Dopamine Receptor
Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Dopamine Receptor 相关产品(289)
- GC13156(+)-AJ 76 hydrochlorideCAS: 85379-09-5
(+)-AJ 76 hydrochloride是一种对突触前受体具有优先作用的多巴胺受体(dopamine receptors, DRs)拮抗剂(hD3、hD4、hD2S、hD2L和rD2受体的pKi值分别为6.95、6.67、6.37、6.21和6.07)。
- GC13786(±)-Salsolinol (hydrochloride)CAS: 79923-51-6纯度: >98.00%
A metabolite of ethanol that targets dopaminergic neurons
- GC14280PD 168568 dihydrochlorideCAS: 210688-56-5
PD 168568 dihydrochloride 是一种具有口服活性的选择性 D4 多巴胺受体拮抗剂,Ki 为 8.8 nM。
- GC143114-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochlorideCAS: 6109-35-9
dopamine release inhibitor
- GC14518Asenapine hydrochlorideCAS: 1412458-61-7纯度: >99.50%
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。
- GC14559Fluphenazine dihydrochlorideCAS: 146-56-5纯度: >99.00%
A dopamine D 1 and D 2 receptor antagonist
- GC14569L-745,870 trihydrochlorideCAS: 866021-03-6纯度: >98.00%
L-745,870 trihydrochloride 是一种有效的、选择性的、脑渗透性和口服活性的多巴胺 D4 受体拮抗剂,Ki 为 0.43 nM。
- GC14593GSK 789472 hydrochlorideCAS: 1257326-24-1
dopamine D3 receptor antagonist and D2 partial agonist
- GC14826Carmoxirole hydrochlorideCAS: 115092-85-8纯度: >98.00%
Carmoxirole hydrochloride (EMD 45609 hydrochloride) 是一种选择性的、外周作用的多巴胺 D2 受体激动剂,在体内表现出抗高血压活性。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC13156 | (+)-AJ 76 hydrochloride | 85379-09-5 | - | |
(+)-AJ 76 hydrochloride是一种对突触前受体具有优先作用的多巴胺受体(dopamine receptors, DRs)拮抗剂(hD3、hD4、hD2S、hD2L和rD2受体的pKi值分别为6.95、6.67、6.37、6.21和6.07)。 | ||||
| GC13169 | SKF 77434 hydrobromide | 300561-58-4 | - | |
A dopamine D 1 receptor partial agonist | ||||
| GC13183 | SB 277011A dihydrochloride | 1226917-67-4 | - | |
A selective dopamine D 3 antagonist | ||||
| GC13573 | Nomifensine | 32795-47-4 | >99.50% | |
An inhibitor of norepinephrine and dopamine reuptake | ||||
| GC13627 | Ziprasidone hydrochloride monohydrate | 138982-67-9 | >99.50% | |
An atypical antipsychotic | ||||
| GC13786 | (±)-Salsolinol (hydrochloride) | 79923-51-6 | >98.00% | |
A metabolite of ethanol that targets dopaminergic neurons | ||||
| GC13931 | Bromocriptine mesylate | 22260-51-1 | >99.00% / >98.00% | |
A dopamine receptor agonist | ||||
| GC14048 | SKF 38393 hydrobromide | 20012-10-6 | - | |
A partial agonist of dopamine D 1 -like receptors | ||||
| GC14160 | Blonanserin | 132810-10-7 | >98.50% | |
A dopamine and serotonin receptor antagonist | ||||
| GC14280 | PD 168568 dihydrochloride | 210688-56-5 | - | |
PD 168568 dihydrochloride 是一种具有口服活性的选择性 D4 多巴胺受体拮抗剂,Ki 为 8.8 nM。 | ||||
| GC14281 | L-DOPA methyl ester (hydrochloride) | 1421-65-4 | - | |
A dopamine precursor | ||||
| GC14311 | 4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride | 6109-35-9 | - | |
dopamine release inhibitor | ||||
| GC14491 | B-HT 920 | 36085-73-1 | >99.50% | |
A potent agonist of D 2 receptors | ||||
| GC14518 | Asenapine hydrochloride | 1412458-61-7 | >99.50% | |
Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。 | ||||
| GC14559 | Fluphenazine dihydrochloride | 146-56-5 | >99.00% | |
A dopamine D 1 and D 2 receptor antagonist | ||||
| GC14569 | L-745,870 trihydrochloride | 866021-03-6 | >98.00% | |
L-745,870 trihydrochloride 是一种有效的、选择性的、脑渗透性和口服活性的多巴胺 D4 受体拮抗剂,Ki 为 0.43 nM。 | ||||
| GC14593 | GSK 789472 hydrochloride | 1257326-24-1 | - | |
dopamine D3 receptor antagonist and D2 partial agonist | ||||
| GC14610 | A 412997 dihydrochloride | 1347744-96-0 | - | |
Selective D4 agonist | ||||
| GC14694 | NGD 94-1 | 178928-68-2 | >99.50% | |
High affinity D4 receptor ligand | ||||
| GC14714 | Bupropion hydrochloride | 31677-93-7 | >99.50% | |
An Analytical Reference Material | ||||
| GC14822 | Remoxipride hydrochloride | 73220-03-8 | - | |
An atypical antipsychotic | ||||
| GC14826 | Carmoxirole hydrochloride | 115092-85-8 | >98.00% | |
Carmoxirole hydrochloride (EMD 45609 hydrochloride) 是一种选择性的、外周作用的多巴胺 D2 受体激动剂,在体内表现出抗高血压活性。 | ||||
| GC14865 | RuBi-Dopa | - | - | |
dopamine receptor activator | ||||
| GC14873 | 2-CMDO | 24140-98-5 | - | |
Dopamine D2-like receptor antagonist | ||||
