Estrogen/progestogen Receptor(雌激素/孕激素受体)

Cat.No. 产品名称 Information

GC47554 Letrozole-d4

来曲唑 d4

An internal standard for the quantification of letrozole

GC14704 Levonorgestrel

左炔诺孕酮; D-Norgestrel

Levonorgestrel是一种口服有效的孕酮抑制剂。

GC61971 Liarozole

利阿唑,R75251

A CYP26A1 inhibitor

GC11781 Medroxyprogesterone

甲羟孕酮; 17α-Hydroxy-6α-methylprogesterone; U8840

A progesterone receptor agonist

GC12974 Medroxyprogesterone acetate

醋酸甲羟孕酮; Medroxyprogesterone 17-acetate; Farlutin

Medroxyprogesterone acetate（MPA）是一种人工合成的孕激素。

GC11688 Megestrol Acetate

醋酸甲地孕酮

A synthetic progestogen

GC62061 Melengestrol acetate

醋酸美伦孕酮

A synthetic progestogen

GC25627 Menotropin

Human Menopausal Gonadotrophin

Menotropin (Human Menopausal Gonadotrophin) is a hormonally active medication for the treatment of fertility disturbances, which are extracted from the urine of postmenopausal women.

GC17161 Methylpiperidino pyrazole

MPP

Methylpiperidino pyrazole是一种对雌激素受体α（Erα）具有高度选择性的拮抗剂，其半数抑制浓度（IC₅₀）为20.01nM。

GC47674 Mifepristone-d3

RU486-d3; RU 38486-d3

A neuropeptide with diverse biological activities

GC11881 MPP dihydrochloride

MPP二盐酸盐

MPP dihydrochloride是一种选择性雌激素受体α（ERα）拮抗剂。

GC47747 Napyradiomycin A1 A fungal metabolite with diverse biological activities

GC17200 Nestoron

醋酸烯诺孕酮; ST-1435; Elcometrine

A synthetic progestin

GC52189 Nomegestrol

诺美孕酮

A derivative of 19-norprogesterone

GC48788 Norethindrone-d6

炔诺酮D6,Norethisterone-d6

An internal standard for the quantification of norethindrone

GC48803 Norethynodrel

异炔诺酮,Enidrel; SC 4642; NSC 15432

A synthetic progestin

GC47797 Norgestimate-d6

炔诺肟酯-D6

An internal standard for the quantification of norgestimate

GC45530 Norgestrel-d6

左炔诺孕酮 d6

An internal standard for the quantification of norgestrel

GC44479 o,p'-DDE

3-邻氯苯基-2-对氯苯-1,1'-二乙烯

A metabolite and degradation product of the pesticide DDT

GC16719 Ormeloxifene

苯并吡喃,Centchroman

estrogen receptor modulator

GC11996 Ospemifene

奥培米芬; FC-1271a

A selective estrogen receptor modulator

GC44528 p,p'-DDT

4,4'-DDT, 4,4'-Dichlorodiphenyltrichloroethane, p,p'-Dichlorodiphenyltrichloroethane, Dicophaner, NSC 8939

p,p'-DDT is an organochlorine pesticide that induces 94.2% mortality of malaria mosquito (A.

GC91296 p-Carboxyphenyl Sulfate

Benzoic Acid-4-sulfate, 4-Carboxyphenyl Sulfate, para-Carboxyphenyl Sulfate, 4-Hydroxybenzoic Acid Sulfate, p-Hydroxybenzoic Acid Sulfate, para-Hydroxybenzoic Acid Sulfate

一种硫酸化的酚酸。

GC11863 PHTPP PHTPP是一种选择性ERβ完全拮抗剂，对ERβ的选择性是ERα的36倍。PHTPP可以选择性拮抗ERβ的配体结合和转录功能，阻断其对肿瘤细胞的抑制作用，从而促进细胞增殖。PHTPP被用于验证ERβ的功能。

GC41266 Pregnanediol-3-Glucuronide

Pregnanediol-3α-Glucuronide

A metabolite of progesterone

GC48724 Pregnanetriol

孕三醇

A metabolite of 17α-hydroxyprogesterone

GC47973 PRGL493 An ACSL4 inhibitor

GC12408 Progesterone

孕酮; Pregn-4-ene-3,20-dione

An endogenous hormone and hormone precursor

GC44691 Progesterone 3-biotin An affinity probe

GC44692 Progesterone 3-PEG11-biotin A hydrophilic affinity probe

GC44693 Progesterone-3-biotinyl Photoaffinity Probe

P4, P4 Binding Probe

A photoaffinity probe

GC47976 Progesterone-d9

氘代黄体酮/氘代4-烯-3,20-二酮,Pregn-4-ene-3,20-dione-d9

An internal standard for the quantification of progesterone

GC47979 Propiconazole-d7 An internal standard for the quantification of propiconazole

GC14370 Propyl pyrazole triol (PPT)

PPT

Propyl pyrazole triol (PPT)是一种选择性雌激素受体α（ERα）激动剂，可通过在神经系统激活ERα，保护神经元免受氧化应激与炎症损伤。

GC12644 Quinestrol

炔雌醇环戊醚,Estrovis?,Ethynyl Estradiol-3-cyclopentyl ether,W 3566

A synthetic estrogen

GC25832 Raloxifene

Keoxifene, Pharoxifene, LY-139481, LY-156758, CCRIS-7129

Raloxifene (Keoxifene, Pharoxifene, LY-139481, LY-156758, CCRIS-7129) is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women.

GC13350 Raloxifene HCl

盐酸雷洛昔芬; Keoxifene hydrochloride; LY156758; LY139481 hydrochloride

A selective estrogen receptor modulator

GC48023 Raloxifene-d4 (hydrochloride)

雷洛昔芬-D4,盐酸盐

An internal standard for the quantification of raloxifene

GC17856 RU 58668 Pure antiestrogen that downregulates estrogen receptor expression

GC61267 SAR439859

SAR439859

Amcenestrant (SAR439859, compound 43d) is an orally available and nonsteroidal selective estrogen receptor degrader (SERD) with potential antineoplastic activity. SAR439859 is a potent estrogen receptor (ER) antagonist with EC50 of 0.2 nM for ERα degradation.