关于 "Reverse Transcriptase" 的结果28+ 个结果
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- TirucallolCAS: 514-46-5
A triterpenoid with reverse transcriptase inhibitory and anti-inflammatory activities
Others - Ro 26-4550 trifluoroacetateCAS: 1217448-66-2
reversible inhibitor of interleukin-2 (IL-2) binding to its receptor
- Cruzain-IN-1CAS: 1199523-24-4
Cruzain-IN-1 is a selective inhibitor of trypanosomal cysteine proteases and a covalent and reversible Cruzain inhibitor with IC50 of 10 nM.
Others - Anhydrotetracycline (hydrochloride)CAS: 13803-65-1
Anhydrotetracycline (hydrochloride)是一种四环素生物合成前体,是竞争性四环素破坏酶广谱抑制剂。Anhydrotetracycline (hydrochloride)是真核细胞中四环素阻遏蛋白(TetR)和反向四环素阻遏蛋白(revTetR)转录抑制因子的调节因子。
- Golgicide ACAS: 1139889-93-2
Golgicide A是一种高度特异且可逆的顺式高尔基体ADP-核糖基化因子鸟嘌呤核苷酸交换因子(ArfGEF GBF1)抑制剂,Golgicide A通过选择性靶向GBF1并减少Arf1的活化,从而阻断细胞内的囊泡运输和蛋白质分泌。
Others
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC63228 | Tirucallol | 514-46-5 | Others | ||
A triterpenoid with reverse transcriptase inhibitory and anti-inflammatory activities | |||||
| GC11274 | Abacavir sulfate | 188062-50-2 | Reverse Transcriptase | ||
An antiviral nucleoside analog | |||||
| GC19510 | Alovudine | 25526-93-6 | Others | ||
A nucleoside analog | |||||
| GC14697 | HA 130 | 1229652-21-4 | PDE | ||
A reversible autotaxin inhibitor | |||||
| GC17921 | Tolcapone | 134308-13-7 | Amyloid β | ||
A reversible COMT inhibitor | |||||
| GC15751 | Exo1 | 461681-88-9;75541-83-2 | Others | ||
A reversible inhibitor of exocytosis | |||||
| GC41267 | β-cyano-L-Alanine | 6232-19-5 | Others | ||
A reversible inhibitor of H2S synthesis | |||||
| GC19340 | Sugammadex sodium | 343306-79-6 | Others | ||
A steroid-based neuromuscular blocker reversing agent | |||||
| GC14469 | Pirlindole mesylate | 207572-66-5 | Heme oxygenase | ||
A selective and reversible MAO-A inhibitor | |||||
| GC67613 | Sugammadex | 343306-71-8 | Others | ||
A steroid-based neuromuscular blocker reversing agent | |||||
| GC13566 | NVP 231 | 362003-83-6 | Others | ||
A potent and reversible inhibitor of ceramide kinase | |||||
| GC12565 | Ro 26-4550 trifluoroacetate | 1217448-66-2 | Cytokine | ||
reversible inhibitor of interleukin-2 (IL-2) binding to its receptor | |||||
| GC18091 | Entacapone sodium salt | 1047659-02-8 | COMT | ||
A reversible COMT inhibitor | |||||
| GC12361 | Darapladib | 356057-34-6 | Phospholipase | ||
A reversible inhibitor of Lp-PLA2 | |||||
| GC30348 | Cruzain-IN-1 | 1199523-24-4 | Others | ||
Cruzain-IN-1 is a selective inhibitor of trypanosomal cysteine proteases and a covalent and reversible Cruzain inhibitor with IC50 of 10 nM. | |||||
| GC25581 | LM11A-31 | 289475-77-0 | Others | ||
LM11A-31 is a small molecule p75NTR Ligand that reverses cholinergic neurite dystrophy in alzheimer's diseasemousemodels with mid- to late-stage disease progression | |||||
| GC63794 | ARN19702 | 1971937-18-4 | Others | ||
ARN19702 is an orally active, reversible N-Acylethanolamine acid amidase(NAAA) inhibitor (IC50 on human NAAA = 230 nM) that produces remarkable protective effects against multiple sclerosis in mice. | |||||
| GC63192 | Simufilam | 1224591-33-6 | Others | ||
Simufilam(PTI-125) is potent, orally active small drug against AD, which interacts to filamin and controls the actin cytoskeleton. Simufilam reduces tau hyperphosphorylation, amyloid and tau formation by preventing and reversing the binding of Aβ42 to α7nAChR. | |||||
| GC16227 | Anhydrotetracycline (hydrochloride) | 13803-65-1 | Transcription Factors | ||
Anhydrotetracycline (hydrochloride)是一种四环素生物合成前体,是竞争性四环素破坏酶广谱抑制剂。Anhydrotetracycline (hydrochloride)是真核细胞中四环素阻遏蛋白(TetR)和反向四环素阻遏蛋白(revTetR)转录抑制因子的调节因子。 | |||||
| GC15671 | Latrunculin A | 76343-93-6 | Arp2/3 Complex | ||
一种可逆抑制肌动蛋白聚合的药物 | |||||
| GC50284 | JZP 361 | 1680193-80-9 | Others | ||
JZP 361 是一种有效、可逆和选择性的人重组 MAGL (hMAGL) 抑制剂,IC50 为 46 nM。 | |||||
| GC16585 | Golgicide A | 1139889-93-2 | Others | ||
Golgicide A是一种高度特异且可逆的顺式高尔基体ADP-核糖基化因子鸟嘌呤核苷酸交换因子(ArfGEF GBF1)抑制剂,Golgicide A通过选择性靶向GBF1并减少Arf1的活化,从而阻断细胞内的囊泡运输和蛋白质分泌。 | |||||
| GC15820 | GSK837149A | 13616-29-0 | Synthases/Synthetases | ||
A selective FASN inhibitor | |||||
| GC50341 | T 3364366 | 1356354-09-0 | Others | ||
T 3364366 是一种可逆的、缓慢结合的噻吩并嘧啶酮 delta-5 去饱和酶 (D5D) 抑制剂,在 HepG2 和 RLN-10 细胞中的 IC50 分别为 1.9 nM 和 2.1 nM。 | |||||
