Drug Metabolite(药物代谢物)

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Products for Drug Metabolite

Cat.No. 产品名称 Information
GC44912 Solifenacin N-Glucuronide A metabolite of solifenacin
GC44895 Sitagliptin N-Sulfate (sodium salt) A metabolite of (–)-sitagliptin
GC44890 Silodosin Glucuronide (sodium salt)
赛洛多辛β-D-葡萄糖苷酸钠盐

An active metabolite of silodosin
GC44820 Resveratrol-3-O-Sulfate (sodium salt) An active metabolite of resveratrol
GC44810 Reduced Haloperidol
还原氟哌啶醇
An active metobolite of haloperidol
GC44803 rac-7-hydroxy Propranolol (hydrochloride)
7-羟基普萘洛尔盐酸盐
An isomer and metabolite of propranolol
GC44799 Quinidine N-oxide A quinidine metabolite
GC44699 Propranolol β-D-Glucuronide (sodium salt) A major metabolite of propranolol
GC44676 Pravastatin lactone
普伐他汀类酯
A metabolite of pravastatin
GC44668 Posaconazole D-Glucuronide
Posaconazole N-β-D-Glucuronide
A metabolite of posaconazole
GC44665 PNU 142300
利奈唑胺杂质8
An inactive metabolite of linezolid
GC44650 Pitavastatin lactone
匹伐他汀内酯
A major phase 2 metabolite of pitavastatin
GC44628 Phenylephrine-3-O-Sulfate A metabolite of phenylephrine
GC44627 Phenylephrine Glucuronide
苯福林葡糖苷酸
A metabolite of phenylephrine
GC44599 Perindoprilat
培哚普利,S-9780
An active ACE inhibitor
GC44555 Pantoprazole sulfone
泮托拉唑杂质A
A pantoprazole metabolite
GC44554 Pantoprazole Sulfide
泮托拉唑硫醚
A pantoprazole metabolite
GC44527 p,p'-DDE
2，2-双（4-氯苯基）-1，1-二氯乙烯,4,4'-DDE; p,p'-Dichlorodiphenyldichloroethylene
A metabolite and degradation product of the pesticide DDT
GC44509 Omeprazole sulfide
奥美拉唑硫醚,Ufiprazole
An intermediate for omeprazole synthesis
GC44492 O-Desmethyl Metoprolol
O-去甲基美托洛尔
A major active metabolite of metoprolol
GC44451 Norfluoxetine (hydrochloride)
去甲氟西汀,Desmethylfluoxetine
Norfluoxetine (hydrochloride)是Fluoxetine在肝脏中通过N-去甲基化产生的活性代谢物，具有口服活性。
GC44358 Nebivolol O-β-D-Glucuronide An active metabolite of nebivolol
GC44351 N-Desmethyl Sildenafil (citrate) A major metabolite of sildenafil
GC44350 N-Desmethyl Sildenafil
N-去甲基西地那非,Desmethylsildenafil; UK-103,320
A major metabolite of sildenafil
GC44349 N-desmethyl Levofloxacin
左氧氟沙星相关物质A
An active metabolite of levofloxacin
GC44348 N-desmethyl Bendamustine
盐酸苯达莫司汀乙酯水解杂质
An active metabolite of bendamustine
GC44345 N-Desethyl Vardenafil
N-去乙基伐地那非
A vardenafil metabolite
GC44304 N-Acetyl-S-allyl-L-cysteine A primary metabolite of L-deoxyalliin
GC44299 N-Acetyl-4-benzoquinone imine
N-乙酰基-4-苯醌亚胺
A reactive CYP450 metabolite of acetaminophen
GC44294 N-acetyl Dapsone
N-乙酰氨苯砜
A metabolite of dapsone
GC44246 Moxifloxacin N-Sulfate (sodium salt) A metabolite of moxifloxacin
GC44033 Lansoprazole sulfone
兰索拉唑磺酸盐
A metabolite of lansoprazole
GC43896 Iloperidone metabolite P95
伊潘立酮代谢物P95
A metabolite of iloperidone
GC43895 Iloperidone metabolite P88
伊潘立酮代谢物; P88; Hydroxy Iloperidone
An active metabolite of iloperidone
GC43881 Hydroxy Varenicline
伐伦克林杂质
A metabolite of varenicline
GC43879 Hydroxy Ebastine An ebastine metabolite
GC43878 Hydroxy Dimetridazole
1-甲基-5-硝基-2-羟甲基咪唑,Hydroxy Dimetridazole
A metabolite of dimetridazole
GC43743 Gemfibrozil 1-O-β-Glucuronide
吉非罗齐酰基β-D-葡萄糖醛酸
A major metabolite of gemfibrozil
GC43697 Formoterol O-β-D-Glucuronide
福莫特罗杂质14
A metabolite of formoterol
GC43675 Florfenicol amine (hydrochloride)
氟苯尼考胺盐酸盐
A veterinary antibiotic metabolite
GC43646 Ezetimibe Hydroxy Glucuronide
依泽替米贝羟基-b-D-葡萄糖醛酸
A minor phase II metabolite of ezetimibe
GC43565 Doxorubicinol (hydrochloride)
13-Dihydroadriamycin hydrochloride
A doxorubicin metabolite
GC43493 DL-Sulforaphane N-acetyl-L-cysteine
SFNNAC
An anticancer agent
GC43444 Diclofenac Acyl-β-D-Glucuronide
双氯芬酸酰基-Β-D-葡糖苷酸
An active metabolite of diclofenac
GC43423 Desmethylene Paroxetine (hydrochloride)
帕罗西汀杂质5
A major metabolite of the SSRI paroxetine
GC43422 Desmethyldoxepin (hydrochloride)
N-去甲盐酸多塞平,Desmethyldoxepin hydrochloride
The primary metabolite of doxepin
GC43419 Desmethyl Erlotinib
2-[[4-[(3-乙炔基苯基)氨基]-7-(2-甲氧基乙氧基)-6-喹唑啉基]氧基]乙醇,OSI-420 free base; CP-373420
A metabolite of erlotinib
GC43418 Desethylene Ciprofloxacin (hydrochloride)
脱乙烯环丙沙星盐酸盐
A major metabolite and degradation product of ciprofloxacin
GC43412 Desacetyl Bisacodyl
苉可硫酸钠杂质B
An active metabolite of the laxatives bisacodyl and sodium picosulfate
GC43401 Dehydro Nifedipine
4-(2硝基苯基)-2,6-二甲基吡啶-3,5二羧酸二甲酯
An active metabolite of nifedipine