关于 "TRP Channel" 的结果35+ 个结果
- (Trp⁶³,Trp⁶⁴)-C3a (63-77)CAS: 130154-64-2
(Trp?³,Trp??)-C3a (63-77), synthetic superagonist analog of complement 3a, exhibited the greatest biological potency of all peptides tested. The peptide was 12-15 times more active than natural C3a. Such an optimal potency was obtained by introducing a bulky hydrophobic group such as Trp-Trp which binds more strongly to the hydrophobic site on the receptor than does the corresponding site on the natural ligand.
- WRW4 (trifluoroacetate salt)
WRW4 (trifluoroacetate salt)是一种选择性的甲酰肽受体2（FPR2，曾称FPRL1）拮抗剂，为人工合成的C端酰胺化六肽，抑制WKYMVm与FPRL2结合的IC 50 值为0.23μM。
- (Trp?)-KemptideCAS: 80224-16-4
Chocktide ((Trp?)-Kemptide) is readily phosphorylated by cAMP-dependent protein kinase.
- (Trp¹¹)-NeurotensinCAS: 75644-95-0
This neurotensin analog, in which Tyr¹¹ is substituted by Trp, was found to be as potent as neurotensin in both binding and biological assays in the rat. In contrast, this analog was about 10 times less potent than neurotensin in the guinea-pig.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GA22955 | H-Trp-Trp-OH | 20696-60-0 | - | ||
| GC18268 | Cyclo(L-Trp-L-Trp) | 20829-55-4 | Bacterial Diseases | ||
A cyclic dipeptide | |||||
| GA20317 | (Trp⁶³,Trp⁶⁴)-C3a (63-77) | 130154-64-2 | - | ||
(Trp?³,Trp??)-C3a (63-77), synthetic superagonist analog of complement 3a, exhibited the greatest biological potency of all peptides tested. The peptide was 12-15 times more active than natural C3a. Such an optimal potency was obtained by introducing a bulky hydrophobic group such as Trp-Trp which binds more strongly to the hydrophobic site on the receptor than does the corresponding site on the natural ligand. | |||||
| GC52457 | WRW4 (trifluoroacetate salt) | - | Pulmonary Diseases | ||
WRW4 (trifluoroacetate salt)是一种选择性的甲酰肽受体2（FPR2，曾称FPRL1）拮抗剂，为人工合成的C端酰胺化六肽，抑制WKYMVm与FPRL2结合的IC50值为0.23μM。 | |||||
| GC52388 | [D-Lys3]-GHRP-6 (trifluoroacetate salt) | - | Endocrinology and Hormones | ||
An antagonist of GHS-R1a | |||||
| GA24052 | (Trp?)-Kemptide | 80224-16-4 | Peptides | ||
Chocktide ((Trp?)-Kemptide) is readily phosphorylated by cAMP-dependent protein kinase. | |||||
| GA20314 | (Trp¹¹)-Neurotensin | 75644-95-0 | - | ||
This neurotensin analog, in which Tyr¹¹ is substituted by Trp, was found to be as potent as neurotensin in both binding and biological assays in the rat. In contrast, this analog was about 10 times less potent than neurotensin in the guinea-pig. | |||||
| GA20316 | (Trp⁶)-LHRH | 156126-74-8 | - | ||
| GC78592 | F4-Trp | 72120-72-0 | - | ||
F4-Trp (4,5,6,7-Tetrafluoro-L-tryptophan) 是一种靶向 α3β4 型烟碱型乙酰胆碱受体 (α3β4nAChR) 的配体。 | |||||
| GA10571 | Fmoc-Trp-ol | 153815-60-2 | Fmoc-Amino Acids and Derivatives | ||
Fmoc-Trp-ol | |||||
| GB57441 | Boc-Trp-OBzl | 57229-67-1 | - | ||