关于 "LPL Receptor" 的结果28+ 个结果
- Galanin Receptor Ligand M35CAS: 142846-71-7
Galanin Receptor Ligand M35 是一种高亲和力的甘丙肽受体配体，在大鼠脊髓、大鼠海马和离体小鼠胰岛中起着甘丙肽受体拮抗剂的作用。Galanin Receptor Ligand M35 对人 GalR1 和 GalR2 的 Ki 值分别为 0.11 nM、2.0 nM。
- A2A receptor antagonist 1CAS: 443103-97-7
A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。
- GABAA receptor agent 1CAS: 1571-87-5
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity.
- Thrombin Receptor AntagonistCAS: 207553-92-2
The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor. MSRPACPNDKYE has served as model peptide in protein modification and MS studies.
- cFMS Receptor Inhibitor IVCAS: 959626-45-0
cFMS Receptor Inhibitor IV (Compound 42) 是一种有效的 cFMS 抑制剂，IC50 为 0.017 μM。
- A2B receptor antagonist 1CAS: 531506-36-2
A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。
- S1p receptor agonist 1CAS: 1514888-56-2
S1p receptor agonist 1 是一种有效且具有口服活性的 S1P 受体激动剂，具有诱导 S1P1 内化的活性 (EC50=9.83 nM)。
- Androgen receptor antagonist 1CAS: 1338812-36-4
Androgenreceptorantagonist1是一种口服有效的完整雄激素受体(AR)拮抗剂，IC50为59nM。Androgenreceptorantagonist1可用于合成PROTACAR降解剂，1μM和10μMPROTACAR降解剂作用于LNCaP细胞，分别导致24%和47%AR蛋白降解。
- AMPA receptor modulator-8CAS: 2034182-75-5
AMPA receptormodulator-8 (Example 270) 是一种AMPA receptor调节剂，对 TARP-γ2 的IC50为 0.02 nM。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GP21888 | LPL Human | - | Lipase | ||
Lipoprotein Lipase Human Recombinant | |||||
| GP21889 | LPL Human, HEK | - | Lipase | ||
Lipoprotein Lipase Human Recombinant, HEK | |||||
| GC36102 | Galanin Receptor Ligand M35 | 142846-71-7 | Peptides | ||
Galanin Receptor Ligand M35 是一种高亲和力的甘丙肽受体配体，在大鼠脊髓、大鼠海马和离体小鼠胰岛中起着甘丙肽受体拮抗剂的作用。Galanin Receptor Ligand M35 对人 GalR1 和 GalR2 的 Ki 值分别为 0.11 nM、2.0 nM。 | |||||
| GC11275 | C34 | 40592-88-9 | HSC | ||
C34是一种可口服的Toll样受体4(TLR4)选择性拮抗剂，C34通过抑制TLR4/MyD88/NF-κB信号通路，减少促炎细胞因子的产生，从而发挥抗炎作用。 | |||||
| GC43083 | C3a Receptor Agonist | 944997-60-8 | Neuroscience | ||
C3a Receptor Agonist是一种选择性的补体3a受体（C3aR）特异性激动剂。 | |||||
| GC16363 | TGR5 Receptor Agonist | 1197300-24-5 | GPCR19 | ||
A TGR5 agonist | |||||
| GP20716 | Leptin Receptor Human | - | Leptin | ||
Leptin Binding Domain Human Recombinant | |||||
| GP20717 | Leptin Receptor Chicken | - | Leptin | ||
Leptin Receptor Chicken Recombinant | |||||
| GP20896 | sRANK Receptor Human | - | RANK Ligand | ||
Soluble RANK Receptor Human Recombinant | |||||
| GC32019 | Interferon receptor agonist | 2215120-36-6 | IFNAR | ||
干扰素受体激动剂（化合物 6）是一种干扰素 (IFN) 受体诱导剂。 | |||||
| GC30918 | A2A receptor antagonist 1 | 443103-97-7 | Adenosine Receptor | ||
A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。 | |||||
| GC60862 | GABAA receptor agent 1 | 1571-87-5 | GABA Receptor | ||
GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity. | |||||
| GA23607 | Thrombin Receptor Antagonist | 207553-92-2 | - | ||
The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor.
MSRPACPNDKYE has served as model peptide in protein modification and MS studies. | |||||
| GC19170 | Glucagon receptor antagonists-4 | 1393124-08-7 | Glucagon Receptor | ||
A GCGR antagonist | |||||
| GC65976 | cFMS Receptor Inhibitor IV | 959626-45-0 | c-FMS | ||
cFMS Receptor Inhibitor IV (Compound 42) 是一种有效的 cFMS 抑制剂，IC50 为 0.017 μM。 | |||||
| GC19272 | Orexin 2 Receptor Agonist | 1796565-52-0 | OX Receptor | ||
An orexin 2 receptor agonist | |||||
| GC39554 | AT2 receptor agonist C21 | 477775-14-7 | Cardiomyopathy | ||
An AT2 receptor agonist | |||||
| GC31974 | A2B receptor antagonist 1 | 531506-36-2 | Adenosine Receptor | ||
A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。 | |||||
| GC30759 | H3 receptor-MO-1 | 1240914-03-7 | Histamine Receptor | ||
H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。 | |||||
| GC31310 | H3 receptor antagonist 1 | 935840-13-4 | Histamine Receptor | ||
H3receptorantagonist1是组胺H3(histamineH3)受体拮抗剂，可用于神经疾病的研究。 | |||||
| GC19316 | S1p receptor agonist 1 | 1514888-56-2 | LPL Receptor | ||
S1p receptor agonist 1 是一种有效且具有口服活性的 S1P 受体激动剂，具有诱导 S1P1 内化的活性 (EC50=9.83 nM)。 | |||||
| GC60582 | Androgen receptor antagonist 1 | 1338812-36-4 | - | ||
Androgenreceptorantagonist1是一种口服有效的完整雄激素受体(AR)拮抗剂，IC50为59nM。Androgenreceptorantagonist1可用于合成PROTACAR降解剂，1μM和10μMPROTACAR降解剂作用于LNCaP细胞，分别导致24%和47%AR蛋白降解。 | |||||
| GC11399 | Glucocorticoid receptor agonist | 1245526-82-2 | Glucocorticoid Receptor | ||
糖皮质激素受体激动剂是一种有效的糖皮质激素受体激动剂。 | |||||
| GC78467 | AMPA receptor modulator-8 | 2034182-75-5 | - | ||
AMPA receptormodulator-8 (Example 270) 是一种AMPA receptor调节剂，对 TARP-γ2 的IC50为 0.02 nM。 | |||||