Other Apoptosis
Other Apoptosis(其他细胞凋亡)
Other Apoptosis 相关产品(883)
- GC13035Bay 11-7821CAS: 19542-67-7纯度: >99.50% / >95.00%
Bay 11-7821是一种IκBα磷酸化和NF-κB抑制剂,选择性且不可逆地抑制TNF-α诱导的IκB-α磷酸化(IC 50 值约为10μM),并减少NF-κB和粘附分子的表达。Bay 11-7821抑制泛素特异性蛋白酶USP7和USP21,IC 50 分别为0.19、0.96μM。
- GC1304417-DMAG (Alvespimycin) HClCAS: 467214-21-7纯度: >98.00%
17-DMAG (Alvespimycin) HCl是一种有效的Hsp90的抑制剂,其IC 50 值为62nM。
- GC13065Chelerythrine ChlorideCAS: 3895-92-9纯度: >98.50% / >98.00%
Chelerythrine Chloride是一种强效且可渗透细胞的蛋白激酶C(protein kinase C, PKC)抑制剂,IC 50 值为660nM。
- GC13232VerbascosideCAS: 61276-17-3纯度: >99.50%
Verbascoside是一种从Lantana camara中分离得到的蛋白激酶C(PKC)抑制剂,IC 50 值为25µM。
- GC13332Aurora A Inhibitor ICAS: 1158838-45-9纯度: >99.00%
A potent and selective inhibitor of Aurora A kinase
- GC13442Sanguinarine chlorideCAS: 5578-73-4纯度: >99.00%
A natural alkaloid with anti-inflammatory and anti-oxidant properties
- GC13484GriseofulvinCAS: 126-07-8纯度: >98.50%
A fungal metabolite with antifungal and anticancer activities
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13035 | Bay 11-7821 | 19542-67-7 | >99.50% / >95.00% | |
Bay 11-7821是一种IκBα磷酸化和NF-κB抑制剂,选择性且不可逆地抑制TNF-α诱导的IκB-α磷酸化(IC 50 值约为10μM),并减少NF-κB和粘附分子的表达。Bay 11-7821抑制泛素特异性蛋白酶USP7和USP21,IC 50 分别为0.19、0.96μM。 | ||||
| GC13044 | 17-DMAG (Alvespimycin) HCl | 467214-21-7 | >98.00% | |
17-DMAG (Alvespimycin) HCl是一种有效的Hsp90的抑制剂,其IC 50 值为62nM。 | ||||
| GC13055 | Mocetinostat (MGCD0103, MG0103) | 726169-73-9 | >99.00% | |
An orally available HDAC inhibitor | ||||
| GC13065 | Chelerythrine Chloride | 3895-92-9 | >98.50% / >98.00% | |
Chelerythrine Chloride是一种强效且可渗透细胞的蛋白激酶C(protein kinase C, PKC)抑制剂,IC 50 值为660nM。 | ||||
| GC13070 | Cytarabine | 147-94-4 | >99.50% | |
Cytarabine(Ara-C)是一种胞嘧啶类似物,主要抑制DNA聚合酶的功能来阻断DNA合成。 | ||||
| GC13091 | CP-724714 | 383432-38-0 | >99.00% | |
A selective HER2/ErbB2 tyrosine kinase inhibitor | ||||
| GC13168 | AG 825 | 149092-50-2 | >98.00% | |
An inhibitor of Her2/Neu tyrosine kinase activity | ||||
| GC13202 | D4476 | 301836-43-1 | >98.00% | |
Inhibitor of CK1 and ALK5 | ||||
| GC13210 | Flubendazole | 31430-15-6 | >99.50% | |
An anthelmintic | ||||
| GC13219 | ONO-4059 | 1351635-67-0 | >99.50% | |
A derivative of ONO-4059 | ||||
| GC13232 | Verbascoside | 61276-17-3 | >99.50% | |
Verbascoside是一种从Lantana camara中分离得到的蛋白激酶C(PKC)抑制剂,IC 50 值为25µM。 | ||||
| GC13246 | Ibandronate sodium | 138926-19-9 | >98.00% | |
A bisphosphonate bone resorption inhibitor | ||||
| GC13286 | ZM336372 | 208260-29-1 | - | |
An activator of the Raf-1 signalling pathway | ||||
| GC13332 | Aurora A Inhibitor I | 1158838-45-9 | >99.00% | |
A potent and selective inhibitor of Aurora A kinase | ||||
| GC13339 | Ketoprofen | 22071-15-4 | >99.50% | |
A non-selective COX inhibitor | ||||
| GC13359 | Topotecan HCl | 119413-54-6 | >99.00% | |
Topotecan HCl是一种毒药类的拓扑异构酶I抑制剂。 | ||||
| GC13383 | EPZ004777 | 1338466-77-5 | >98.00% | |
EPZ004777 作为一种有效的表观遗传调节剂,可以逆转 TGF-β1 诱导的 T 调节细胞,可用于治疗多种免疫疾病。 | ||||
| GC13394 | Ispinesib (SB-715992) | 336113-53-2 | >98.00% | |
An Eg5 inhibitor | ||||
| GC13408 | CI994 (Tacedinaline) | 112522-64-2 | >98.00% | |
An inhibitor of HDAC1, -2, and -3 | ||||
| GC13410 | Masitinib (AB1010) | 790299-79-5 | >99.50% | |
An inhibitor of c-Kit | ||||
| GC13433 | AZ 960 | 905586-69-8 | >98.00% | |
A JAK2 inhibitor | ||||
| GC13442 | Sanguinarine chloride | 5578-73-4 | >99.00% | |
A natural alkaloid with anti-inflammatory and anti-oxidant properties | ||||
| GC13474 | Garcinol | 78824-30-3 | >95.00% | |
Garcinol是组蛋白乙酰转移酶p300和PCAF的非特异性抑制剂,IC 50 分别为7μM和5μM。 | ||||
| GC13484 | Griseofulvin | 126-07-8 | >98.50% | |
A fungal metabolite with antifungal and anticancer activities | ||||
