Opioid Receptor
Opioid Receptor(阿片受体)
Opioid receptor is a group of G protein-coupled receptors with opioids as ligands.
Opioid Receptor 相关产品(145)
- GC12534ICI 199,441 hydrochlorideCAS: 115199-84-3纯度: >97.00%
ICI 199,441 hydrochloride 是一种有效的选择性 κ-阿片受体激动剂。
- GC13645nor-Binaltorphimine dihydrochlorideCAS: 113158-34-2纯度: >98.00%
nor-Binaltorphimine dihydrochloride是一种有效的选择性κ阿片受体(KOR)拮抗剂。
- GC16588Naloxonazine dihydrochlorideCAS: 880759-65-9
Naloxonazine dihydrochloride 是一种特异性的 μ-阿片受体拮抗剂,IC50 为 5.4 nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC12143 | Deltorphin I | 122752-15-2 | - | |
Deltorphin I 是一种 δ-阿片受体激动剂,具有高亲和力和选择性。 | ||||
| GC12534 | ICI 199,441 hydrochloride | 115199-84-3 | >97.00% | |
ICI 199,441 hydrochloride 是一种有效的选择性 κ-阿片受体激动剂。 | ||||
| GC12663 | N-Benzylnaltrindole hydrochloride | 1206487-81-1 | - | |
δ2 opioid receptor antagonist | ||||
| GC12688 | (+)-U-50488 hydrochloride | 114528-81-3 | - | |
An Analytical Reference Material | ||||
| GC13097 | ICI 204,448 hydrochloride | 121264-04-8 | - | |
κ opioid receptor agonist | ||||
| GC13189 | Cyprodime hydrochloride | 118111-54-9 | - | |
μ-opioid receptor antagonist | ||||
| GC13546 | Dynorphin A | 80448-90-4 | >98.50% | |
Dynorphin A是一种内源性阿片肽,可激活孤儿受体XOR1-K + 通道,EC 50 值为45nM。 | ||||
| GC13581 | SB 205607 dihydrobromide | 148545-09-9 | - | |
non-peptide δ1 opioid receptor agonist | ||||
| GC13645 | nor-Binaltorphimine dihydrochloride | 113158-34-2 | >98.00% | |
nor-Binaltorphimine dihydrochloride是一种有效的选择性κ阿片受体(KOR)拮抗剂。 | ||||
| GC13688 | Naltrindole hydrochloride | 111469-81-9 | - | |
A potent, selective δ-opioid receptor antagonist | ||||
| GC13910 | Salvinorin A | 83729-01-5 | >95.00% | |
An Analytical Reference Material | ||||
| GC14525 | ML 190 | 1355244-02-8 | - | |
ML 190 是一种选择性 κ 阿片受体 (KOR) 拮抗剂,IC50 分别为 120 nM 和 EC50 分别为 129 nM 。 | ||||
| GC14739 | GR 89696 fumarate | 126766-32-3 | - | |
κ-opioid agonist | ||||
| GC14774 | DSLET | 75644-90-5 | - | |
δ Opioid receptor agonist | ||||
| GC14979 | N-MPPP Hydrochloride | 207452-97-9 | - | |
High affinity κ agonist | ||||
| GC15078 | Dynorphin B | 83335-41-5 | - | |
An endogenous κ 1b -opioid receptor agonist | ||||
| GC15313 | BRL 52537 hydrochloride | 112282-24-3 | - | |
κ/μ opioid receptor agonist,potent and selective | ||||
| GC15843 | GNTI dihydrochloride | 351183-88-5 | - | |
κ opioid receptor antagonist | ||||
| GC15874 | FIT | 85951-63-9 | - | |
δ-opioid agonist, irreversible | ||||
| GC15938 | β-Funaltrexamine hydrochloride | 72786-10-8 | >95.00% | |
μ opioid receptor antagonist | ||||
| GC16193 | ICI 174,864 | 89352-67-0 | - | |
Selective δ opioid antagonist | ||||
| GC16521 | BW 373U86 | 155836-50-3 | >99.00% | |
BW 373U86 (SNC86) 是一种 δ-阿片受体激动剂,IC50 为 1.49 nM。 | ||||
| GC16588 | Naloxonazine dihydrochloride | 880759-65-9 | - | |
Naloxonazine dihydrochloride 是一种特异性的 μ-阿片受体拮抗剂,IC50 为 5.4 nM。 | ||||
| GC17553 | DIPPA hydrochloride | 155512-52-0 | - | |
DIPPA(盐酸盐)是一种不可逆、长效、选择性和高亲和力的 κ-阿片受体拮抗剂。 | ||||
