: 1000578-26-6
纯度: >98.00%
A 5-HT 7 receptor agonist
GC17734 Pindolol
CAS: 13523-86-9
纯度: >99.50% / >99.00%
A β 1 - and β 2 -AR antagonist
GC17826 Tegaserod maleate
CAS: 189188-57-6
纯度: >98.00%
A potent 5-HT 4 agonist
GC17854 PNU 142633
CAS: 187665-65-2
纯度: >98.00%
PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂，对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
GC17974 Latrepirdine dihydrochloride
CAS: 97657-92-6
纯度: >99.50% / >98.00%
A neuroprotective agent
GC18244 Eltoprazine (hydrochloride)
CAS: 98206-09-8
纯度: >99.50%
A partial agonist of 5-HT 1A , 5-HT 1B , and 5-HT 2B receptors
GC19176 GSK163090
CAS: 844903-58-8
纯度: >99.50%
GSK163090 是一种有效的、选择性的和具有口服活性的 5-HT1A/1B/1D 受体拮抗剂，pKi 值分别为 9.4/8.5/9.7。
GC19294 Piboserod
CAS: 152811-62-6
纯度: >98.00%
A selective, potent 5-HT 4 receptor antagonist
GC19354 TG6-10-1
CAS: 1415716-58-3
纯度: >99.50%
A potent EP 2 receptor antagonist
GC19389 YL0919
CAS: 1339058-04-6
纯度: >99.50%
YL0919 (YL0919) 是一种具有双重活性的口服抗抑郁药，作为高度选择性的 5-HT 摄取阻滞剂和有效的 5-HT1Areceptor 激动剂 (Ki=0.19 nM)。
GC25253 Cinitapride Hydrogen Tartrate
CAS: 1207859-16-2
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors
GC25259 Cisapride hydrate
CAS: 260779-88-2
Cisapride (Propulsid, Alimix, Propulsin, Enteropride, Kinestase) acts directly as a selective serotonin 5-HT4 receptor agonist with IC50 of 0.483 μM. And It also acts indirectly as a parasympathomimetic.

分类产品列表
货号	产品名称	CAS号	纯度
GC14940	5-Methoxytryptamine	608-07-1	>99.00%
GC15367	EMDT oxalate	263744-72-5	-
GC15367	EMDT 草酸盐是一种选择性 5-HT6 激动剂，具有抗抑郁作用。
GC15639	Ramosetron Hydrochloride	132907-72-3	>99.50%
GC15639	A potent, selective 5-HT 3 receptor antagonist
GC15660	SB 399885 hydrochloride	402713-81-9	>99.50%
GC15660	A 5-HT 6 receptor antagonist
GC15985	Cariprazine	839712-12-8	>99.00%
GC15985	An atypical antipsychotic
GC16017	Rotigotine hydrochloride	125572-93-2	>99.00%
GC16017	A non-selective dopamine receptor agonist
GC16135	Cinanserin hydrochloride	54-84-2	>99.50%
GC16135	A 5-HT receptor antagonist
GC16202	Sarpogrelate hydrochloride	135159-51-2	>98.00%
GC16202	Sarpogrelate hydrochloride是一种高选择性5-羟色胺（5-HT）2受体拮抗剂（5-HT 2A : pK i = 8.52；5-HT 2B : pK i = 6.57；5-HT 2C : pK i = 7.43）。
GC16324	Nefazodone hydrochloride	82752-99-6	>98.00%
GC16324	A serotonin, norepinephrine, and dopamine reuptake inhibitor
GC16634	Sumatriptan	103628-46-2	>98.00%
GC16634	Sumatriptan是一种具有口服活性的5-HT1受体激动剂，对5-HT1D、5-HT1B和5-HT1F受体的IC 50 值分别为7.3nM、9.3nM和17.8nM。
GC16891	Quetiapine Fumarate	111974-72-2	>98.00%
GC16891	An antagonist of diverse neurological receptors
GC17488	Trimipramine (maleate)	521-78-8	>99.50% / >98.00%
GC17488	A tricyclic antidepressant
GC17525	AS 19	1000578-26-6	>98.00%
GC17525	A 5-HT 7 receptor agonist
GC17734	Pindolol	13523-86-9	>99.50% / >99.00%
GC17734	A β 1 - and β 2 -AR antagonist
GC17826	Tegaserod maleate	189188-57-6	>98.00%
GC17826	A potent 5-HT 4 agonist
GC17854	PNU 142633	187665-65-2	>98.00%
GC17854	PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂，对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
GC17974	Latrepirdine dihydrochloride	97657-92-6	>99.50% / >98.00%
GC17974	A neuroprotective agent
GC18244	Eltoprazine (hydrochloride)	98206-09-8	>99.50%
GC18244	A partial agonist of 5-HT 1A , 5-HT 1B , and 5-HT 2B receptors
GC19176	GSK163090	844903-58-8	>99.50%
GC19176	GSK163090 是一种有效的、选择性的和具有口服活性的 5-HT1A/1B/1D 受体拮抗剂，pKi 值分别为 9.4/8.5/9.7。
GC19294	Piboserod	152811-62-6	>98.00%
GC19294	A selective, potent 5-HT 4 receptor antagonist
GC19354	TG6-10-1	1415716-58-3	>99.50%
GC19354	A potent EP 2 receptor antagonist
GC19389	YL0919	1339058-04-6	>99.50%
GC19389	YL0919 (YL0919) 是一种具有双重活性的口服抗抑郁药，作为高度选择性的 5-HT 摄取阻滞剂和有效的 5-HT1Areceptor 激动剂 (Ki=0.19 nM)。
GC25253	Cinitapride Hydrogen Tartrate	1207859-16-2	-
GC25253	Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors
GC25259	Cisapride hydrate	260779-88-2	-
GC25259	Cisapride (Propulsid, Alimix, Propulsin, Enteropride, Kinestase) acts directly as a selective serotonin 5-HT4 receptor agonist with IC50 of 0.483 μM. And It also acts indirectly as a parasympathomimetic.