5-HT Receptor
5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
5-HT Receptor 相关产品(419)
- GC14093Indatraline hydrochlorideCAS: 96850-13-4
Indatraline hydrochloride (Lu 19-005) 是一种非选择性单胺转运蛋白抑制剂,可阻断神经递质(多巴胺、血清素和去甲肾上腺素)的再摄取,其功效与可卡因相似。
- GC14518Asenapine hydrochlorideCAS: 1412458-61-7纯度: >99.50%
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。
- GC15013VilazodoneCAS: 163521-12-8纯度: >99.00%
Vilazodone (EMD 68843; SB 659746A) 是一种强效、选择性和口服活性的血清素再摄取抑制剂 (SSRI) 和部分 5-HT1A 受体激动剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC14008 | Anpirtoline hydrochloride | 99201-87-3 | - | |
5-HT1B receptor agonist | ||||
| GC14019 | MDL 73005EF hydrochloride | 102908-60-1 | - | |
5-HT1A receptor antagonist | ||||
| GC14035 | Citalopram hydrobromide | 59729-32-7 | >99.50% | |
A selective serotonin reuptake inhibitor | ||||
| GC14093 | Indatraline hydrochloride | 96850-13-4 | - | |
Indatraline hydrochloride (Lu 19-005) 是一种非选择性单胺转运蛋白抑制剂,可阻断神经递质(多巴胺、血清素和去甲肾上腺素)的再摄取,其功效与可卡因相似。 | ||||
| GC14160 | Blonanserin | 132810-10-7 | >98.50% | |
A dopamine and serotonin receptor antagonist | ||||
| GC14262 | Desvenlafaxine Succinate | 386750-22-7 | >99.50% | |
An active metabolite of venlafaxine | ||||
| GC14437 | Vortioxetine (Lu AA21004) HBr | 960203-27-4 | >99.50% | |
A multimodal serotonergic agent | ||||
| GC14491 | B-HT 920 | 36085-73-1 | >99.50% | |
A potent agonist of D 2 receptors | ||||
| GC14512 | Fenspiride HCl | 5053-08-7 | >99.50% | |
A histamine H 1 receptor antagonist | ||||
| GC14518 | Asenapine hydrochloride | 1412458-61-7 | >99.50% | |
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。 | ||||
| GC14550 | SB271046 | 209481-20-9 | - | |
An orally-available 5-HT 6 antagonist | ||||
| GC14563 | Ketanserin | 74050-98-9 | >99.00% / >97.00% | |
A potent 5-HT 2 receptor antagonist | ||||
| GC14743 | WY 45233 succinate | 448904-47-0 | - | |
serotonin and noradrenalin reuptake inhibitor | ||||
| GC14788 | Tianeptine | 66981-73-5 | >98.00% | |
An atypical antidepressant | ||||
| GC14805 | (S)-WAY 100135 dihydrochloride | 149007-54-5 | - | |
A 5-HT 1A receptor antagonist | ||||
| GC14891 | MM 77 dihydrochloride | 159187-70-9 | - | |
MM 77 dihydrochloride 是一种有效的 5-HT1A 受体的突触后拮抗剂。 | ||||
| GC14927 | Trazodone HCl | 25332-39-2 | >98.00% | |
An Analytical Reference Material | ||||
| GC14966 | 8-Hydroxy-DPAT hydrobromide | 76135-31-4 | - | |
A 5-HT 1A receptor agonist | ||||
| GC15013 | Vilazodone | 163521-12-8 | >99.00% | |
Vilazodone (EMD 68843; SB 659746A) 是一种强效、选择性和口服活性的血清素再摄取抑制剂 (SSRI) 和部分 5-HT1A 受体激动剂。 | ||||
| GC15025 | Fluvoxamine maleate | 61718-82-9 | >99.50% | |
A selective serotonin reuptake inhibitor | ||||
| GC15107 | Clomipramine HCl | 17321-77-6 | >99.00% | |
A tricyclic antidepressant | ||||
| GC15121 | Lasmiditan | 439239-90-4 | - | |
An Analytical Reference Standard | ||||
| GC15153 | Almotriptan Malate | 181183-52-8 | >98.00% | |
An agonist of 5-HT 1B and 5-HT 1D receptors | ||||
| GC15223 | Tropisetron Hydrochloride | 105826-92-4 | >99.50% | |
A 5-HT 3 receptor antagonist | ||||
