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ATPase(ATP酶)

ATPase is a class of enzymes that catalyze the decomposition of ATP into ADP and a free phosphate ion, including some co-transporters and pumps.

Products for  ATPase

  1. Cat.No. 产品名称 Information
  2. GC16859 Oligomycin A

    寡霉素A; MCH 32

    Oligomycin A 是一种 ATP 合酶抑制剂,可抑制线粒体偶联膜上依赖 ATP 和氧化磷酸化的过程。
  3. GC16409 Oligomycin B

    寡霉素 B

    A nonselective inhibitor of the mitochondrial F1FO ATP synthase
  4. GC16221 Oligomycin C

    寡霉素C

    A mitochondrial F1FO ATP synthase inhibitor
  5. GC16533 Oligomycin Complex

    寡霉素

    寡霉素复合物(Oligomycin complex)由寡霉素A、B和C的混合物组成。
  6. GC12832 Omecamtiv mecarbil

    4-[[2-氟-3-[N'-(6-甲基吡啶-3-基)脲基]苯基]甲基]哌嗪-1-羧酸甲酯,CK-1827452; CK1827452

    A cardiac-specific myosin activator
  7. GC47826 Omeprazole sulfone-d3

    OMEP sulfone-d3, OMP sulfone-d3, OMZ sulfone-d3

    An internal standard for the quantification of omeprazole sulfone
  8. GC49663 Pantoprazole sulfone N-oxide

    泮托拉唑砜N-氧化物

    A potential impurity found in bulk preparations of pantoprazole
  9. GC45539 Pantoprazole-d6

    BY1023-d6; SKF96022-d6

    An internal standard for the quantification of pantoprazole
  10. GC12788 Paprotrain

    (ALPHAZ)-ALPHA-(3-吡啶基亚甲基)-1H-吲哚-3-乙腈

    A MKLP-2 inhibitor
  11. GC45944 para-amino-Blebbistatin

    (-)-4'-amino-Blebbistatin, p-amino-Blebbistatin, (S)-4'-amino-Blebbistatin

    A more stable and less phototoxic form of (–)-blebbistatin with enhanced water solubility
  12. GC11082 Paxilline

    蕈青霉素

    Paxilline是一种致震颤真菌生物碱,可有效抑制高电导Ca2+ 激活K+ (BK)通道,IC50约为10nM,Ki=1.9nM。
  13. GC10444 PF-03716556

    PF-03716556; PF03716556

    A potent and selective H+/K+-ATPase inhibitor
  14. GC17027 POM 1

    聚钨酸钠,Sodium polyoxotungstate; POM-1

    POM 1是一种核苷三磷酸二磷酸水解酶(NTPDase)抑制剂,对NTPDase1(CD39)、NTPDase3和NTPDase2的Ki值分别为2.58μM、3.26μM和28.8μM。
  15. GC10371 PSB 06126 PSB 06126 是一种选择性三磷酸核苷二磷酸水解酶 (NTPDase) 抑制剂,对大鼠 NTPDase 1 的 Ki 值分别为 0.33 μM,对 NTPDase 2 和 NTPDase 3 的 Ki 值分别为 19.1 μM 和 2.22 μM。
  16. GC13186 PSB 069 带有对氯苯氨基残基的 PSB 069 是一种有效的、耐受性良好且非选择性的 NTPDases1, 2, 3 抑制剂(Ki\u003d16~18 μM)。
  17. GC49627 Rabeprazole sulfone

    雷贝拉唑杂质E

    A metabolite of rabeprazole
  18. GC10906 RBC8 A Ral inhibitor
  19. GC11151 SCH 28080 An inhibitor of H+/K+-ATPases
  20. GC14368 Sodium Orthovanadate

    钒酸钠

    A protein tyrosine phosphatase inhibitor
  21. GC60348 Supinoxin

    RX-5902

    Supinoxin (RX-5902) 是磷酸化 p68 RNA 解旋酶 (P-p68) 的强效口服活性抑制剂,并且是一个一流的抗肿瘤试剂 (anti-cancer agent)。Supinoxin 与 Y593 磷酸化的 p68 相互作用并减弱 β-catenin 的核穿梭性。 Supinoxin 诱导细胞凋亡 (apoptosis) 并抑制 TNBC 癌细胞系的生长,IC50 的范围为 10 nM 至 20 nM。
  22. GC15418 TAK-438

    富马酸沃诺拉赞

    A selective and reversible proton pump inhibitor
  23. GC18005 Tenatoprazole

    泰妥拉唑,TU-199

    A proton pump inhibitor
  24. GC25991 Tetrathiomolybdate Tetrathiomolybdate (TM) is used in the clinic for the treatment of Wilson's disease by inducing dimerization of the metal-binding domain of the cellular copper efflux protein ATP7B (WLN4) through a unique sulfur-bridged Mo2S6O2 cluster.
  25. GC11482 Thapsigargin

    毒胡萝卜素

    他普西加林是一种肌浆网/内质网Ca2+ ATP酶泵的抑制剂。
  26. GC49503 Thujopsene

    罗汉柏烯

    A sesquiterpene with diverse biological activities
  27. GC72771 Triciribine phosphate sodium

    TCN-P sodium

    Triciribine phosphate sodium通过变构机制抑制氨基磷酸核糖基转移酶,影响从头嘌呤生物合成的第一步。
  28. GC61374 Vonoprazan Fumarate

    富马酸沃诺拉赞; TAK-438

    A selective and reversible proton pump inhibitor
  29. GC49430 Wee1 Inhibitor An inhibitor of Wee1

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