Dopamine Receptor
Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Dopamine Receptor 相关产品(289)
- GC11810PG 01037 dihydrochlorideCAS: 675599-62-9纯度: >99.50%
A selective dopamine D 3 receptor antagonist
- GC12179GBR 13069 dihydrochlorideCAS: 67469-45-8
GBR 13069 dihydrochloride是一种具有选择性的多巴胺摄取抑制剂（IC 50 =40~51nM）。
- GC12428Ro 10-5824 dihydrochlorideCAS: 189744-94-3纯度: >99.50%
Ro 10-5824 dihydrochloride 是一种选择性多巴胺 D4 受体部分激动剂，Ki 为 5.2 nM。
- GC12456GBR 12783 dihydrochlorideCAS: 67469-75-4纯度: >98.00%
GBR 12783 dihydrochloride 是一种特异性、有效和选择性的多巴胺摄取抑制剂，抑制大鼠和小鼠纹状体突触体对 [3H] 多巴胺的摄取，IC50 分别为 1.8 nM 和 1.2 nM。
- GC12986RisperidoneCAS: 106266-06-2纯度: >98.00%
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂，对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。
- GC13031Trifluoperazine 2HClCAS: 440-17-5纯度: >99.00% / >98.00%
An anti-adrenergic and anti-dopaminergic agent
- GC13036L-741,742 hydrochlorideCAS: 874882-93-6
highly potent and selective D4 dopamine receptor antagonist
- GC13109FananserinCAS: 127625-29-0纯度: >99.50%
Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11521 | Ziprasidone HCl | 122883-93-6 | - | |
An atypical antipsychotic | ||||
| GC11602 | Piribedil dihydrochloride | 1451048-94-4 | - | |
A dopamine receptor agonist | ||||
| GC11795 | ABT 724 trihydrochloride | 587870-77-7 | >99.00% | |
A dopamine D 4 receptor agonist | ||||
| GC11810 | PG 01037 dihydrochloride | 675599-62-9 | >99.50% | |
A selective dopamine D 3 receptor antagonist | ||||
| GC11902 | PNU 96415E | 170856-41-4 | - | |
PNU 96415E 是一种选择性 D4/5-HT2A 拮抗剂。 | ||||
| GC11945 | BTCP maleate | 207455-25-2 | - | |
dopamine reuptake inhibitor | ||||
| GC11977 | Thioridazine HCl | 130-61-0 | >99.50% | |
A typical antipsychotic | ||||
| GC12015 | Sonepiprazole | 170858-33-0 | - | |
A selective D 4 receptor antagonist | ||||
| GC12158 | SKF 81297 hydrobromide | 67287-39-2 | - | |
A selective dopamine D 1 -like receptor agonist | ||||
| GC12179 | GBR 13069 dihydrochloride | 67469-45-8 | - | |
GBR 13069 dihydrochloride是一种具有选择性的多巴胺摄取抑制剂（IC 50 =40~51nM）。 | ||||
| GC12293 | Perphenazine | 58-39-9 | >99.50% | |
A typical antipsychotic | ||||
| GC12355 | Eticlopride hydrochloride | 97612-24-3 | - | |
A dopamine D 2 and D 3 receptor antagonist | ||||
| GC12428 | Ro 10-5824 dihydrochloride | 189744-94-3 | >99.50% | |
Ro 10-5824 dihydrochloride 是一种选择性多巴胺 D4 受体部分激动剂，Ki 为 5.2 nM。 | ||||
| GC12456 | GBR 12783 dihydrochloride | 67469-75-4 | >98.00% | |
GBR 12783 dihydrochloride 是一种特异性、有效和选择性的多巴胺摄取抑制剂，抑制大鼠和小鼠纹状体突触体对 [3H] 多巴胺的摄取，IC50 分别为 1.8 nM 和 1.2 nM。 | ||||
| GC12466 | FAUC-365 | 474432-66-1 | - | |
A dopamine D 3 receptor antagonist | ||||
| GC12495 | Olanzapine | 132539-06-1 | >99.00% / >98.00% / >99.50% | |
Olanzapine是一种单胺拮抗剂。 | ||||
| GC12543 | Nemonapride | 75272-39-8 | - | |
An antipsychotic | ||||
| GC12641 | 3-CPMT | 14008-79-8 | >99.00% | |
dopamine uptake inhibitor | ||||
| GC12800 | PAOPA | 114200-31-6 | - | |
dopamine D2 receptor modulator | ||||
| GC12870 | (+)-UH 232 maleate | 95999-12-5 | - | |
D2 antagonist | ||||
| GC12986 | Risperidone | 106266-06-2 | >98.00% | |
Risperidone是一种5-羟色胺5-HT₂受体阻断剂、P-糖蛋白抑制剂和强效多巴胺D₂受体拮抗剂，对5-HT₂A和多巴胺D₂受体的Ki值分别为4.8nM和5.9nM。 | ||||
| GC13031 | Trifluoperazine 2HCl | 440-17-5 | >99.00% / >98.00% | |
An anti-adrenergic and anti-dopaminergic agent | ||||
| GC13036 | L-741,742 hydrochloride | 874882-93-6 | - | |
highly potent and selective D4 dopamine receptor antagonist | ||||
| GC13109 | Fananserin | 127625-29-0 | >99.50% | |
Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂，对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。 | ||||