Dopamine Receptor
Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Dopamine Receptor 相关产品(289)
- GC15326Flupenthixol dihydrochlorideCAS: 2413-38-9纯度: >98.00%
Flupentixol 是一种具有口服活性的 D1/D2 多巴胺受体拮抗剂和新型 PI3K 抑制剂(PI3Kα;IC50=127 nM)。
- GC156063α-Bis-(4-fluorophenyl) methoxytropane hydrochlorideCAS: 202646-03-5
dopamine uptake and transport inhibitor
- GC162676-Hydroxydopamine hydrobromideCAS: 636-00-0纯度: >98.00%
6-Hydroxydopamine hydrobromide (6-OHDA) 是儿茶酚胺、多巴胺和去甲肾上腺素的结构类似物,对儿茶酚胺能神经元发挥毒性作用。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15016 | SKF 83566 hydrobromide | 108179-91-5 | - | |
A dopamine D 1 receptor antagonist | ||||
| GC15107 | Clomipramine HCl | 17321-77-6 | >99.00% | |
A tricyclic antidepressant | ||||
| GC15326 | Flupenthixol dihydrochloride | 2413-38-9 | >98.00% | |
Flupentixol 是一种具有口服活性的 D1/D2 多巴胺受体拮抗剂和新型 PI3K 抑制剂(PI3Kα;IC50=127 nM)。 | ||||
| GC15463 | Iloperidone | 133454-47-4 | >99.50% | |
An atypical antipsychotic | ||||
| GC15498 | A 68930 hydrochloride | 130465-39-3 | - | |
A 68930 hydrochloride 作为多巴胺 D1 受体激动剂,可用于支气管扩张的研究。 | ||||
| GC15546 | Alizapride HCl | 59338-87-3 | >99.00% | |
A dopamine D 2 receptor antagonist | ||||
| GC15606 | 3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride | 202646-03-5 | - | |
dopamine uptake and transport inhibitor | ||||
| GC15619 | L-741,626 | 81226-60-0 | >99.00% / >98.00% | |
A dopamine D 2 receptor antagonist | ||||
| GC15754 | WAY-100635 Maleate | 1092679-51-0 | >99.00% | |
A serotonin 5-HT 1A antagonist | ||||
| GC15763 | PNU 177864 hydrochloride | 250266-51-4 | - | |
dopamine D3 receptor antagonist | ||||
| GC15792 | CY 208-243 | 100999-26-6 | >99.50% | |
CY 208-243 是一种选择性多巴胺 D1 受体激动剂,具有抗帕金森病活性。 | ||||
| GC15856 | 3'-Fluorobenzylspiperone maleate | 1135278-61-3 | - | |
ligand for the D2 receptor | ||||
| GC16017 | Rotigotine hydrochloride | 125572-93-2 | >99.00% | |
A non-selective dopamine receptor agonist | ||||
| GC16049 | AMI-193 | 510-74-7 | >98.50% | |
AMI-193 (AMI-193) 是一种有效的、选择性的 5-HT2 和多巴胺 D2 受体拮抗剂,Kis 分别为 2 nM 和 3 nM。 | ||||
| GC16229 | Azaperone | 1649-18-9 | >98.00% / >99.00% | |
An Analytical Reference Standard | ||||
| GC16267 | 6-Hydroxydopamine hydrobromide | 636-00-0 | >98.00% | |
6-Hydroxydopamine hydrobromide (6-OHDA) 是儿茶酚胺、多巴胺和去甲肾上腺素的结构类似物,对儿茶酚胺能神经元发挥毒性作用。 | ||||
| GC16270 | WAY-100635 maleate salt | 634908-75-1 | >98.00% | |
A serotonin 5-HT 1A antagonist | ||||
| GC16574 | 7-Hydroxy-DPAT hydrobromide | 76135-30-3 | - | |
A dopamine D 3 receptor agonist | ||||
| GC16686 | U 99194 maleate | 234757-41-6 | - | |
D3 antagonist | ||||
| GC16730 | Lisuride maleate | 19875-60-6 | >99.50% | |
New Product | ||||
| GC16769 | Raclopride | 84225-95-6 | >99.50% | |
Raclopride是一种取代的苯甲酰胺,是具有高选择性的多巴胺D 2 和D 3 受体拮抗剂。 | ||||
| GC16782 | Benocyclidine | 112726-66-6 | >98.00% | |
An Analytical Reference Standard | ||||
| GC16903 | GR 103691 | 162408-66-4 | >99.50% | |
A dopamine D 3 receptor antagonist | ||||
| GC16916 | 7-Hydroxy-PIPAT maleate | 159559-71-4 | - | |
D3 receptor agonist | ||||
