关于 "CYP3A/CYP450" 的结果18+ 个结果
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC35075 | 20-HETE | 79551-86-3 | Endogenous Metabolite | ||
A cytochrome P450 (CYP450) metabolite of arachidonic acid | |||||
| GC40440 | (±)8(9)-EET | - | PPAR | ||
A racemic version of a CYP450 metabolite of arachidonic acid | |||||
| GC19458 | 6β-hydroxy Testosterone | 62-99-7 | Androgen Receptor | ||
CYP3A metabolite of testosterone | |||||
| GC42888 | Azamulin | 76530-44-4 | P450 | ||
A selective CYP3A inhibitor | |||||
| GC14269 | Cobicistat (GS-9350) | 1004316-88-4 | HIV | ||
An inhibitor of CYP3A | |||||
| GC40528 | 11α-hydroxy Testosterone | 3066-12-4 | Androgen Receptor | ||
A CYP3A metabolite of testosterone | |||||
| GC13836 | 2,3-dihydrothieno-Thiadiazole Carboxylate | 152467-47-5 | P450 | ||
Selective CYP450 inhibitor | |||||
| GC16575 | Alizarin | 72-48-0 | P450 | ||
A CYP450 inhibitor | |||||
| GC49030 | 7-Ethoxycoumarin | 31005-02-4 | Enzyme Substrates | ||
A CYP450 substrate | |||||
| GC52062 | 7-Benzyloxy-4-(trifluoromethyl)coumarin | 220001-53-6 | P450 | ||
A fluorogenic substrate for CYP1A2 and CYP3A | |||||
| GC16259 | SKF 525A (hydrochloride) | 62-68-0 | P450 | ||
A nonspecific CYP450 inhibitor | |||||
| GC10554 | 3-Cyano-7-ethoxycoumarin | 117620-77-6 | CYP3A/CYP450 | ||
A fluorogenic CYP450 substrate | |||||
| GC42605 | 7-ethoxy-4-Methylcoumarin | 87-05-8 | - | ||
A fluorescent CYP450 substrate | |||||
| GC41945 | 16-hydroxy Hexadecanoic Acid | 506-13-8 | P450 | ||
CYP450 metabolite of palmitic acid | |||||
| GC40272 | (±)8(9)-DiHET | 192461-96-4 | Cyclooxygenase | ||
A CYP450 metabolite of arachidonic acid | |||||
| GC40705 | CAY10668 | - | - | ||
A potential inhibitor of CYP450 1B1 | |||||
| GC42083 | 20-HETE Ethanolamide | 942069-11-6 | Endocannabinoid/Endocannabinoid-like | ||
A putative CYP450 metabolite of AEA | |||||
| GC44299 | N-Acetyl-4-benzoquinone imine | 50700-49-7 | Drug Metabolite | ||
A reactive CYP450 metabolite of acetaminophen | |||||
