Calcium Channel
Calcium Channel(钙离子通道)
Calcium channel is an ion channel that selectively permeable to calcium ions. It serves vital functions in cellular signal transduction.
Calcium Channel 相关产品(321)
- GC33458Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione)CAS: 127-48-0纯度: >98.00%
An anticonvulsant
- GC33486DehydronitrosonisoldipineCAS: 87375-91-5纯度: >98.00% / >99.50%
Dehydronitrosonisoldipine是尼索地平（Nisoldipine）的衍生物，在保留钙离子通道拮抗活性的同时，还具备抑制无菌α和TIR基序蛋白1（SARM1）的功能，因而成为一种双重生物活性化合物。
- GC34049Aranidipine (MPC1304)CAS: 86780-90-7纯度: >99.00%
Aranidipine (MPC1304) (MPC1304) 是一种 Ca2+ 通道拮抗剂，具有强效和持久的抗高血压作用。
- GC34912Levamlodipine besylateCAS: 150566-71-5纯度: >99.50%
Levamlodipine Besylate is a powerful dihydropyridine calcium channel blocker, possessing vasodilation properties and used in the treatment of hypertension and angina.
- GC35325Amlodipine maleateCAS: 88150-47-4纯度: >99.50%
Amlodipine (Amvaz, UK-48340) maleate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
- GC35619Cav 2.2 blocker 1CAS: 1567335-29-8纯度: >99.00%
Cav 2.2 blocker 1 (compound 9) is a N-type calcium channel (Cav 2.2) blocker for the treatment of pain with IC50 of 0.001 μM.
- GC35963Efonidipine hydrochloride monoethanolateCAS: 111011-76-8纯度: >99.00%
An L- and T-type calcium channel inhibitor
- GC36097Gabapentin enacarbilCAS: 478296-72-9纯度: >98.00%
Gabapentin enacarbil (XP-13512)是gabapentin的原药。
- GC36105GallopamilCAS: 16662-47-8纯度: >98.00%
Gallopamil (Methoxyverapamil) 是一种维拉帕米的甲氧基衍生物 (methoxy derivative of verapamil)，也是一种苯基烷基胺钙 (phenylalkylamine calcium)拮抗剂。Gallopamil 可以作用于血管系统，心脏及其淋巴结构。Gallopamil 以浓度依赖性方式抑制酸分泌，IC50 为 10.9 μM.
- GC36371JTV-519 free baseCAS: 145903-06-6
JTV-519 free base (K201 free base) 是 Ca2+ 依赖性的肌质网 Ca2+ 刺激的 ATP 酶 (SERCA) 阻断剂。JTV-519 free base (K201 free base) 也是横纹肌中兰尼碱受体 (ryanodine receptors) 的部分激动剂。JTV-519 free base (K201 free base) 是一种心脏保护剂。
- GC36955Praeruptorin ECAS: 78478-28-1
Praeruptorin E, isolated from Peucedanum praeruptorum Dunn., is a cardiotonic agent with selective cardiac calcium channel agonistic effect.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC32672 | AE0047 Hydrochloride | 116308-56-6 | - | |
AE0047Hydrochloride是一种calcium阻滞剂，可用于高血压症的研究。 | ||||
| GC33176 | Teludipine hydrochloride (GR53992B) | 108700-03-4 | - | |
特鲁地平是一种亲脂性钙通道阻滞剂。 | ||||
| GC33458 | Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) | 127-48-0 | >98.00% | |
An anticonvulsant | ||||
| GC33486 | Dehydronitrosonisoldipine | 87375-91-5 | >98.00% / >99.50% | |
Dehydronitrosonisoldipine是尼索地平（Nisoldipine）的衍生物，在保留钙离子通道拮抗活性的同时，还具备抑制无菌α和TIR基序蛋白1（SARM1）的功能，因而成为一种双重生物活性化合物。 | ||||
| GC33695 | Ethosuximide | 77-67-8 | >99.00% | |
An anticonvulsant | ||||
| GC33720 | ABT-639 hydrochloride | 1235560-31-2 | - | |
A T-type calcium channel blocker | ||||
| GC33732 | Syntide 2 | 108334-68-5 | - | |
A protein kinase substrate | ||||
| GC34049 | Aranidipine (MPC1304) | 86780-90-7 | >99.00% | |
Aranidipine (MPC1304) (MPC1304) 是一种 Ca2+ 通道拮抗剂，具有强效和持久的抗高血压作用。 | ||||
| GC34912 | Levamlodipine besylate | 150566-71-5 | >99.50% | |
Levamlodipine Besylate is a powerful dihydropyridine calcium channel blocker, possessing vasodilation properties and used in the treatment of hypertension and angina. | ||||
| GC35325 | Amlodipine maleate | 88150-47-4 | >99.50% | |
Amlodipine (Amvaz, UK-48340) maleate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain. | ||||
| GC35451 | Azelnidipine D7 | - | - | |
Azelnidipine D7是Azelnidipine氘代化合物标准品。 | ||||
| GC35469 | Barnidipine | 104713-75-9 | - | |
A calcium channel blocker | ||||
| GC35619 | Cav 2.2 blocker 1 | 1567335-29-8 | >99.00% | |
Cav 2.2 blocker 1 (compound 9) is a N-type calcium channel (Cav 2.2) blocker for the treatment of pain with IC50 of 0.001 μM. | ||||
| GC35738 | CP-060 | 180090-15-7 | - | |
CP-?060 是一种 Ca2+ 拮抗剂，能够抑制 Ca2+ 过载，具有抗氧化、保护心脏的作用。 | ||||
| GC35963 | Efonidipine hydrochloride monoethanolate | 111011-76-8 | >99.00% | |
An L- and T-type calcium channel inhibitor | ||||
| GC36097 | Gabapentin enacarbil | 478296-72-9 | >98.00% | |
Gabapentin enacarbil (XP-13512)是gabapentin的原药。 | ||||
| GC36105 | Gallopamil | 16662-47-8 | >98.00% | |
Gallopamil (Methoxyverapamil) 是一种维拉帕米的甲氧基衍生物 (methoxy derivative of verapamil)，也是一种苯基烷基胺钙 (phenylalkylamine calcium)拮抗剂。Gallopamil 可以作用于血管系统，心脏及其淋巴结构。Gallopamil 以浓度依赖性方式抑制酸分泌，IC50 为 10.9 μM. | ||||
| GC36178 | Gomisin J | 66280-25-9 | >99.00% | |
A lignan with diverse biological activities | ||||
| GC36371 | JTV-519 free base | 145903-06-6 | - | |
JTV-519 free base (K201 free base) 是 Ca2+ 依赖性的肌质网 Ca2+ 刺激的 ATP 酶 (SERCA) 阻断剂。JTV-519 free base (K201 free base) 也是横纹肌中兰尼碱受体 (ryanodine receptors) 的部分激动剂。JTV-519 free base (K201 free base) 是一种心脏保护剂。 | ||||
| GC36713 | Ned 19 | 874374-25-1 | - | |
Ned 19 是一种选择性膜透性非竞争性 NAADP 拮抗剂，抑制 NAADP 介导的 Ca2+ 信号传导，IC50 为 65 nM。 Ned 19 强烈抑制小鼠的肿瘤生长和血管形成以及肺转移。 | ||||
| GC36766 | NP118809 | 41332-24-5 | >98.50% | |
NP118809 是一种有效的 N 型钙通道 (N-type calcium channel) 阻滞剂，IC50 值为 0.11 μM；同时可较弱地抑制 L 型钙通道 (L-type calcium channel)，IC50 值为 12.2 μM。 | ||||
| GC36843 | Palonidipine | 96515-73-0 | - | |
Palonidipine 是一种钙拮抗剂，有治疗心绞痛和高血压的潜力。 | ||||
| GC36955 | Praeruptorin E | 78478-28-1 | - | |
Praeruptorin E, isolated from Peucedanum praeruptorum Dunn., is a cardiotonic agent with selective cardiac calcium channel agonistic effect. | ||||
| GC37710 | Syntide 2 (TFA) | - | >99.50% | |
A protein kinase substrate | ||||