关于 "Nuclear Receptors" 的结果29+ 个结果

一种Nurr1受体激动剂

A nuclear receptor cell-based reporter assay

Nuclear Receptor Binding Factor 2 Human Recombinant

Nuclear Receptor-Interacting Protein 3 Human Recombinant

Proline-Rich Nuclear Receptor Coactivator 2 Human Recombinant

An agonist of the heme-dependent nuclear receptor REV-ERBα

Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain

CIA 1 is an inhibitor of the nuclear receptor COUP-TFII (IC50 ranged from 1.2 μM to 7.6 μM, in prostate cancer cell lines).

TLX agonist 1 (CCRP2, SUN23314) is a modulator of orphan nuclear receptor tailless (TLX, NR2E1) with EC50 of 1.0 μM and Kd of 650 nM. TLX agonist 1 (CCRP2, SUN23314) binds to recombinant TLX protein and enhances TLX transcriptional repressive activity.

AZD-5153 6-hydroxy-2-naphthoic acid (HNT salt) is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor with pKi of 8.3 for BRD4. AZD-5153 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes. NSD3, via H3K36me2, acts as an epigenetic deregulator to facilitate the expression of oncogenesis-promoting genes.

A fluorescent DNA probe for live and fixed cells

NucPE1 (Nuclear Peroxy Emerald 1) (Nuclear Peroxy Emerald 1) 是一种核定位荧光过氧化氢，可特异性定位于细胞核，而无需附加靶向部分。

NLS, cell-penetrating peptide containing 7 amino acids homologous to the SV40 T antigen, was capable of inducing the transport of several carrier proteins to the nucleus. The terminal cysteine permits the attachment of this peptide to any protein using a heterobifunctional crosslinking reagent. Coupling to plasmid DNA has also been realized by M.G.SebastyÉn and coworkers. Heterodimerization of TAT and NLS yields an even more effective transfecting peptide.

NuclearporecomplexproteinNup98(315-360)是核孔复合物(NPC)蛋白的315-360片段部分。

C3a Receptor Agonist是一种选择性的补体3a受体（C3aR）特异性激动剂。

A TGR5 agonist

Leptin Binding Domain Human Recombinant

Leptin Receptor Chicken Recombinant

Soluble RANK Receptor Human Recombinant

干扰素受体激动剂（化合物 6）是一种干扰素 (IFN) 受体诱导剂。

A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。

GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity.

The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor. MSRPACPNDKYE has served as model peptide in protein modification and MS studies.

A GCGR antagonist